UY32067A - Compuestos de pirrolo-pirimidina y sus usos - Google Patents

Compuestos de pirrolo-pirimidina y sus usos

Info

Publication number
UY32067A
UY32067A UY0001032067A UY32067A UY32067A UY 32067 A UY32067 A UY 32067A UY 0001032067 A UY0001032067 A UY 0001032067A UY 32067 A UY32067 A UY 32067A UY 32067 A UY32067 A UY 32067A
Authority
UY
Uruguay
Prior art keywords
pirrolo
compounds
need
pyrimidine compounds
cdk8
Prior art date
Application number
UY0001032067A
Other languages
English (en)
Spanish (es)
Inventor
Besong Gilbert
Christopher Thomas Brain
Clinton A Brooks
Miles Stuart Congreve
Dagostin Claudio
He Gon
Hou Ying
Howard Steven
Li Yue
Lu Yipin
Mortenson Paul
Smith Troy
Sung Moo
Woodhead Steven
Wrona Wojciech
Original Assignee
Novartis Ag
Astex Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41171100&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY32067(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag, Astex Therapeutics Ltd filed Critical Novartis Ag
Priority to UY0001038935A priority Critical patent/UY38935A/es
Publication of UY32067A publication Critical patent/UY32067A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
UY0001032067A 2008-08-22 2009-08-21 Compuestos de pirrolo-pirimidina y sus usos UY32067A (es)

Priority Applications (1)

Application Number Priority Date Filing Date Title
UY0001038935A UY38935A (es) 2008-08-22 2009-08-21 Compuestos de pirrolo-pirimidina y sus usos

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US9103708P 2008-08-22 2008-08-22

Publications (1)

Publication Number Publication Date
UY32067A true UY32067A (es) 2010-03-26

Family

ID=41171100

Family Applications (2)

Application Number Title Priority Date Filing Date
UY0001032067A UY32067A (es) 2008-08-22 2009-08-21 Compuestos de pirrolo-pirimidina y sus usos
UY0001038935A UY38935A (es) 2008-08-22 2009-08-21 Compuestos de pirrolo-pirimidina y sus usos

Family Applications After (1)

Application Number Title Priority Date Filing Date
UY0001038935A UY38935A (es) 2008-08-22 2009-08-21 Compuestos de pirrolo-pirimidina y sus usos

Country Status (48)

Country Link
US (8) US8685980B2 (enExample)
EP (2) EP2716643A1 (enExample)
JP (2) JP5560496B2 (enExample)
KR (2) KR20130140222A (enExample)
CN (2) CN102186856B (enExample)
AR (2) AR073116A1 (enExample)
AU (1) AU2009284098B2 (enExample)
BR (1) BRPI0917791B1 (enExample)
CA (1) CA2734802C (enExample)
CL (1) CL2011000306A1 (enExample)
CO (1) CO6341561A2 (enExample)
CR (1) CR20110101A (enExample)
CU (1) CU24062B1 (enExample)
CY (2) CY1115703T1 (enExample)
DK (1) DK2331547T3 (enExample)
DO (1) DOP2011000057A (enExample)
EA (1) EA019094B1 (enExample)
EC (1) ECSP11010843A (enExample)
ES (1) ES2522346T3 (enExample)
FR (1) FR17C1059I2 (enExample)
GE (1) GEP20135785B (enExample)
HN (1) HN2011000542A (enExample)
HR (1) HRP20141018T1 (enExample)
HU (1) HUS1700051I1 (enExample)
IL (1) IL211164A (enExample)
JO (1) JO2924B1 (enExample)
LT (1) LTC2331547I2 (enExample)
LU (1) LUC00048I2 (enExample)
MA (1) MA32555B1 (enExample)
ME (1) ME01282B (enExample)
MX (1) MX2011001879A (enExample)
MY (1) MY150560A (enExample)
NI (1) NI201100042A (enExample)
NL (1) NL300909I2 (enExample)
NO (1) NO2017059I1 (enExample)
NZ (1) NZ591176A (enExample)
PE (1) PE20110419A1 (enExample)
PL (1) PL2331547T3 (enExample)
PT (1) PT2331547E (enExample)
RS (1) RS53574B1 (enExample)
SI (1) SI2331547T1 (enExample)
SM (1) SMT201500017B (enExample)
TN (1) TN2011000062A1 (enExample)
TW (1) TWI468409B (enExample)
UA (1) UA103628C2 (enExample)
UY (2) UY32067A (enExample)
WO (1) WO2010020675A1 (enExample)
ZA (1) ZA201100994B (enExample)

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