PT2834241T - Formas polimórficas de (s)-2-(1-(9h-purin-6-ilamino)propil)-5-fluoro-3-fenil quinazolina-4(3h)-ona - Google Patents

Formas polimórficas de (s)-2-(1-(9h-purin-6-ilamino)propil)-5-fluoro-3-fenil quinazolina-4(3h)-ona

Info

Publication number
PT2834241T
PT2834241T PT137572301T PT13757230T PT2834241T PT 2834241 T PT2834241 T PT 2834241T PT 137572301 T PT137572301 T PT 137572301T PT 13757230 T PT13757230 T PT 13757230T PT 2834241 T PT2834241 T PT 2834241T
Authority
PT
Portugal
Prior art keywords
phenylquinazolin
purin
ylamino
fluoro
propyl
Prior art date
Application number
PT137572301T
Other languages
English (en)
Original Assignee
Gilead Calistoga Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49117265&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2834241(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Calistoga Llc filed Critical Gilead Calistoga Llc
Publication of PT2834241T publication Critical patent/PT2834241T/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
PT137572301T 2012-03-05 2013-03-05 Formas polimórficas de (s)-2-(1-(9h-purin-6-ilamino)propil)-5-fluoro-3-fenil quinazolina-4(3h)-ona PT2834241T (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261606870P 2012-03-05 2012-03-05

Publications (1)

Publication Number Publication Date
PT2834241T true PT2834241T (pt) 2021-02-05

Family

ID=49117265

Family Applications (1)

Application Number Title Priority Date Filing Date
PT137572301T PT2834241T (pt) 2012-03-05 2013-03-05 Formas polimórficas de (s)-2-(1-(9h-purin-6-ilamino)propil)-5-fluoro-3-fenil quinazolina-4(3h)-ona

Country Status (32)

Country Link
US (3) US8865730B2 (pt)
EP (1) EP2834241B1 (pt)
JP (2) JP2015509537A (pt)
KR (1) KR20140133590A (pt)
CN (2) CN104334560A (pt)
AP (1) AP2014007875A0 (pt)
AR (1) AR090253A1 (pt)
AU (1) AU2013203620B2 (pt)
BR (1) BR112014021935A2 (pt)
CA (1) CA2864305C (pt)
CL (1) CL2014002358A1 (pt)
CO (1) CO7071131A2 (pt)
CR (1) CR20140460A (pt)
EA (3) EA025407B1 (pt)
EC (1) ECSP14020478A (pt)
ES (1) ES2848273T3 (pt)
HK (1) HK1206345A1 (pt)
IN (1) IN2014DN07105A (pt)
MA (1) MA37379A1 (pt)
MD (1) MD20140100A2 (pt)
MX (1) MX2014010656A (pt)
NZ (1) NZ629684A (pt)
PE (1) PE20141792A1 (pt)
PH (1) PH12014501920A1 (pt)
PL (1) PL2834241T3 (pt)
PT (1) PT2834241T (pt)
SG (1) SG11201405446PA (pt)
SI (1) SI2834241T1 (pt)
TW (1) TW201350486A (pt)
UY (1) UY34656A (pt)
WO (1) WO2013134288A1 (pt)
ZA (1) ZA201405870B (pt)

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CN107573345B (zh) * 2017-09-12 2020-01-10 浙江乐普药业股份有限公司 一种艾代拉利司及其中间体的制备方法
CN109575027A (zh) * 2017-09-29 2019-04-05 宁波爱诺医药科技有限公司 一种抗肿瘤药物艾德力布的一水合物及其制备方法
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