DK1194425T3 - Substituerede benzimidazoler - Google Patents

Substituerede benzimidazoler

Info

Publication number
DK1194425T3
DK1194425T3 DK00938780T DK00938780T DK1194425T3 DK 1194425 T3 DK1194425 T3 DK 1194425T3 DK 00938780 T DK00938780 T DK 00938780T DK 00938780 T DK00938780 T DK 00938780T DK 1194425 T3 DK1194425 T3 DK 1194425T3
Authority
DK
Denmark
Prior art keywords
substituted benzimidazoles
nfkappab
prophylaxis
pharmaceuticals
disorders
Prior art date
Application number
DK00938780T
Other languages
English (en)
Inventor
Hans Ulrich Stilz
Armin Walser
Bernhard Neises
William Jerome Bock Jr
Gary A Flynn
Joerg Habermann
Gerhard Jahne
Olaf Ritzeler
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE1999128424 external-priority patent/DE19928424A1/de
Priority claimed from DE2000106297 external-priority patent/DE10006297A1/de
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Application granted granted Critical
Publication of DK1194425T3 publication Critical patent/DK1194425T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
DK00938780T 1999-06-23 2000-06-09 Substituerede benzimidazoler DK1194425T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE1999128424 DE19928424A1 (de) 1999-06-23 1999-06-23 Substituierte Benzimidazole
DE2000106297 DE10006297A1 (de) 2000-02-12 2000-02-12 Substituierte Benzimidazole

Publications (1)

Publication Number Publication Date
DK1194425T3 true DK1194425T3 (da) 2005-11-21

Family

ID=26004312

Family Applications (1)

Application Number Title Priority Date Filing Date
DK00938780T DK1194425T3 (da) 1999-06-23 2000-06-09 Substituerede benzimidazoler

Country Status (29)

Country Link
US (1) US6358978B1 (da)
EP (1) EP1194425B1 (da)
JP (1) JP4763949B2 (da)
KR (1) KR100718830B1 (da)
CN (1) CN1168727C (da)
AT (1) ATE301651T1 (da)
AU (1) AU769350B2 (da)
BR (1) BR0012450B1 (da)
CA (1) CA2377085C (da)
CZ (1) CZ302775B6 (da)
DE (1) DE50010931D1 (da)
DK (1) DK1194425T3 (da)
EE (1) EE04813B1 (da)
ES (1) ES2246240T3 (da)
HK (1) HK1047582B (da)
HR (1) HRP20010944B1 (da)
HU (1) HU228466B1 (da)
IL (1) IL147184A0 (da)
ME (1) MEP56108A (da)
MX (1) MXPA01012283A (da)
NO (1) NO323597B1 (da)
NZ (1) NZ516348A (da)
PL (1) PL206826B1 (da)
PT (1) PT1194425E (da)
RS (1) RS50340B (da)
RU (1) RU2261248C2 (da)
SI (1) SI1194425T1 (da)
SK (1) SK286857B6 (da)
WO (1) WO2001000610A1 (da)

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