SK284868B6 - 1-Ar(alk)ylimidazolín-2-óny, spôsob ich prípravy, ich použitie a farmaceutický prostriedok s ich obsahom - Google Patents

1-Ar(alk)ylimidazolín-2-óny, spôsob ich prípravy, ich použitie a farmaceutický prostriedok s ich obsahom Download PDF

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Publication number
SK284868B6
SK284868B6 SK216-98A SK21698A SK284868B6 SK 284868 B6 SK284868 B6 SK 284868B6 SK 21698 A SK21698 A SK 21698A SK 284868 B6 SK284868 B6 SK 284868B6
Authority
SK
Slovakia
Prior art keywords
alk
ylimidazolin
chlorophenyl
morpholinoimidazolin
alkyl
Prior art date
Application number
SK216-98A
Other languages
English (en)
Slovak (sk)
Other versions
SK21698A3 (en
Inventor
Hans-Joachim Lankau
Manfred Menzer
Klaus Unverferth
Karl Gewald
Harry Sch�Fer
Original Assignee
Elbion Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7771261&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK284868(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Elbion Ag filed Critical Elbion Ag
Publication of SK21698A3 publication Critical patent/SK21698A3/sk
Publication of SK284868B6 publication Critical patent/SK284868B6/sk

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88Nitrogen atoms, e.g. allantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
SK216-98A 1995-09-05 1996-07-26 1-Ar(alk)ylimidazolín-2-óny, spôsob ich prípravy, ich použitie a farmaceutický prostriedok s ich obsahom SK284868B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19532668A DE19532668A1 (de) 1995-09-05 1995-09-05 Neue, antikonvulsiv wirkende 1-Ar(alk)yl-imidazolin-2-one, die in 4-Stellung einen disubstituierten Amin-Rest enthalten, und Verfahren zu deren Herstellung
PCT/EP1996/003295 WO1997009314A1 (fr) 1995-09-05 1996-07-26 Nouvelles 1-ar(alk)yl-imidazolin-2-ones a effet anticonvulsif contenant un reste amine bisubstitue en position 4 et procede permettant de les preparer

Publications (2)

Publication Number Publication Date
SK21698A3 SK21698A3 (en) 1998-10-07
SK284868B6 true SK284868B6 (sk) 2006-01-05

Family

ID=7771261

Family Applications (1)

Application Number Title Priority Date Filing Date
SK216-98A SK284868B6 (sk) 1995-09-05 1996-07-26 1-Ar(alk)ylimidazolín-2-óny, spôsob ich prípravy, ich použitie a farmaceutický prostriedok s ich obsahom

Country Status (32)

Country Link
EP (1) EP0863880B1 (fr)
JP (1) JP4030578B2 (fr)
CN (1) CN1103762C (fr)
AR (1) AR003502A1 (fr)
AT (1) ATE254606T1 (fr)
AU (1) AU700602B2 (fr)
BG (1) BG63917B1 (fr)
BR (1) BR9610359A (fr)
CA (1) CA2184871C (fr)
CZ (1) CZ291839B6 (fr)
DE (2) DE19532668A1 (fr)
DK (1) DK0863880T3 (fr)
EA (1) EA000535B1 (fr)
EE (1) EE03562B1 (fr)
ES (1) ES2208758T3 (fr)
FR (1) FR13C0049I2 (fr)
GE (1) GEP20022652B (fr)
HK (1) HK1015776A1 (fr)
HU (1) HU225956B1 (fr)
IL (1) IL123333A (fr)
LT (1) LT4482B (fr)
LU (1) LU92263I2 (fr)
NO (1) NO313829B1 (fr)
NZ (1) NZ315624A (fr)
PL (1) PL188287B1 (fr)
PT (1) PT863880E (fr)
SK (1) SK284868B6 (fr)
TR (1) TR199800476T1 (fr)
TW (1) TW422838B (fr)
UA (1) UA46790C2 (fr)
WO (1) WO1997009314A1 (fr)
ZA (1) ZA967014B (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19721580A1 (de) * 1997-05-23 1998-11-26 Dresden Arzneimittel Verwendung von 1-Ar(alk)yl-imidazolin-2-one zur Behandlung von Angst- und Spannungszuständen
US20050070537A1 (en) 2002-10-10 2005-03-31 Chris Rundfeldt Use of dihydroimidazolones for the treatment of dogs
EP2027856A1 (fr) * 2003-07-11 2009-02-25 Boehringer Ingelheim Vetmedica Gmbh Procédé de traitement ou de prévention des troubles d système nerveux central avec des composants disposant d'un récepteur de benzodiazépine sélectif
EP2093218A1 (fr) * 2008-02-22 2009-08-26 Ruggero Fariello Imidazolidinones substitués d'arylalkyl
JP2014521713A (ja) 2011-08-12 2014-08-28 ベーリンガー インゲルハイム フェトメディカ ゲゼルシャフト ミット ベシュレンクテル ハフツング 味をマスキングした医薬組成物
US9820988B2 (en) 2014-03-24 2017-11-21 Boehringer Ingelheim Vetmedica Gmbh Treatment of epileptic disorders in feline animals
IT202100000782A1 (it) 2021-01-18 2022-07-18 Procos Spa Processo per la sintesi di imepitoina

