SG11201405446PA - POLYMORPHIC FORMS OF (<i>S</i>)-2-(1-(9H-PURIN-6-YLAMINO)PROPYL)-5-FLUORO-3-PHENYLQUINAZOLIN-4(<i>3H</i>)-ONE - Google Patents

POLYMORPHIC FORMS OF (<i>S</i>)-2-(1-(9H-PURIN-6-YLAMINO)PROPYL)-5-FLUORO-3-PHENYLQUINAZOLIN-4(<i>3H</i>)-ONE

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Publication number
SG11201405446PA
SG11201405446PA SG11201405446PA SG11201405446PA SG11201405446PA SG 11201405446P A SG11201405446P A SG 11201405446PA SG 11201405446P A SG11201405446P A SG 11201405446PA SG 11201405446P A SG11201405446P A SG 11201405446PA SG 11201405446P A SG11201405446P A SG 11201405446PA
Authority
SG
Singapore
Prior art keywords
phenylquinazolin
purin
ylamino
fluoro
propyl
Prior art date
Application number
SG11201405446PA
Inventor
Ernest Carra
Michael Gerber
Bing Shi
Keiko Sujino
Duong Tran
Fang Wang
Jerry B Evarts
Original Assignee
Gilead Calistoga Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49117265&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201405446P(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Calistoga Llc filed Critical Gilead Calistoga Llc
Publication of SG11201405446PA publication Critical patent/SG11201405446PA/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs
SG11201405446PA 2012-03-05 2013-03-05 POLYMORPHIC FORMS OF (<i>S</i>)-2-(1-(9H-PURIN-6-YLAMINO)PROPYL)-5-FLUORO-3-PHENYLQUINAZOLIN-4(<i>3H</i>)-ONE SG11201405446PA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261606870P 2012-03-05 2012-03-05
PCT/US2013/029157 WO2013134288A1 (en) 2012-03-05 2013-03-05 Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3h)-one

Publications (1)

Publication Number Publication Date
SG11201405446PA true SG11201405446PA (en) 2014-10-30

Family

ID=49117265

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201405446PA SG11201405446PA (en) 2012-03-05 2013-03-05 POLYMORPHIC FORMS OF (<i>S</i>)-2-(1-(9H-PURIN-6-YLAMINO)PROPYL)-5-FLUORO-3-PHENYLQUINAZOLIN-4(<i>3H</i>)-ONE

Country Status (32)

Country Link
US (3) US8865730B2 (en)
EP (1) EP2834241B1 (en)
JP (2) JP2015509537A (en)
KR (1) KR20140133590A (en)
CN (2) CN104334560A (en)
AP (1) AP2014007875A0 (en)
AR (1) AR090253A1 (en)
AU (1) AU2013203620B2 (en)
BR (1) BR112014021935A2 (en)
CA (1) CA2864305C (en)
CL (1) CL2014002358A1 (en)
CO (1) CO7071131A2 (en)
CR (1) CR20140460A (en)
EA (3) EA025407B1 (en)
EC (1) ECSP14020478A (en)
ES (1) ES2848273T3 (en)
HK (1) HK1206345A1 (en)
IN (1) IN2014DN07105A (en)
MA (1) MA37379A1 (en)
MD (1) MD20140100A2 (en)
MX (1) MX2014010656A (en)
NZ (1) NZ629684A (en)
PE (1) PE20141792A1 (en)
PH (1) PH12014501920A1 (en)
PL (1) PL2834241T3 (en)
PT (1) PT2834241T (en)
SG (1) SG11201405446PA (en)
SI (1) SI2834241T1 (en)
TW (1) TW201350486A (en)
UY (1) UY34656A (en)
WO (1) WO2013134288A1 (en)
ZA (1) ZA201405870B (en)

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US9469643B2 (en) 2016-10-18
US20150080572A1 (en) 2015-03-19
CO7071131A2 (en) 2014-09-30
AR090253A1 (en) 2014-10-29
BR112014021935A2 (en) 2019-09-24
PE20141792A1 (en) 2014-12-07
SI2834241T1 (en) 2021-06-30
IN2014DN07105A (en) 2015-04-24
ES2848273T3 (en) 2021-08-06
CN106146506A (en) 2016-11-23
WO2013134288A1 (en) 2013-09-12
MD20140100A2 (en) 2015-01-31
EA201491473A1 (en) 2015-03-31
PL2834241T3 (en) 2021-07-12
UY34656A (en) 2013-10-31
MA37379A1 (en) 2016-11-30
ZA201405870B (en) 2015-11-25
US8865730B2 (en) 2014-10-21
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