AR002720A1 - Proceso para preparar una composición oral sólida de olanzapina con subrecubrimiento de polímero y recubrimiento coloreado - Google Patents

Proceso para preparar una composición oral sólida de olanzapina con subrecubrimiento de polímero y recubrimiento coloreado

Info

Publication number
AR002720A1
AR002720A1 ARP960101877A AR10187796A AR002720A1 AR 002720 A1 AR002720 A1 AR 002720A1 AR P960101877 A ARP960101877 A AR P960101877A AR 10187796 A AR10187796 A AR 10187796A AR 002720 A1 AR002720 A1 AR 002720A1
Authority
AR
Argentina
Prior art keywords
solid oral
preparing
olanzapine
oral composition
colored coating
Prior art date
Application number
ARP960101877A
Other languages
English (en)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23624847&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR002720(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of AR002720A1 publication Critical patent/AR002720A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

La invención proporciona un procedimiento para preparar formulaciones orales sólidas recubiertas farmacéuticamente apropiadas y aceptables deolanzepina de fórmula (I), mediante la granulación en húmedo (acuosa) bajo condiciones de elevadocizallamiento y secado en lecho fluido.De preferenciacorresponde, a la poliforma Forma II pura que tiene el patrón de difracción de RX (en polvo) detallado en la descripción.
ARP960101877A 1995-03-24 1996-03-22 Proceso para preparar una composición oral sólida de olanzapina con subrecubrimiento de polímero y recubrimiento coloreado AR002720A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US41046595A 1995-03-24 1995-03-24

Publications (1)

Publication Number Publication Date
AR002720A1 true AR002720A1 (es) 1998-04-29

Family

ID=23624847

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP960101877A AR002720A1 (es) 1995-03-24 1996-03-22 Proceso para preparar una composición oral sólida de olanzapina con subrecubrimiento de polímero y recubrimiento coloreado
AR33587496A AR001405A1 (es) 1995-03-24 1996-03-22 Formulación oral de 2-metil-tieno-beno-diacepina.

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR33587496A AR001405A1 (es) 1995-03-24 1996-03-22 Formulación oral de 2-metil-tieno-beno-diacepina.

Country Status (46)

Country Link
US (4) US5919485A (es)
EP (2) EP1093815B1 (es)
JP (1) JPH11502848A (es)
KR (1) KR100408172B1 (es)
CN (1) CN1178662C (es)
AP (1) AP679A (es)
AR (2) AR002720A1 (es)
AT (3) ATE206924T1 (es)
AU (1) AU696601B2 (es)
BG (1) BG62594B1 (es)
BR (1) BR9607791A (es)
CA (1) CA2216372C (es)
CH (1) CH691217A5 (es)
CO (1) CO4700474A1 (es)
CR (1) CR5278A (es)
CZ (1) CZ296007B6 (es)
DE (3) DE69634053T2 (es)
DK (3) DK0733367T3 (es)
EA (1) EA000938B1 (es)
EE (1) EE03551B1 (es)
EG (1) EG24077A (es)
ES (2) ES2232379T3 (es)
FI (1) FI973749A (es)
GB (1) GB2313783B (es)
HU (1) HU225269B1 (es)
IL (1) IL117611A (es)
IS (1) IS1903B (es)
LT (1) LT4350B (es)
LU (1) LU90115B1 (es)
LV (1) LV11983B (es)
MY (1) MY113440A (es)
NO (1) NO320388B1 (es)
NZ (1) NZ306111A (es)
OA (1) OA10511A (es)
PE (1) PE44997A1 (es)
PL (1) PL188316B1 (es)
PT (2) PT1093815E (es)
RO (1) RO118370B1 (es)
SE (1) SE9703206L (es)
SI (3) SI0733367T1 (es)
SK (1) SK283745B6 (es)
TR (1) TR199701018T1 (es)
TW (1) TW426526B (es)
UA (1) UA44766C2 (es)
WO (1) WO1996029995A1 (es)
ZA (1) ZA962338B (es)

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TWI320783B (en) 2005-04-14 2010-02-21 Otsuka Pharma Co Ltd Heterocyclic compound
PL385455A1 (pl) * 2005-04-22 2008-11-24 Teva Pharmaceuticals Usa,Inc. Doustna rozpadająca się farmaceutyczna tabletka preparatów olanzapiny
EP1885383B1 (en) * 2005-05-31 2016-09-21 IAMS Europe B.V. Feline probiotic bifidobacteria
AR052472A1 (es) * 2005-05-31 2007-03-21 Iams Company Lactobacilos probioticos para felinos
US20070014847A1 (en) * 2005-07-05 2007-01-18 Ahmed Salah U Coated capsules and methods of making and using the same
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Also Published As

