ZA200501033B - 2,3,-dihydro-6-nitroimidazoÄ2,1-BÜoxazoles - Google Patents

2,3,-dihydro-6-nitroimidazoÄ2,1-BÜoxazoles Download PDF

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Publication number
ZA200501033B
ZA200501033B ZA200501033A ZA200501033A ZA200501033B ZA 200501033 B ZA200501033 B ZA 200501033B ZA 200501033 A ZA200501033 A ZA 200501033A ZA 200501033 A ZA200501033 A ZA 200501033A ZA 200501033 B ZA200501033 B ZA 200501033B
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ZA
South Africa
Prior art keywords
group
substituted
halogen
unsubstituted
phenyl
Prior art date
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ZA200501033A
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English (en)
Inventor
Hidetsugu Tsubouchi
Hirofumi Sasaki
Hideaki Kuroda
Motohiro Itotani
Takeshi Hasegawa
Yoshikazu Haraguchi
Takeshi Kuroda
Takayuki Matsuzaki
Kuninori Tai
Tai Takayuki
Makoto Komatsu
Makoto Matsumoto
Hiroyuki Hashizume
Tatsuo Tomishige
Yuji Seike
Masanori Kawasaki
Takumi Sumida
Shin Miyamura
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Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of ZA200501033B publication Critical patent/ZA200501033B/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/20—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
ZA200501033A 2002-10-11 2005-02-03 2,3,-dihydro-6-nitroimidazoÄ2,1-BÜoxazoles ZA200501033B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2002298259 2002-10-11

Publications (1)

Publication Number Publication Date
ZA200501033B true ZA200501033B (en) 2006-06-28

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ID=32089299

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200501033A ZA200501033B (en) 2002-10-11 2005-02-03 2,3,-dihydro-6-nitroimidazoÄ2,1-BÜoxazoles

Country Status (26)

Country Link
US (1) US7262212B2 (cs)
EP (2) EP2570418A3 (cs)
JP (1) JP4186065B2 (cs)
KR (1) KR100723847B1 (cs)
CN (4) CN102532162B (cs)
AR (4) AR041198A1 (cs)
AU (1) AU2003272979B2 (cs)
BE (1) BE2014C053I2 (cs)
BR (1) BRPI0314344B8 (cs)
CA (1) CA2497569C (cs)
CY (2) CY1113578T1 (cs)
DK (1) DK1555267T3 (cs)
ES (1) ES2400179T3 (cs)
FR (1) FR14C0066I2 (cs)
HU (1) HUS1400046I1 (cs)
LU (1) LU92517I2 (cs)
MX (1) MXPA05003674A (cs)
MY (1) MY139244A (cs)
PL (3) PL217919B1 (cs)
PT (1) PT1555267E (cs)
RU (1) RU2326121C3 (cs)
SI (1) SI1555267T1 (cs)
TW (1) TWI347946B (cs)
UA (1) UA83200C2 (cs)
WO (1) WO2004033463A1 (cs)
ZA (1) ZA200501033B (cs)

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CN106317072B (zh) * 2015-06-17 2020-03-17 盟科医药技术(上海)有限公司 用于分枝杆菌感染治疗的杂环化合物及其应用
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CN109705022A (zh) * 2018-12-28 2019-05-03 上海彩迩文生化科技有限公司 一种芳香胺中间体的制备方法
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DK1555267T3 (da) 2013-02-11
AU2003272979A1 (en) 2004-05-04
CA2497569C (en) 2011-05-24
CY2014041I2 (el) 2016-07-27
EP1555267B1 (en) 2013-01-16
CA2497569A1 (en) 2004-04-22
BRPI0314344B1 (pt) 2019-11-26
CY2014041I1 (el) 2016-07-27
PL217919B1 (pl) 2014-09-30
UA83200C2 (en) 2008-06-25
EP1555267A1 (en) 2005-07-20
ES2400179T3 (es) 2013-04-08
KR20050061473A (ko) 2005-06-22
FR14C0066I2 (fr) 2015-05-22
TW200420568A (en) 2004-10-16
CN102532162B (zh) 2015-05-27
HK1171018A1 (en) 2013-03-15
EP2570418A3 (en) 2013-07-03
PL404913A1 (pl) 2013-09-30
CY1113578T1 (el) 2016-06-22
EP2570418A2 (en) 2013-03-20
EP1555267A4 (en) 2010-08-18
BRPI0314344B8 (pt) 2021-05-25
MXPA05003674A (es) 2005-06-08
AR091771A2 (es) 2015-02-25
CN1705670A (zh) 2005-12-07
CN100366624C (zh) 2008-02-06
PT1555267E (pt) 2013-01-29
FR14C0066I1 (cs) 2014-10-17
US7262212B2 (en) 2007-08-28
CN102532162A (zh) 2012-07-04
PL409525A1 (pl) 2014-11-10
CN101172981A (zh) 2008-05-07
BR0314344A (pt) 2005-07-12
JP2004149527A (ja) 2004-05-27
RU2326121C2 (ru) 2008-06-10
CN101255170A (zh) 2008-09-03
MY139244A (en) 2009-09-30
RU2326121C3 (ru) 2021-09-17
RU2005114017A (ru) 2006-01-20
AU2003272979B2 (en) 2009-07-23
HUS1400046I1 (hu) 2017-04-28
JP4186065B2 (ja) 2008-11-26
PL376157A1 (en) 2005-12-27
BE2014C053I2 (cs) 2022-08-30
HK1085463A1 (zh) 2006-08-25
LU92517I2 (fr) 2014-10-13
AR041198A1 (es) 2005-05-04
SI1555267T1 (sl) 2013-05-31
US20060094767A1 (en) 2006-05-04
TWI347946B (en) 2011-09-01
WO2004033463A1 (ja) 2004-04-22
KR100723847B1 (ko) 2007-05-31
AR086485A2 (es) 2013-12-18
AR089950A2 (es) 2014-10-01

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