IL154291A0 - Bicyclic pyrrolyl amides as glucogen phosphorylase inhibitors - Google Patents

Bicyclic pyrrolyl amides as glucogen phosphorylase inhibitors

Info

Publication number
IL154291A0
IL154291A0 IL15429101A IL15429101A IL154291A0 IL 154291 A0 IL154291 A0 IL 154291A0 IL 15429101 A IL15429101 A IL 15429101A IL 15429101 A IL15429101 A IL 15429101A IL 154291 A0 IL154291 A0 IL 154291A0
Authority
IL
Israel
Prior art keywords
phosphorylase inhibitors
glucogen
amides
amide derivatives
bicyclic
Prior art date
Application number
IL15429101A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of IL154291A0 publication Critical patent/IL154291A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL15429101A 2000-09-06 2001-08-31 Bicyclic pyrrolyl amides as glucogen phosphorylase inhibitors IL154291A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0021831.3A GB0021831D0 (en) 2000-09-06 2000-09-06 Chemical compounds
PCT/SE2001/001880 WO2002020530A1 (en) 2000-09-06 2001-08-31 Bicyclic pyrrolyl amides as glucogen phosphorylase inhibitors

Publications (1)

Publication Number Publication Date
IL154291A0 true IL154291A0 (en) 2003-09-17

Family

ID=9898927

Family Applications (1)

Application Number Title Priority Date Filing Date
IL15429101A IL154291A0 (en) 2000-09-06 2001-08-31 Bicyclic pyrrolyl amides as glucogen phosphorylase inhibitors

Country Status (31)

Country Link
US (1) US20030232875A1 (xx)
EP (1) EP1317459B1 (xx)
JP (1) JP2004508376A (xx)
KR (1) KR100802369B1 (xx)
CN (2) CN1264846C (xx)
AT (1) ATE263772T1 (xx)
AU (2) AU8283301A (xx)
BG (1) BG107624A (xx)
BR (1) BR0113606A (xx)
CA (1) CA2417594A1 (xx)
CZ (1) CZ2003616A3 (xx)
DE (1) DE60102710T2 (xx)
DK (1) DK1317459T3 (xx)
EE (1) EE200300083A (xx)
ES (1) ES2217183T3 (xx)
GB (1) GB0021831D0 (xx)
HK (1) HK1055299A1 (xx)
HU (1) HUP0400784A3 (xx)
IL (1) IL154291A0 (xx)
IS (1) IS2110B (xx)
MX (1) MXPA03001512A (xx)
NO (1) NO20031024L (xx)
NZ (1) NZ524011A (xx)
PL (1) PL361024A1 (xx)
PT (1) PT1317459E (xx)
RU (1) RU2003104013A (xx)
SK (1) SK2592003A3 (xx)
TR (1) TR200401659T4 (xx)
UA (1) UA73781C2 (xx)
WO (1) WO2002020530A1 (xx)
ZA (1) ZA200301013B (xx)

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DE10215907A1 (de) * 2002-04-11 2003-11-06 Aventis Pharma Gmbh Acyl-4-carboxyphenyl-harnstoffderivate, Verfahren zu deren Herstellung und deren Verwendung
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DE10225635C1 (de) * 2002-06-07 2003-12-24 Aventis Pharma Gmbh N-Benzoylureido-Zimtsäurederivate, Verfahren zu deren Herstellung und deren Verwendung
DK1375477T3 (da) * 2002-06-17 2010-01-25 Saltigo Gmbh Fremgangsmåde til fremstilling af mono-N-sulfonylerede diaminer
WO2004007437A1 (de) * 2002-07-11 2004-01-22 Aventis Pharma Deutschland Gmbh Harnstoff- und urethan-substituierte acylharnstoffe, verfahren zu deren herstellung und deren verwendung als arzneimittel
US7186735B2 (en) 2002-08-07 2007-03-06 Sanofi-Aventis Deutschland Gmbh Acylated arylcycloalkylamines and their use as pharmaceuticals
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GB0318464D0 (en) * 2003-08-07 2003-09-10 Astrazeneca Ab Chemical compounds
GB0318463D0 (en) * 2003-08-07 2003-09-10 Astrazeneca Ab Chemical compounds
GB0319759D0 (en) * 2003-08-22 2003-09-24 Astrazeneca Ab Chemical compounds
GB0319690D0 (en) * 2003-08-22 2003-09-24 Astrazeneca Ab Chemical compounds
WO2005020986A1 (en) * 2003-08-29 2005-03-10 Astrazeneca Ab Heterocyclic amide derivatives which posses glycogen phosphorylase inhibitory activity
WO2005020985A1 (en) * 2003-08-29 2005-03-10 Astrazeneca Ab Indolamide derivatives which possess glycogen phosphorylase inhibitory activity
GB0320422D0 (en) * 2003-08-30 2003-10-01 Astrazeneca Ab Chemical compounds
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JP5432526B2 (ja) 2006-01-06 2014-03-05 サノビオン ファーマシューティカルズ インク モノアミン再取り込み阻害剤としてのシクロアルキルアミン
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Also Published As

Publication number Publication date
KR20030025305A (ko) 2003-03-28
SK2592003A3 (en) 2003-08-05
HK1055299A1 (en) 2004-01-02
HUP0400784A2 (hu) 2004-07-28
CA2417594A1 (en) 2002-03-14
CZ2003616A3 (cs) 2003-05-14
RU2003104013A (ru) 2004-08-20
MXPA03001512A (es) 2003-06-09
CN1264846C (zh) 2006-07-19
UA73781C2 (en) 2005-09-15
AU2001282833B2 (en) 2006-07-06
PL361024A1 (en) 2004-09-20
JP2004508376A (ja) 2004-03-18
EE200300083A (et) 2004-12-15
GB0021831D0 (en) 2000-10-18
EP1317459A1 (en) 2003-06-11
NO20031024D0 (no) 2003-03-05
NO20031024L (no) 2003-03-05
IS6727A (is) 2003-02-24
CN1896078A (zh) 2007-01-17
AU8283301A (en) 2002-03-22
HUP0400784A3 (en) 2007-09-28
NZ524011A (en) 2004-08-27
DE60102710D1 (de) 2004-05-13
ES2217183T3 (es) 2004-11-01
TR200401659T4 (tr) 2004-09-21
BG107624A (bg) 2004-01-30
US20030232875A1 (en) 2003-12-18
BR0113606A (pt) 2003-06-24
DE60102710T2 (de) 2005-04-14
IS2110B (is) 2006-05-15
ZA200301013B (en) 2004-05-05
CN1473163A (zh) 2004-02-04
WO2002020530A1 (en) 2002-03-14
KR100802369B1 (ko) 2008-02-14
EP1317459B1 (en) 2004-04-07
ATE263772T1 (de) 2004-04-15
DK1317459T3 (da) 2004-07-12
PT1317459E (pt) 2004-08-31

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