Publication number Publication date
LT97149A (en) 1998-01-26
JPH11502848A (ja) 1999-03-09
DE19681287T1 (de) 1998-03-19
EP1093815B1 (en) 2004-12-15
MX9707186A (es) 1997-11-29
DK109097A (da) 1997-11-12
EP0733367B1 (en) 2001-10-17
RO118370B1 (ro) 2003-05-30
US5919485A (en) 1999-07-06
TW426526B (en) 2001-03-21
ES2232379T3 (es) 2005-06-01
CO4700474A1 (es) 1998-12-29
EA199700260A1 (ru) 1998-02-26
AU696601B2 (en) 1998-09-17
CN1179102A (zh) 1998-04-15
TR199701018T1 (xx) 1998-01-21
US7229643B2 (en) 2007-06-12
US6190698B1 (en) 2001-02-20
NZ306111A (en) 1999-02-25
SI0733367T1 (en) 2002-06-30
FI973749A0 (fi) 1997-09-22
PE44997A1 (es) 1997-10-23
LU90115B1 (fr) 1997-09-10
HUP9800410A2 (hu) 1998-07-28
PT733367E (pt) 2002-03-28
DK173323B1 (da) 2000-07-24
LV11983B (en) 1998-07-20
LT4350B (lt) 1998-05-25
NO974363L (no) 1997-11-17
CH691217A5 (de) 2001-05-31
BG101901A (en) 1998-10-30
AT405606B (de) 1999-10-25
DE69615887D1 (de) 2001-11-22
GB9719817D0 (en) 1997-11-19
HU225269B1 (en) 2006-08-28
BR9607791A (pt) 1998-07-07
OA10511A (en) 2002-04-24
SE9703206D0 (sv) 1997-09-05
AU5428096A (en) 1996-10-16
PL322579A1 (en) 1998-02-02
SK128297A3 (en) 1998-03-04
IS1903B (is) 2003-11-20
GB2313783B (en) 1998-11-18
SI9620041A (sl) 1998-06-30
EE9700328A (et) 1998-06-15
DK0733367T3 (da) 2001-11-26
PL188316B1 (pl) 2005-01-31
CZ300197A3 (en) 1997-12-17
US20010018071A1 (en) 2001-08-30
HUP9800410A3 (en) 2000-01-28
BG62594B1 (bg) 2000-03-31
LV11983A (lv) 1998-03-20
DE69634053T2 (de) 2005-12-22
US20050085462A1 (en) 2005-04-21
CN1178662C (zh) 2004-12-08
IS4565A (is) 1997-09-22
ES2164837T3 (es) 2002-03-01
MY113440A (en) 2002-02-28
CR5278A (es) 1996-07-04
NO974363D0 (no) 1997-09-22
UA44766C2 (uk) 2002-03-15
CZ296007B6 (cs) 2005-12-14
SI1093815T1 (en) 2005-06-30
NO320388B1 (no) 2005-11-28
IL117611A0 (en) 1996-07-23
ZA962338B (en) 1997-09-22
AP679A (en) 1998-09-28
EG24077A (en) 2008-05-11
KR100408172B1 (ko) 2004-02-18
SK283745B6 (sk) 2003-12-02
SE9703206L (sv) 1997-09-05
AR001405A1 (es) 1997-10-22
PT1093815E (pt) 2005-03-31
DE69634053D1 (de) 2005-01-20
AP9701064A0 (en) 1997-10-31
ATE284695T1 (de) 2005-01-15
EP0733367A1 (en) 1996-09-25
KR19980703189A (ko) 1998-10-15
ATA902296A (de) 1999-02-15
CA2216372A1 (en) 1996-10-03
EA000938B1 (ru) 2000-06-26
US6780433B2 (en) 2004-08-24
EE03551B1 (et) 2001-12-17
DK1093815T3 (da) 2005-04-25
CA2216372C (en) 2007-11-20
FI973749A (fi) 1997-09-22
WO1996029995A1 (en) 1996-10-03
GB2313783A (en) 1997-12-10
ATE206924T1 (de) 2001-11-15
IL117611A (en) 2002-05-23
EP1093815A1 (en) 2001-04-25
DE69615887T2 (de) 2002-04-11

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