EA201691327A1 - Полиморфные формы (s)-2-(1-(9h-пурин-6-иламино)пропил)-5-фтор-3-фенилхиназолин-4(3h)-она - Google Patents

Полиморфные формы (s)-2-(1-(9h-пурин-6-иламино)пропил)-5-фтор-3-фенилхиназолин-4(3h)-она

Info

Publication number
EA201691327A1
EA201691327A1 EA201691327A EA201691327A EA201691327A1 EA 201691327 A1 EA201691327 A1 EA 201691327A1 EA 201691327 A EA201691327 A EA 201691327A EA 201691327 A EA201691327 A EA 201691327A EA 201691327 A1 EA201691327 A1 EA 201691327A1
Authority
EA
Eurasian Patent Office
Prior art keywords
purin
propyl
ftor
chinazolin
ilamino
Prior art date
Application number
EA201691327A
Other languages
English (en)
Inventor
Эрнест Карра
Майкл Гербер
Бин Ши
Кейко Судзино
Дуонг Трэн
Фан ВАН
Джерри Б. Эвартс
Original Assignee
Джилид Калистога Ллс
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49117265&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201691327(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Джилид Калистога Ллс filed Critical Джилид Калистога Ллс
Publication of EA201691327A1 publication Critical patent/EA201691327A1/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

В изобретении предложены полиморфы (S)-2-(1-(9Н-пурин-6-иламино)пропил)-5-фтор-3-фенилхиназолин-4(3H)-она, содержащие их композиции, способы их получения и способы их применения.
EA201691327A 2012-03-05 2013-03-05 Полиморфные формы (s)-2-(1-(9h-пурин-6-иламино)пропил)-5-фтор-3-фенилхиназолин-4(3h)-она EA201691327A1 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261606870P 2012-03-05 2012-03-05

Publications (1)

Publication Number Publication Date
EA201691327A1 true EA201691327A1 (ru) 2017-03-31

Family

ID=49117265

Family Applications (3)

Application Number Title Priority Date Filing Date
EA201491473A EA025407B1 (ru) 2012-03-05 2013-03-05 Полиморфная форма i (s)-2-(1-(9h-пурин-6-иламино)пропил)-5-фтор-3-фенилхиназолин-4(3h)-она
EA201691327A EA201691327A1 (ru) 2012-03-05 2013-03-05 Полиморфные формы (s)-2-(1-(9h-пурин-6-иламино)пропил)-5-фтор-3-фенилхиназолин-4(3h)-она
EA201690461A EA201690461A1 (ru) 2012-03-05 2013-03-05 Полиморфные формы (s)-2-(1-(9h-пурин-6-иламино)пропил)-5-фтор-3-фенилхиназолин-4(3h)-она

Family Applications Before (1)

Application Number Title Priority Date Filing Date
EA201491473A EA025407B1 (ru) 2012-03-05 2013-03-05 Полиморфная форма i (s)-2-(1-(9h-пурин-6-иламино)пропил)-5-фтор-3-фенилхиназолин-4(3h)-она

Family Applications After (1)

Application Number Title Priority Date Filing Date
EA201690461A EA201690461A1 (ru) 2012-03-05 2013-03-05 Полиморфные формы (s)-2-(1-(9h-пурин-6-иламино)пропил)-5-фтор-3-фенилхиназолин-4(3h)-она

Country Status (32)

Country Link
US (3) US8865730B2 (ru)
EP (1) EP2834241B1 (ru)
JP (2) JP2015509537A (ru)
KR (1) KR20140133590A (ru)
CN (2) CN104334560A (ru)
AP (1) AP2014007875A0 (ru)
AR (1) AR090253A1 (ru)
AU (1) AU2013203620B2 (ru)
BR (1) BR112014021935A2 (ru)
CA (1) CA2864305C (ru)
CL (1) CL2014002358A1 (ru)
CO (1) CO7071131A2 (ru)
CR (1) CR20140460A (ru)
EA (3) EA025407B1 (ru)
EC (1) ECSP14020478A (ru)
ES (1) ES2848273T3 (ru)
HK (1) HK1206345A1 (ru)
IN (1) IN2014DN07105A (ru)
MA (1) MA37379A1 (ru)
MD (1) MD20140100A2 (ru)
MX (1) MX2014010656A (ru)
NZ (1) NZ629684A (ru)
PE (1) PE20141792A1 (ru)
PH (1) PH12014501920A1 (ru)
PL (1) PL2834241T3 (ru)
PT (1) PT2834241T (ru)
SG (1) SG11201405446PA (ru)
SI (1) SI2834241T1 (ru)
TW (1) TW201350486A (ru)
UY (1) UY34656A (ru)
WO (1) WO2013134288A1 (ru)
ZA (1) ZA201405870B (ru)

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