SG186077A1 - The use of inhibitors of bruton's tyrosine kinase (btk) - Google Patents

The use of inhibitors of bruton's tyrosine kinase (btk) Download PDF

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Publication number
SG186077A1
SG186077A1 SG2012087243A SG2012087243A SG186077A1 SG 186077 A1 SG186077 A1 SG 186077A1 SG 2012087243 A SG2012087243 A SG 2012087243A SG 2012087243 A SG2012087243 A SG 2012087243A SG 186077 A1 SG186077 A1 SG 186077A1
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SG
Singapore
Prior art keywords
inhibitor
cells
cancer treatment
treatment regimen
substituted
Prior art date
Application number
SG2012087243A
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English (en)
Inventor
Joseph J Buggy
Laurence Elias
Gwen Fyfe
Eric Hedrick
David J Loury
Tarak D Mody
Original Assignee
Pharmacyclics Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45067334&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG186077(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Inc filed Critical Pharmacyclics Inc
Publication of SG186077A1 publication Critical patent/SG186077A1/en

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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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