SI3456717T1 - 4,6-diamino-kinolin-3-karbonitrilni derivat kot modulator cancer osaka thyroid (COT) za zdravljenje vnetne bolezni - Google Patents

4,6-diamino-kinolin-3-karbonitrilni derivat kot modulator cancer osaka thyroid (COT) za zdravljenje vnetne bolezni

Info

Publication number
SI3456717T1
SI3456717T1 SI201631197T SI201631197T SI3456717T1 SI 3456717 T1 SI3456717 T1 SI 3456717T1 SI 201631197 T SI201631197 T SI 201631197T SI 201631197 T SI201631197 T SI 201631197T SI 3456717 T1 SI3456717 T1 SI 3456717T1
Authority
SI
Slovenia
Prior art keywords
cot
diamino
quinoline
modulator
inflammatory disease
Prior art date
Application number
SI201631197T
Other languages
English (en)
Slovenian (sl)
Inventor
Elizabeth M. Bacon
Gayatri Balan
Chien-Hung Chou
Christopher T. Clark
Jeromy J. Cottell
Musong Kim
Thorsten A. Kirschberg
John O. Link
Gary Phillips
Scott D. Schroeder
Neil H. Squires
Kirk L. Stevens
James G. Taylor
William J. Watkins
Nathan E. Wright
Sheila M. Zipfel
Original Assignee
Gilead Sciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Publication of SI3456717T1 publication Critical patent/SI3456717T1/sl

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    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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SI201631197T 2015-07-06 2016-06-30 4,6-diamino-kinolin-3-karbonitrilni derivat kot modulator cancer osaka thyroid (COT) za zdravljenje vnetne bolezni SI3456717T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562189158P 2015-07-06 2015-07-06
US201562269060P 2015-12-17 2015-12-17
EP18186568.4A EP3456717B1 (en) 2015-07-06 2016-06-30 4,6-diamino-quinoline-3-carbonitrile derivative as cancer osaka thyroid (cot) modulator for treating inflammatory disease

Publications (1)

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SI3456717T1 true SI3456717T1 (sl) 2021-08-31

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ID=56411943

Family Applications (3)

Application Number Title Priority Date Filing Date
SI201631197T SI3456717T1 (sl) 2015-07-06 2016-06-30 4,6-diamino-kinolin-3-karbonitrilni derivat kot modulator cancer osaka thyroid (COT) za zdravljenje vnetne bolezni
SI201631907T SI3896064T1 (sl) 2015-07-06 2016-06-30 4,6-diamino-kinolin-3-karbonitrilni derivati kot modulatorji raka osaka thyroid (cot) za zdravljenje crohnove bolezni in ulceroznega kolitisa
SI201630202T SI3191470T1 (sl) 2015-07-06 2016-06-30 Modulatorji COT in postopki njihove uporabe

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Application Number Title Priority Date Filing Date
SI201631907T SI3896064T1 (sl) 2015-07-06 2016-06-30 4,6-diamino-kinolin-3-karbonitrilni derivati kot modulatorji raka osaka thyroid (cot) za zdravljenje crohnove bolezni in ulceroznega kolitisa
SI201630202T SI3191470T1 (sl) 2015-07-06 2016-06-30 Modulatorji COT in postopki njihove uporabe

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US (8) US20170008905A1 (enExample)
EP (4) EP3896064B1 (enExample)
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PH12018500031B1 (en) 2018-07-09
PT3896064T (pt) 2025-07-03
MA39422B1 (fr) 2019-03-29
ES2734713T3 (es) 2019-12-11
EP4613332A2 (en) 2025-09-10
KR20180022982A (ko) 2018-03-06
WO2017007689A1 (en) 2017-01-12
MX2017004737A (es) 2017-06-19
TWI699361B (zh) 2020-07-21
EP3456717B1 (en) 2021-03-17
UY36771A (es) 2017-01-31
KR20190045416A (ko) 2019-05-02
LT3191470T (lt) 2019-05-10
AU2020257055A1 (en) 2020-11-12
CN114380799A (zh) 2022-04-22
KR20220129667A (ko) 2022-09-23
CA2971640A1 (en) 2017-01-12

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