ZA201405870B - Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)-5-fluoro-3-phenylquinazolin-4(3h)-one - Google Patents

Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)-5-fluoro-3-phenylquinazolin-4(3h)-one

Info

Publication number
ZA201405870B
ZA201405870B ZA2014/05870A ZA201405870A ZA201405870B ZA 201405870 B ZA201405870 B ZA 201405870B ZA 2014/05870 A ZA2014/05870 A ZA 2014/05870A ZA 201405870 A ZA201405870 A ZA 201405870A ZA 201405870 B ZA201405870 B ZA 201405870B
Authority
ZA
South Africa
Prior art keywords
phenylquinazolin
purin
ylamino
fluoro
polymorphic forms
Prior art date
Application number
ZA2014/05870A
Other languages
English (en)
Inventor
Jerry B Evarts
Fang Wang
Duong Tran
Keiko Sujino
Bing Shi
Michael Gerber
Ernest Carra
Original Assignee
Gilead Calistoga Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49117265&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA201405870(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Calistoga Llc filed Critical Gilead Calistoga Llc
Publication of ZA201405870B publication Critical patent/ZA201405870B/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
ZA2014/05870A 2012-03-05 2014-08-11 Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)-5-fluoro-3-phenylquinazolin-4(3h)-one ZA201405870B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261606870P 2012-03-05 2012-03-05
PCT/US2013/029157 WO2013134288A1 (en) 2012-03-05 2013-03-05 Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3h)-one

Publications (1)

Publication Number Publication Date
ZA201405870B true ZA201405870B (en) 2015-11-25

Family

ID=49117265

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA2014/05870A ZA201405870B (en) 2012-03-05 2014-08-11 Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)-5-fluoro-3-phenylquinazolin-4(3h)-one

Country Status (31)

Country Link
US (3) US8865730B2 (cg-RX-API-DMAC7.html)
EP (1) EP2834241B1 (cg-RX-API-DMAC7.html)
JP (2) JP2015509537A (cg-RX-API-DMAC7.html)
KR (1) KR20140133590A (cg-RX-API-DMAC7.html)
CN (2) CN106146506A (cg-RX-API-DMAC7.html)
AP (1) AP2014007875A0 (cg-RX-API-DMAC7.html)
AR (1) AR090253A1 (cg-RX-API-DMAC7.html)
AU (1) AU2013203620B2 (cg-RX-API-DMAC7.html)
BR (1) BR112014021935A2 (cg-RX-API-DMAC7.html)
CA (1) CA2864305C (cg-RX-API-DMAC7.html)
CL (1) CL2014002358A1 (cg-RX-API-DMAC7.html)
CO (1) CO7071131A2 (cg-RX-API-DMAC7.html)
CR (1) CR20140460A (cg-RX-API-DMAC7.html)
EA (3) EA201691327A1 (cg-RX-API-DMAC7.html)
EC (1) ECSP14020478A (cg-RX-API-DMAC7.html)
ES (1) ES2848273T3 (cg-RX-API-DMAC7.html)
IN (1) IN2014DN07105A (cg-RX-API-DMAC7.html)
MA (1) MA37379A1 (cg-RX-API-DMAC7.html)
MD (1) MD20140100A2 (cg-RX-API-DMAC7.html)
MX (1) MX2014010656A (cg-RX-API-DMAC7.html)
NZ (1) NZ629684A (cg-RX-API-DMAC7.html)
PE (1) PE20141792A1 (cg-RX-API-DMAC7.html)
PH (1) PH12014501920A1 (cg-RX-API-DMAC7.html)
PL (1) PL2834241T3 (cg-RX-API-DMAC7.html)
PT (1) PT2834241T (cg-RX-API-DMAC7.html)
SG (1) SG11201405446PA (cg-RX-API-DMAC7.html)
SI (1) SI2834241T1 (cg-RX-API-DMAC7.html)
TW (1) TW201350486A (cg-RX-API-DMAC7.html)
UY (1) UY34656A (cg-RX-API-DMAC7.html)
WO (1) WO2013134288A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA201405870B (cg-RX-API-DMAC7.html)

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