ATE263163T1 - Krytallinischer fungizider polymorph - Google Patents

Krytallinischer fungizider polymorph

Info

Publication number
ATE263163T1
ATE263163T1 AT98951994T AT98951994T ATE263163T1 AT E263163 T1 ATE263163 T1 AT E263163T1 AT 98951994 T AT98951994 T AT 98951994T AT 98951994 T AT98951994 T AT 98951994T AT E263163 T1 ATE263163 T1 AT E263163T1
Authority
AT
Austria
Prior art keywords
polymorphous
fungicidal
crystalline
fungicidal polymorphous
crystalline fungicidal
Prior art date
Application number
AT98951994T
Other languages
German (de)
English (en)
Inventor
David R Andrews
William Leong
Anantha R Sudhakar
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Application granted granted Critical
Publication of ATE263163T1 publication Critical patent/ATE263163T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
AT98951994T 1997-10-07 1998-10-05 Krytallinischer fungizider polymorph ATE263163T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US94618397A 1997-10-07 1997-10-07
PCT/US1998/020476 WO1999018097A1 (en) 1997-10-07 1998-10-05 Crystalline antifungal polymorph

Publications (1)

Publication Number Publication Date
ATE263163T1 true ATE263163T1 (de) 2004-04-15

Family

ID=25484068

Family Applications (1)

Application Number Title Priority Date Filing Date
AT98951994T ATE263163T1 (de) 1997-10-07 1998-10-05 Krytallinischer fungizider polymorph

Country Status (30)

Country Link
EP (1) EP1021439B1 (OSRAM)
JP (4) JP2001519346A (OSRAM)
KR (1) KR100626109B1 (OSRAM)
CN (1) CN1125067C (OSRAM)
AR (1) AR015947A1 (OSRAM)
AT (1) ATE263163T1 (OSRAM)
AU (1) AU759982B2 (OSRAM)
BR (1) BR9812866A (OSRAM)
CA (1) CA2305803C (OSRAM)
CO (1) CO4970829A1 (OSRAM)
CZ (1) CZ299835B6 (OSRAM)
DE (1) DE69822859T2 (OSRAM)
DK (1) DK1021439T3 (OSRAM)
ES (1) ES2217594T3 (OSRAM)
HU (1) HU225233B1 (OSRAM)
ID (1) ID29290A (OSRAM)
IL (1) IL135331A (OSRAM)
IN (1) IN1998CH02232A (OSRAM)
MX (1) MX225999B (OSRAM)
MY (1) MY130126A (OSRAM)
NO (1) NO318827B1 (OSRAM)
NZ (1) NZ503662A (OSRAM)
PE (1) PE120499A1 (OSRAM)
PH (1) PH11998002606B1 (OSRAM)
PL (1) PL189317B1 (OSRAM)
PT (1) PT1021439E (OSRAM)
SK (1) SK285190B6 (OSRAM)
TW (1) TW589310B (OSRAM)
WO (1) WO1999018097A1 (OSRAM)
ZA (1) ZA989063B (OSRAM)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2130540A1 (en) * 2008-06-02 2009-12-09 Sandoz AG Pharmaceutical compositions containing a crystalline form of posaconazole
EP2141159A1 (en) 2008-07-03 2010-01-06 Sandoz AG A Crystalline form of posaconazole
CA2767489A1 (en) 2009-07-09 2011-01-13 Sandoz Ag A crystalline form of posaconazole
WO2011144656A1 (en) 2010-05-19 2011-11-24 Sandoz Ag Preparation of posaconazole intermediates
MX2012013331A (es) 2010-05-19 2013-02-01 Sandoz Ag Purificacion de posaconazol y de intermediarios de posaconazol.
CN102892750B (zh) 2010-05-19 2016-03-02 桑多斯股份公司 制备手性酰肼的方法
AU2011254654B2 (en) * 2010-05-19 2016-01-07 Sandoz Ag Process for the preparation of chiral triazolones
CN108329303A (zh) 2011-06-16 2018-07-27 桑多斯股份公司 制备手性化合物的方法
WO2013042138A2 (en) 2011-09-19 2013-03-28 Msn Laboratories Limited Process for the preparation of triazole antifungal drug, its intermediates and polymorphs thereof
EP3024828B1 (en) * 2013-07-25 2017-05-17 Sandoz AG Improved process for the preparation of crystalline form iv of posaconazole
ITMI20132118A1 (it) * 2013-12-18 2015-06-19 Djada Pharmaceutical Sa Una forma cristallina di posaconazolo
ITMI20132115A1 (it) * 2013-12-18 2015-06-19 Djada Pharmaceutical Sa Una forma cristallina di posaconazolo
ITMI20132117A1 (it) * 2013-12-18 2015-06-19 Djada Pharmaceutical Sa Una forma cristallina di posaconazolo
ITMI20132114A1 (it) 2013-12-18 2015-06-19 Djada Pharmaceutical Sa Una forma cristallina di posaconazolo
CN111825717A (zh) 2014-10-21 2020-10-27 阿瑞雅德制药公司 5-氯-n4-[2-(二甲基磷酰基)苯基]-n2-{2-甲氧基-4-[4-(4-甲基哌嗪-1-基)哌啶-1-基]苯基}嘧啶-2,4-二胺的晶形
CN104387374A (zh) * 2014-10-21 2015-03-04 江苏恒盛药业有限公司 泊沙康唑晶型i的制备工艺
CN104370894A (zh) * 2014-10-21 2015-02-25 江苏恒盛药业有限公司 无定型泊沙康唑的制备工艺
PL3331501T3 (pl) 2015-08-08 2020-03-31 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Preparat o zwiększonej odporności na warunki przewodu pokarmowego zawierający pozakonazol
HK1256362A1 (zh) 2015-12-24 2019-09-20 Takeda Pharmaceutical Company Limited 共晶、其制造方法及含有共晶的药物
EP3210599B1 (en) 2016-02-26 2024-08-28 Alfred E. Tiefenbacher (GmbH & Co. KG) Gastro-resistant formulation containing posaconazole and a polymeric precipitation inhibitor
CN105949278B (zh) * 2016-03-30 2019-12-06 南京曼杰生物科技有限公司 一种取代的四氢呋喃水溶性衍生物及其应用
WO2017032908A1 (en) 2016-07-08 2017-03-02 Synthon B.V. Pharmaceutical composition comprising amorphous posaconazole
TR201620462A2 (tr) 2016-12-31 2018-07-23 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi POSAKONAZOL İÇEREN FARMASÖTİK BİLEŞİMLER ve ÜRETİM YÖNTEMİ
TR201722493A2 (tr) 2017-12-28 2019-07-22 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Posakonazol i̇çeren kati farmasöti̇k kompozi̇syon
WO2022034232A1 (en) 2020-08-13 2022-02-17 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Gastro-resistant high-strength formulation containing posaconazole
AU2022324717A1 (en) 2021-11-25 2024-06-13 Alfred E. Tiefenbacher (Gmbh Und Co. Kg) Granules containing posaconazole
EP4091604B1 (en) 2021-11-25 2024-04-03 Alfred E. Tiefenbacher (GmbH & Co. KG) Granules containing posaconazole

