ZA200603226B - Amide derivatives - Google Patents

Amide derivatives Download PDF

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Publication number
ZA200603226B
ZA200603226B ZA200603226A ZA200603226A ZA200603226B ZA 200603226 B ZA200603226 B ZA 200603226B ZA 200603226 A ZA200603226 A ZA 200603226A ZA 200603226 A ZA200603226 A ZA 200603226A ZA 200603226 B ZA200603226 B ZA 200603226B
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ZA
South Africa
Prior art keywords
cyclopropyl
alkyl
methyl
oxoquinazolin
alkoxy
Prior art date
Application number
ZA200603226A
Other languages
English (en)
Inventor
Brown Dearg Sutherland
Nash Ian Alun
Original Assignee
Astrazeneca Ab
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29595715&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200603226(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of ZA200603226B publication Critical patent/ZA200603226B/en

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    • CCHEMISTRY; METALLURGY
    • C04CEMENTS; CONCRETE; ARTIFICIAL STONE; CERAMICS; REFRACTORIES
    • C04BLIME, MAGNESIA; SLAG; CEMENTS; COMPOSITIONS THEREOF, e.g. MORTARS, CONCRETE OR LIKE BUILDING MATERIALS; ARTIFICIAL STONE; CERAMICS; REFRACTORIES; TREATMENT OF NATURAL STONE
    • C04B35/00Shaped ceramic products characterised by their composition; Ceramics compositions; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/622Forming processes; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/626Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B
    • C04B35/63Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
    • C04B35/632Organic additives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/91Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
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    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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ZA200603226A 2003-10-24 2006-04-21 Amide derivatives ZA200603226B (en)

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GBGB0324790.5A GB0324790D0 (en) 2003-10-24 2003-10-24 Amide derivatives

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ZA200603226B true ZA200603226B (en) 2007-04-25

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US (1) US7750154B2 (ja)
EP (1) EP1682520B1 (ja)
JP (1) JP4987478B2 (ja)
KR (1) KR101127697B1 (ja)
CN (2) CN103012376A (ja)
AR (1) AR046308A1 (ja)
AT (1) ATE499347T1 (ja)
AU (1) AU2004285749B2 (ja)
BR (1) BRPI0415746A (ja)
CA (1) CA2543351C (ja)
DE (1) DE602004031543D1 (ja)
ES (1) ES2359409T3 (ja)
GB (1) GB0324790D0 (ja)
HK (1) HK1091830A1 (ja)
IL (1) IL175065A (ja)
IS (1) IS8450A (ja)
MX (1) MXPA06004465A (ja)
MY (1) MY140729A (ja)
NO (1) NO20062370L (ja)
NZ (1) NZ547095A (ja)
RU (1) RU2375352C2 (ja)
SA (1) SA04250351B1 (ja)
SG (1) SG147409A1 (ja)
TW (1) TWI343378B (ja)
UA (1) UA83867C2 (ja)
UY (1) UY28578A1 (ja)
WO (1) WO2005042502A1 (ja)
ZA (1) ZA200603226B (ja)

Families Citing this family (42)

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Publication number Priority date Publication date Assignee Title
BR0009083B1 (pt) 1999-03-17 2011-11-01 derivado de amida compreendendo um núcleo de quinazolinona, processo para a preparação de um derivado de amida, composição farmacêutica, e, uso de um derivado de amida.
GB0329572D0 (en) 2003-12-20 2004-01-28 Astrazeneca Ab Amide derivatives
US20050261278A1 (en) 2004-05-21 2005-11-24 Weiner David M Selective serotonin receptor inverse agonists as therapeutics for disease
MX2007008334A (es) 2005-01-10 2007-09-11 Acadia Pharm Inc Derivados aminofenilo como moduladores de receptor de androgeno selectivos.
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