ZA200809290B - Modulators of ATP-binding cassett transporters - Google Patents
Modulators of ATP-binding cassett transportersInfo
- Publication number
- ZA200809290B ZA200809290B ZA200809290A ZA200809290A ZA200809290B ZA 200809290 B ZA200809290 B ZA 200809290B ZA 200809290 A ZA200809290 A ZA 200809290A ZA 200809290 A ZA200809290 A ZA 200809290A ZA 200809290 B ZA200809290 B ZA 200809290B
- Authority
- ZA
- South Africa
- Prior art keywords
- transporters
- atp
- modulators
- cassett
- binding
- Prior art date
Links
Classifications
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US79045906P | 2006-04-07 | 2006-04-07 |
Publications (1)
Publication Number | Publication Date |
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ZA200809290B true ZA200809290B (en) | 2009-10-28 |
Family
ID=38477342
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA200809290A ZA200809290B (en) | 2006-04-07 | 2008-10-29 | Modulators of ATP-binding cassett transporters |
Country Status (22)
Country | Link |
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US (9) | US7776905B2 (el) |
EP (5) | EP3327016B1 (el) |
JP (3) | JP5420395B2 (el) |
CN (2) | CN103254177A (el) |
AU (1) | AU2007235260B2 (el) |
BR (1) | BRPI0710965B8 (el) |
CA (2) | CA2648719C (el) |
CY (3) | CY1116979T1 (el) |
DK (3) | DK2674428T3 (el) |
ES (4) | ES2659364T3 (el) |
HU (4) | HUE036165T2 (el) |
IL (1) | IL194576A (el) |
IN (1) | IN2014KN02423A (el) |
LT (1) | LT3091011T (el) |
MX (1) | MX2008012945A (el) |
NZ (3) | NZ571803A (el) |
PL (4) | PL3091011T3 (el) |
PT (3) | PT2674428T (el) |
RU (1) | RU2451018C2 (el) |
SI (4) | SI2674428T1 (el) |
WO (1) | WO2007117715A2 (el) |
ZA (1) | ZA200809290B (el) |
Families Citing this family (106)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20100074949A1 (en) | 2008-08-13 | 2010-03-25 | William Rowe | Pharmaceutical composition and administration thereof |
AU2004272599A1 (en) | 2003-09-06 | 2005-03-24 | Vertex Pharmaceuticals Incorporated | Modulators of ATP-binding cassette transporters |
DE602004022319D1 (de) * | 2003-11-14 | 2009-09-10 | Vertex Pharma | Thiazole udn oxazole als modulatoren von atp-bindungs-kassetten-transportern |
US7977322B2 (en) | 2004-08-20 | 2011-07-12 | Vertex Pharmaceuticals Incorporated | Modulators of ATP-binding cassette transporters |
WO2005075435A1 (en) * | 2004-01-30 | 2005-08-18 | Vertex Pharmaceuticals Incorporated | Modulators of atp-binding cassette transporters |
EP2522659A3 (en) | 2004-06-24 | 2013-11-27 | Vertex Pharmaceuticals Incorporated | Modulators of ATP-binding cassette transporters |
EP1912983B1 (en) | 2005-08-11 | 2011-06-08 | Vertex Pharmaceuticals, Inc. | Modulators of cystic fibrosis transmembrane conductance regulator |
PL2774925T3 (pl) | 2005-11-08 | 2017-07-31 | Vertex Pharmaceuticals Incorporated | Heterocykliczne modulatory transporterów z kasetą wiążącą ATP |
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2007
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