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL103558A0 (en) * 1991-10-30 1993-03-15 Schering Corp Tri-substituted tetrahydrofuran antifungals
DE122006000004I2 (de) * 1993-12-21 2007-03-29 Schering Corp Fungizide Tetrahydrofurane
SK282059B6 (sk) * 1994-01-24 2001-10-08 Janssen Pharmaceutica N. V. Azoly, spôsob ich výroby a farmaceutické prostriedky na ich báze
US5625064A (en) * 1995-04-19 1997-04-29 Schering Corporation Process for the preparation of triazolones
CN1073109C (zh) * 1995-06-02 2001-10-17 先灵公司 四氢呋喃杀真菌剂

Also Published As

Publication number Publication date
MX225999B (es) 2005-02-02
KR20010030959A (ko) 2001-04-16
NO20001779L (no) 2000-06-06
PE120499A1 (es) 1999-12-04
ID29290A (id) 2001-08-16
AU759982B2 (en) 2003-05-01
NO20001779D0 (no) 2000-04-06
SK5122000A3 (en) 2000-09-12
JP2012153729A (ja) 2012-08-16
IL135331A (en) 2005-08-31
PT1021439E (pt) 2004-07-30
CN1281449A (zh) 2001-01-24
JP2012153730A (ja) 2012-08-16
BR9812866A (pt) 2000-08-08
AU9780398A (en) 1999-04-27
PH11998002606B1 (en) 2006-08-10
CA2305803A1 (en) 1999-04-15
JP2008106075A (ja) 2008-05-08
HUP0004899A3 (en) 2002-03-28
CN1125067C (zh) 2003-10-22
CA2305803C (en) 2009-12-22
EP1021439A1 (en) 2000-07-26
DE69822859D1 (de) 2004-05-06
ES2217594T3 (es) 2004-11-01
CZ299835B6 (cs) 2008-12-10
TW589310B (en) 2004-06-01
NO318827B1 (no) 2005-05-09
JP2001519346A (ja) 2001-10-23
EP1021439B1 (en) 2004-03-31
IL135331A0 (en) 2001-05-20
IN1998CH02232A (OSRAM) 2005-03-04
PL339659A1 (en) 2001-01-02
KR100626109B1 (ko) 2006-09-20
NZ503662A (en) 2002-10-25
SK285190B6 (sk) 2006-08-03
PL189317B1 (pl) 2005-07-29
CZ20001264A3 (cs) 2000-08-16
MY130126A (en) 2007-06-29
HUP0004899A2 (hu) 2002-02-28
HK1029588A1 (en) 2001-04-06
HU225233B1 (en) 2006-08-28
CO4970829A1 (es) 2000-11-07
AR015947A1 (es) 2001-05-30
DE69822859T2 (de) 2005-01-27
ZA989063B (en) 1999-04-06
MXPA00003404A (es) 2000-11-01
WO1999018097A1 (en) 1999-04-15
DK1021439T3 (da) 2004-05-10

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