MXPA03001512A - Pirrolilamidas biciclicas como inhibidores de glucogeno fosforilasa. - Google Patents

Pirrolilamidas biciclicas como inhibidores de glucogeno fosforilasa.

Info

Publication number
MXPA03001512A
MXPA03001512A MXPA03001512A MXPA03001512A MXPA03001512A MX PA03001512 A MXPA03001512 A MX PA03001512A MX PA03001512 A MXPA03001512 A MX PA03001512A MX PA03001512 A MXPA03001512 A MX PA03001512A MX PA03001512 A MXPA03001512 A MX PA03001512A
Authority
MX
Mexico
Prior art keywords
phosphorylase inhibitors
glucogen
amides
amide derivatives
bicyclic
Prior art date
Application number
MXPA03001512A
Other languages
English (en)
Inventor
Julie B Bartlett
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of MXPA03001512A publication Critical patent/MXPA03001512A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pyrrole Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Enzymes And Modification Thereof (AREA)
MXPA03001512A 2000-09-06 2001-08-31 Pirrolilamidas biciclicas como inhibidores de glucogeno fosforilasa. MXPA03001512A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0021831.3A GB0021831D0 (en) 2000-09-06 2000-09-06 Chemical compounds
PCT/SE2001/001880 WO2002020530A1 (en) 2000-09-06 2001-08-31 Bicyclic pyrrolyl amides as glucogen phosphorylase inhibitors

Publications (1)

Publication Number Publication Date
MXPA03001512A true MXPA03001512A (es) 2003-06-09

Family

ID=9898927

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA03001512A MXPA03001512A (es) 2000-09-06 2001-08-31 Pirrolilamidas biciclicas como inhibidores de glucogeno fosforilasa.

Country Status (31)

Country Link
US (1) US20030232875A1 (es)
EP (1) EP1317459B1 (es)
JP (1) JP2004508376A (es)
KR (1) KR100802369B1 (es)
CN (2) CN1896078A (es)
AT (1) ATE263772T1 (es)
AU (2) AU2001282833B2 (es)
BG (1) BG107624A (es)
BR (1) BR0113606A (es)
CA (1) CA2417594A1 (es)
CZ (1) CZ2003616A3 (es)
DE (1) DE60102710T2 (es)
DK (1) DK1317459T3 (es)
EE (1) EE200300083A (es)
ES (1) ES2217183T3 (es)
GB (1) GB0021831D0 (es)
HK (1) HK1055299A1 (es)
HU (1) HUP0400784A3 (es)
IL (1) IL154291A0 (es)
IS (1) IS2110B (es)
MX (1) MXPA03001512A (es)
NO (1) NO20031024L (es)
NZ (1) NZ524011A (es)
PL (1) PL361024A1 (es)
PT (1) PT1317459E (es)
RU (1) RU2003104013A (es)
SK (1) SK2592003A3 (es)
TR (1) TR200401659T4 (es)
UA (1) UA73781C2 (es)
WO (1) WO2002020530A1 (es)
ZA (1) ZA200301013B (es)

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DE10225635C1 (de) * 2002-06-07 2003-12-24 Aventis Pharma Gmbh N-Benzoylureido-Zimtsäurederivate, Verfahren zu deren Herstellung und deren Verwendung
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WO2005020985A1 (en) * 2003-08-29 2005-03-10 Astrazeneca Ab Indolamide derivatives which possess glycogen phosphorylase inhibitory activity
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Also Published As

Publication number Publication date
KR100802369B1 (ko) 2008-02-14
ZA200301013B (en) 2004-05-05
GB0021831D0 (en) 2000-10-18
CN1896078A (zh) 2007-01-17
PT1317459E (pt) 2004-08-31
JP2004508376A (ja) 2004-03-18
IL154291A0 (en) 2003-09-17
CA2417594A1 (en) 2002-03-14
HUP0400784A2 (hu) 2004-07-28
EP1317459B1 (en) 2004-04-07
TR200401659T4 (tr) 2004-09-21
RU2003104013A (ru) 2004-08-20
HUP0400784A3 (en) 2007-09-28
SK2592003A3 (en) 2003-08-05
NO20031024D0 (no) 2003-03-05
BG107624A (bg) 2004-01-30
ES2217183T3 (es) 2004-11-01
IS6727A (is) 2003-02-24
NZ524011A (en) 2004-08-27
CN1473163A (zh) 2004-02-04
ATE263772T1 (de) 2004-04-15
EE200300083A (et) 2004-12-15
PL361024A1 (en) 2004-09-20
EP1317459A1 (en) 2003-06-11
US20030232875A1 (en) 2003-12-18
IS2110B (is) 2006-05-15
DE60102710T2 (de) 2005-04-14
BR0113606A (pt) 2003-06-24
AU2001282833B2 (en) 2006-07-06
WO2002020530A1 (en) 2002-03-14
NO20031024L (no) 2003-03-05
AU8283301A (en) 2002-03-22
CZ2003616A3 (cs) 2003-05-14
HK1055299A1 (en) 2004-01-02
DE60102710D1 (de) 2004-05-13
UA73781C2 (en) 2005-09-15
KR20030025305A (ko) 2003-03-28
CN1264846C (zh) 2006-07-19
DK1317459T3 (da) 2004-07-12

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