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4044021A (en) * 1971-10-21 1977-08-23 American Cyanamid Company Tetrasubstituted imidazolidine diuretics useful in the treatment of hyperaldosteronism
BE790380A (fr) 1971-10-21 1973-04-20 American Cyanamid Co Nouvelles (p-chloro) phenyl-1 methyl-3 imidazolidines, 2,4-disubstituees utiles notamment comme agents diuretiques antialdosterone et leur procede de preparation
US3932452A (en) * 1975-02-07 1976-01-13 Morton-Norwich Products, Inc. 1-Arylmethyl-2-imidazolidinones

Also Published As

Publication number Publication date
CA2184871C (fr) 2001-08-21
AU6737596A (en) 1997-03-27
LT98047A (en) 1998-10-26
UA46790C2 (uk) 2002-06-17
TR199800476T1 (xx) 1998-06-22
AU700602B2 (en) 1999-01-07
CA2184871A1 (fr) 1997-03-06
WO1997009314A1 (fr) 1997-03-13
CZ291839B6 (cs) 2003-06-18
ES2208758T3 (es) 2004-06-16
ZA967014B (en) 1997-08-18
EE03562B1 (et) 2001-12-17
EP0863880B1 (fr) 2003-11-19
PL188287B1 (pl) 2005-01-31
SK21698A3 (en) 1998-10-07
GEP20022652B (en) 2002-03-25
BG63917B1 (bg) 2003-06-30
DE59610827D1 (de) 2003-12-24
EP0863880A1 (fr) 1998-09-16
BG102287A (en) 1998-09-30
IL123333A (en) 2001-10-31
NO980906D0 (no) 1998-03-02
HK1015776A1 (en) 1999-10-22
PT863880E (pt) 2004-04-30
NZ315624A (en) 1998-11-25
ATE254606T1 (de) 2003-12-15
NO980906L (no) 1998-03-02
CN1200728A (zh) 1998-12-02
EA000535B1 (ru) 1999-10-28
EA199800271A1 (ru) 1998-10-29
LU92263I2 (fr) 2013-10-07
BR9610359A (pt) 1999-07-06
JPH11512101A (ja) 1999-10-19
HU225956B1 (en) 2008-01-28
DK0863880T3 (da) 2004-03-22
CZ66198A3 (cs) 1998-07-15
CN1103762C (zh) 2003-03-26
TW422838B (en) 2001-02-21
FR13C0049I1 (fr) 2013-09-27
EE9800063A (et) 1998-08-17
IL123333A0 (en) 1998-09-24
JP4030578B2 (ja) 2008-01-09
FR13C0049I2 (fr) 2014-03-28
AR003502A1 (es) 1998-08-05
LT4482B (lt) 1999-03-25
HUP9802941A2 (hu) 1999-09-28
HUP9802941A3 (en) 1999-10-28
PL325413A1 (en) 1998-07-20
NO313829B1 (no) 2002-12-09
MX9801742A (es) 1998-08-30
DE19532668A1 (de) 1997-03-06

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PC4A Assignment and transfer of rights

Owner name: BIOTIE THERAPIES GMBH, RADEBEUL, DE

Free format text: FORMER OWNER: ELBION AG, RADEBEUL, DE

Effective date: 20110426

PC4A Assignment and transfer of rights

Owner name: BIOCREA GMBH, RADEBEUL, DE

Free format text: FORMER OWNER: BIOTIE THERAPIES GMBH, RADEBEUL, DE

Effective date: 20110407

MK4A Patent expired

Expiry date: 20160726