AU2016355710B2 - Modulators of ROR-gamma - Google Patents

Modulators of ROR-gamma Download PDF

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Publication number
AU2016355710B2
AU2016355710B2 AU2016355710A AU2016355710A AU2016355710B2 AU 2016355710 B2 AU2016355710 B2 AU 2016355710B2 AU 2016355710 A AU2016355710 A AU 2016355710A AU 2016355710 A AU2016355710 A AU 2016355710A AU 2016355710 B2 AU2016355710 B2 AU 2016355710B2
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Australia
Prior art keywords
ethylsulfonyl
carboxamide
benzyl
trifluoromethyl
methyl
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Ceased
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AU2016355710A
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AU2016355710A1 (en
Inventor
David A. Claremon
Lawrence Wayne Dillard
Yi Fan
Lanqi Jia
Suresh B. Singh
Colin M. Tice
Zhenrong Xu
Jing Yuan
Linghang Zhuang
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Vitae Pharmaceuticals LLC
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Vitae Pharmaceuticals LLC
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Assigned to VITAE PHARMACEUTICALS, LLC reassignment VITAE PHARMACEUTICALS, LLC Alteration of Name(s) of Applicant(s) under S113 Assignors: VITAE PHARMACEUTICALS, INC.
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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AU2016355710A 2015-11-20 2016-11-17 Modulators of ROR-gamma Ceased AU2016355710B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201562257964P 2015-11-20 2015-11-20
US62/257,964 2015-11-20
US201662320805P 2016-04-11 2016-04-11
US62/320,805 2016-04-11
PCT/US2016/062422 WO2017087608A1 (en) 2015-11-20 2016-11-17 Modulators of ror-gamma

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AU2016355710A1 AU2016355710A1 (en) 2018-05-31
AU2016355710B2 true AU2016355710B2 (en) 2021-03-25

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US (1) US11008340B2 (https=)
EP (2) EP3377482B1 (https=)
JP (1) JP6914257B2 (https=)
KR (1) KR20180086221A (https=)
CN (1) CN108463458B (https=)
AU (1) AU2016355710B2 (https=)
BR (1) BR112018010018A2 (https=)
CA (1) CA3005658A1 (https=)
IL (2) IL259421B (https=)
MA (1) MA53943A (https=)
MX (2) MX385332B (https=)
RU (1) RU2018121946A (https=)
SA (1) SA518391624B1 (https=)
WO (1) WO2017087608A1 (https=)

Families Citing this family (26)

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Publication number Priority date Publication date Assignee Title
AU2015210833B2 (en) 2014-02-03 2019-01-03 Vitae Pharmaceuticals, Llc Dihydropyrrolopyridine inhibitors of ROR-gamma
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