MA40551A - Composés actifs envers des bromodomaines - Google Patents
Composés actifs envers des bromodomainesInfo
- Publication number
- MA40551A MA40551A MA040551A MA40551A MA40551A MA 40551 A MA40551 A MA 40551A MA 040551 A MA040551 A MA 040551A MA 40551 A MA40551 A MA 40551A MA 40551 A MA40551 A MA 40551A
- Authority
- MA
- Morocco
- Prior art keywords
- bromodomains
- active against
- compounds active
- compounds
- against bromodomains
- Prior art date
Links
- 102000001805 Bromodomains Human genes 0.000 title 1
- 108050009021 Bromodomains Proteins 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4704—2-Quinolinones, e.g. carbostyril
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- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
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- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- 2015-07-29 US US15/501,058 patent/US10752640B2/en active Active
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- 2015-07-29 EP EP15744908.3A patent/EP3174868B1/fr active Active
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- 2015-07-29 CN CN201580041641.4A patent/CN106573915B/zh active Active
- 2015-07-29 DK DK15744908.3T patent/DK3174868T3/da active
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- 2015-07-29 BR BR112017002053-0A patent/BR112017002053A2/pt active Search and Examination
- 2015-07-29 SG SG11201700776XA patent/SG11201700776XA/en unknown
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- 2015-07-29 MA MA040551A patent/MA40551A/fr unknown
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CA2956871C (fr) | 2021-05-18 |
SG10201900631TA (en) | 2019-02-27 |
BR112017002053A2 (pt) | 2018-01-30 |
CA2956871A1 (fr) | 2016-02-04 |
CO2017001994A2 (es) | 2017-05-19 |
NZ729136A (en) | 2021-01-29 |
AU2015295405B2 (en) | 2020-04-09 |
ES2896400T3 (es) | 2022-02-24 |
MY187540A (en) | 2021-09-28 |
EP3174868A1 (fr) | 2017-06-07 |
DK3174868T3 (da) | 2021-11-08 |
AU2015295405A1 (en) | 2017-03-09 |
KR20230133395A (ko) | 2023-09-19 |
EP3174868B1 (fr) | 2021-08-25 |
RU2017104510A3 (fr) | 2019-02-11 |
RU2017104510A (ru) | 2018-09-03 |
CL2017000240A1 (es) | 2017-10-06 |
SG11201700776XA (en) | 2017-02-27 |
US10752640B2 (en) | 2020-08-25 |
IL250320A0 (en) | 2017-03-30 |
ZA201700670B (en) | 2020-07-29 |
KR102633122B1 (ko) | 2024-02-05 |
JP2017522346A (ja) | 2017-08-10 |
JP6759514B2 (ja) | 2020-09-23 |
CN106573915B (zh) | 2020-12-25 |
KR20170038877A (ko) | 2017-04-07 |
US20170349607A1 (en) | 2017-12-07 |
IL250320B (en) | 2022-02-01 |
WO2016016316A1 (fr) | 2016-02-04 |
CN106573915A (zh) | 2017-04-19 |
RU2743074C2 (ru) | 2021-02-15 |
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