AU684255B2 - Arylsulfonamido-substituted hydroxamic acids - Google Patents

Arylsulfonamido-substituted hydroxamic acids Download PDF

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AU684255B2
AU684255B2 AU52655/93A AU5265593A AU684255B2 AU 684255 B2 AU684255 B2 AU 684255B2 AU 52655/93 A AU52655/93 A AU 52655/93A AU 5265593 A AU5265593 A AU 5265593A AU 684255 B2 AU684255 B2 AU 684255B2
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lower alkyl
alkyl
amino
alkoxy
phenyl
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AU5265593A (en
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Lawrence J Macpherson
David Thomas Parker
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Novartis AG
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Ciba Geigy AG
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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/42—Radicals substituted by singly-bound nitrogen atoms having hetero atoms attached to the substituent nitrogen atom
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
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    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
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    • C07C311/19—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom to an acyclic carbon atom of a hydrocarbon radical substituted by carboxyl groups
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    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
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NO940038D0 (no) 1994-01-05
ZA9448B (en) 1994-08-11
MX9400276A (es) 1994-07-29
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CA2112779A1 (en) 1994-07-07
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JP2951527B2 (ja) 1999-09-20
GR3025611T3 (en) 1998-03-31
TW247313B (cg-RX-API-DMAC7.html) 1995-05-11
IL108229A0 (en) 1994-04-12
NO940038L (cg-RX-API-DMAC7.html) 1994-07-07
AU5265593A (en) 1995-05-04
NO180583B (no) 1997-02-03
HK1002633A1 (en) 1998-09-04
DK0606046T3 (da) 1998-05-04
BR1100131A (pt) 2000-03-14
KR940018360A (ko) 1994-08-16
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EP0606046B1 (en) 1997-10-08
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