IN2014DN07105A - - Google Patents

Info

Publication number
IN2014DN07105A
IN2014DN07105A IN7105DEN2014A IN2014DN07105A IN 2014DN07105 A IN2014DN07105 A IN 2014DN07105A IN 7105DEN2014 A IN7105DEN2014 A IN 7105DEN2014A IN 2014DN07105 A IN2014DN07105 A IN 2014DN07105A
Authority
IN
India
Prior art keywords
methods
phenylquinazolin
purin
ylamino
polymorphs
Prior art date
Application number
Inventor
Ernest Carra
Michael Gerber
Bing Shi
Keiko Sujino
Duong Tran
Fang Wang
Jerry B Evarts
Original Assignee
Gilead Calistoga Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49117265&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2014DN07105(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Calistoga Llc filed Critical Gilead Calistoga Llc
Publication of IN2014DN07105A publication Critical patent/IN2014DN07105A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

POLYMORPHS OF (5) 2 (1 (9H PURIN 6 YLAMINO)PROPYL) 5 FLUORO 3 PHENYLQUINAZOLIN 4(3H) ONE COMPOSITIONS THEREOF METHODS FOR THEIR PREPARATION AND METHODS FOR THEIR USE ARE DISCLOSED.
IN7105DEN2014 2012-03-05 2013-03-05 IN2014DN07105A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261606870P 2012-03-05 2012-03-05
PCT/US2013/029157 WO2013134288A1 (en) 2012-03-05 2013-03-05 Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3h)-one

Publications (1)

Publication Number Publication Date
IN2014DN07105A true IN2014DN07105A (en) 2015-04-24

Family

ID=49117265

Family Applications (1)

Application Number Title Priority Date Filing Date
IN7105DEN2014 IN2014DN07105A (en) 2012-03-05 2013-03-05

Country Status (32)

Country Link
US (3) US8865730B2 (en)
EP (1) EP2834241B1 (en)
JP (2) JP2015509537A (en)
KR (1) KR20140133590A (en)
CN (2) CN104334560A (en)
AP (1) AP2014007875A0 (en)
AR (1) AR090253A1 (en)
AU (1) AU2013203620B2 (en)
BR (1) BR112014021935A2 (en)
CA (1) CA2864305C (en)
CL (1) CL2014002358A1 (en)
CO (1) CO7071131A2 (en)
CR (1) CR20140460A (en)
EA (3) EA025407B1 (en)
EC (1) ECSP14020478A (en)
ES (1) ES2848273T3 (en)
HK (1) HK1206345A1 (en)
IN (1) IN2014DN07105A (en)
MA (1) MA37379A1 (en)
MD (1) MD20140100A2 (en)
MX (1) MX2014010656A (en)
NZ (1) NZ629684A (en)
PE (1) PE20141792A1 (en)
PH (1) PH12014501920A1 (en)
PL (1) PL2834241T3 (en)
PT (1) PT2834241T (en)
SG (1) SG11201405446PA (en)
SI (1) SI2834241T1 (en)
TW (1) TW201350486A (en)
UY (1) UY34656A (en)
WO (1) WO2013134288A1 (en)
ZA (1) ZA201405870B (en)

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CN106565716B (en) * 2015-10-10 2021-06-15 上海创诺制药有限公司 Idelalisib crystal form A and preparation method thereof
HU231016B1 (en) * 2015-11-30 2019-11-28 Egis Gyógyszergyár Zrt. New polymorph and solvate of idelalisib
WO2017175184A1 (en) * 2016-04-07 2017-10-12 Laurus Labs Limited Process for preparation of amorphous form of idelalisib
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CN106632337B (en) * 2016-10-18 2018-11-20 湖北生物医药产业技术研究院有限公司 It ends for this crystal form, pharmaceutical composition, preparation method and purposes of Larry
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CN107573345B (en) * 2017-09-12 2020-01-10 浙江乐普药业股份有限公司 Preparation method of erigeron and intermediate thereof
CN109575027A (en) * 2017-09-29 2019-04-05 宁波爱诺医药科技有限公司 A kind of monohydrate and preparation method thereof of anti-tumor drug Ai Delibu
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Also Published As

Publication number Publication date
CO7071131A2 (en) 2014-09-30
ZA201405870B (en) 2015-11-25
CA2864305A1 (en) 2013-09-12
CL2014002358A1 (en) 2015-04-24
PE20141792A1 (en) 2014-12-07
EP2834241A4 (en) 2015-11-11
EA201691327A1 (en) 2017-03-31
US9469643B2 (en) 2016-10-18
UY34656A (en) 2013-10-31
MX2014010656A (en) 2015-03-03
US20150080572A1 (en) 2015-03-19
WO2013134288A1 (en) 2013-09-12
SG11201405446PA (en) 2014-10-30
SI2834241T1 (en) 2021-06-30
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