HK1206345A1 - Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3- phenylquinazolin-4(3h)-one (s)-2-(1-(9h--6-))-5--3--4(3h)- - Google Patents

Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3- phenylquinazolin-4(3h)-one (s)-2-(1-(9h--6-))-5--3--4(3h)-

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Publication number
HK1206345A1
HK1206345A1 HK15106935.8A HK15106935A HK1206345A1 HK 1206345 A1 HK1206345 A1 HK 1206345A1 HK 15106935 A HK15106935 A HK 15106935A HK 1206345 A1 HK1206345 A1 HK 1206345A1
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HK
Hong Kong
Prior art keywords
phenylquinazolin
purin
ylamino
fluoro
propyl
Prior art date
Application number
HK15106935.8A
Other languages
English (en)
Chinese (zh)
Inventor
Ernest Carra
Michael Gerber
Bing Shi
Keiko Sujino
Duong Tran
Fang Wang
B Evarts Jerry
Original Assignee
Gilead Calistoga Llc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49117265&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1206345(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Calistoga Llc filed Critical Gilead Calistoga Llc
Publication of HK1206345A1 publication Critical patent/HK1206345A1/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
HK15106935.8A 2012-03-05 2015-07-21 Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3- phenylquinazolin-4(3h)-one (s)-2-(1-(9h--6-))-5--3--4(3h)- HK1206345A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261606870P 2012-03-05 2012-03-05
PCT/US2013/029157 WO2013134288A1 (en) 2012-03-05 2013-03-05 Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3h)-one

Publications (1)

Publication Number Publication Date
HK1206345A1 true HK1206345A1 (en) 2016-01-08

Family

ID=49117265

Family Applications (1)

Application Number Title Priority Date Filing Date
HK15106935.8A HK1206345A1 (en) 2012-03-05 2015-07-21 Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3- phenylquinazolin-4(3h)-one (s)-2-(1-(9h--6-))-5--3--4(3h)-

Country Status (32)

Country Link
US (3) US8865730B2 (xx)
EP (1) EP2834241B1 (xx)
JP (2) JP2015509537A (xx)
KR (1) KR20140133590A (xx)
CN (2) CN104334560A (xx)
AP (1) AP2014007875A0 (xx)
AR (1) AR090253A1 (xx)
AU (1) AU2013203620B2 (xx)
BR (1) BR112014021935A2 (xx)
CA (1) CA2864305C (xx)
CL (1) CL2014002358A1 (xx)
CO (1) CO7071131A2 (xx)
CR (1) CR20140460A (xx)
EA (3) EA025407B1 (xx)
EC (1) ECSP14020478A (xx)
ES (1) ES2848273T3 (xx)
HK (1) HK1206345A1 (xx)
IN (1) IN2014DN07105A (xx)
MA (1) MA37379A1 (xx)
MD (1) MD20140100A2 (xx)
MX (1) MX2014010656A (xx)
NZ (1) NZ629684A (xx)
PE (1) PE20141792A1 (xx)
PH (1) PH12014501920A1 (xx)
PL (1) PL2834241T3 (xx)
PT (1) PT2834241T (xx)
SG (1) SG11201405446PA (xx)
SI (1) SI2834241T1 (xx)
TW (1) TW201350486A (xx)
UY (1) UY34656A (xx)
WO (1) WO2013134288A1 (xx)
ZA (1) ZA201405870B (xx)

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