SG11201700776XA - Compounds active towards bromodomains - Google Patents

Compounds active towards bromodomains

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Publication number
SG11201700776XA
SG11201700776XA SG11201700776XA SG11201700776XA SG11201700776XA SG 11201700776X A SG11201700776X A SG 11201700776XA SG 11201700776X A SG11201700776X A SG 11201700776XA SG 11201700776X A SG11201700776X A SG 11201700776XA SG 11201700776X A SG11201700776X A SG 11201700776XA
Authority
SG
Singapore
Prior art keywords
bromodomains
compounds active
active towards
towards
compounds
Prior art date
Application number
SG11201700776XA
Other languages
English (en)
Inventor
Seitzberg Jimmi Gerner
Akinleminu Kronborg Tine Titilola
Visnja Poljak
Gitte Friberg
Lene Teuber
Original Assignee
Nuevolution As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nuevolution As filed Critical Nuevolution As
Publication of SG11201700776XA publication Critical patent/SG11201700776XA/en

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    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08—Bridged systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4704—2-Quinolinones, e.g. carbostyril
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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