LT3331885T - Junginiai - Google Patents

Junginiai

Info

Publication number
LT3331885T
LT3331885T LTEP16747519.3T LT16747519T LT3331885T LT 3331885 T LT3331885 T LT 3331885T LT 16747519 T LT16747519 T LT 16747519T LT 3331885 T LT3331885 T LT 3331885T
Authority
LT
Lithuania
Prior art keywords
compounds
Prior art date
Application number
LTEP16747519.3T
Other languages
English (en)
Inventor
Stephen Brand
PeterGeorge DODD
Eun Jung Ko
Maria Marco Martin
Timothy James Miles
Lars Henrik SANDBERG
Michael George Thomas
Stephen Thompson
Original Assignee
Glaxosmithkline Intellectual Property Development Limited
University Of Dundee
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Intellectual Property Development Limited, University Of Dundee filed Critical Glaxosmithkline Intellectual Property Development Limited
Publication of LT3331885T publication Critical patent/LT3331885T/lt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
LTEP16747519.3T 2015-08-07 2016-08-03 Junginiai LT3331885T (lt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP15382418 2015-08-07
PCT/EP2016/068592 WO2017025416A1 (en) 2015-08-07 2016-08-03 Compounds

Publications (1)

Publication Number Publication Date
LT3331885T true LT3331885T (lt) 2021-02-25

Family

ID=53887051

Family Applications (1)

Application Number Title Priority Date Filing Date
LTEP16747519.3T LT3331885T (lt) 2015-08-07 2016-08-03 Junginiai

Country Status (26)

Country Link
US (1) US10479792B2 (lt)
EP (1) EP3331885B1 (lt)
JP (1) JP6838045B2 (lt)
KR (1) KR102652898B1 (lt)
CN (1) CN108137599B (lt)
AR (1) AR105606A1 (lt)
AU (1) AU2016307230B2 (lt)
BR (1) BR112018002597B1 (lt)
CA (1) CA2994997C (lt)
CY (1) CY1124151T1 (lt)
DK (1) DK3331885T3 (lt)
ES (1) ES2856899T3 (lt)
HR (1) HRP20210402T1 (lt)
HU (1) HUE052932T2 (lt)
IL (1) IL257336B (lt)
LT (1) LT3331885T (lt)
MY (1) MY197042A (lt)
PL (1) PL3331885T3 (lt)
PT (1) PT3331885T (lt)
RS (1) RS61434B1 (lt)
RU (1) RU2734877C2 (lt)
SI (1) SI3331885T1 (lt)
SM (1) SMT202100147T1 (lt)
TW (1) TWI746454B (lt)
WO (1) WO2017025416A1 (lt)
ZA (1) ZA201800733B (lt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JOP20190278A1 (ar) * 2017-05-31 2019-11-28 Novartis Ag مركبات 5، 6-ثنائية الحلقة مندمجة وتركيبات لعلاج الأمراض الطفيلية
EA039324B1 (ru) * 2017-11-06 2022-01-13 Новартис Аг 5,6–конденсированные бициклические соединения и композиции для лечения паразитарных заболеваний
RU2717960C1 (ru) * 2019-08-05 2020-03-27 Федеральное Государственное бюджетное учреждение "27 Научный центр" Министерства обороны Российской Федерации СПОСОБ ПОЛУЧЕНИЯ ЗАМЕЩЕННЫХ α-БРОМАРИЛАЦЕТАЛЬДЕГИДОВ С ИСПОЛЬЗОВАНИЕМ БРОМИДА МЕДИ (II)
CN120641418A (zh) * 2022-10-07 2025-09-12 腾维治疗公司 化合物、组合物和方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010059418A1 (en) * 2008-11-19 2010-05-27 The Government Of The U.S.A. As Represented By The Secretary Of The Dept. Of Health & Human Services Substituted triazine and purine compounds, methods of inhibiting cruzain and rhodesain and methods of treating chagas disease and african trypanosomiasis
HUE034503T2 (en) * 2009-07-02 2018-02-28 Sanofi Sa 2,3-Dihydro-1-imidazo [1,2-a] pyrimidin-5-one derivatives, their preparation process and their use in medicine
US9233961B2 (en) * 2013-03-15 2016-01-12 Novartis Ag Compounds and compositions for the treatment of parasitic diseases
US9296754B2 (en) 2013-03-15 2016-03-29 Novartis Ag Compounds and compositions for the treatment of parasitic diseases
WO2014151729A1 (en) * 2013-03-15 2014-09-25 Irm Llc Compounds and compositions for the treatment of parasitic diseases
UY35400A (es) * 2013-03-15 2014-10-31 Novartis Ag Compuestos y composiciones para el tratamiento de enfermedades parasitarias
RS58053B1 (sr) * 2013-12-19 2019-02-28 Novartis Ag [1,2,4] triazolo [1,5-a] pirimidin derivati kao proteazomski inhibitori protozoa za tretman parazitskih bolesti kao što je lišmanijaza

Also Published As

Publication number Publication date
WO2017025416A1 (en) 2017-02-16
IL257336B (en) 2020-11-30
CN108137599B (zh) 2020-10-27
JP2018522058A (ja) 2018-08-09
CA2994997A1 (en) 2017-02-16
MY197042A (en) 2023-05-22
IL257336A (en) 2018-03-29
PT3331885T (pt) 2021-02-11
RU2734877C2 (ru) 2020-10-23
SMT202100147T1 (it) 2021-05-07
CA2994997C (en) 2023-10-10
BR112018002597A8 (pt) 2020-04-07
TWI746454B (zh) 2021-11-21
EP3331885A1 (en) 2018-06-13
AU2016307230A1 (en) 2018-02-22
RU2018107657A (ru) 2019-09-09
ES2856899T3 (es) 2021-09-28
US20180222911A1 (en) 2018-08-09
HRP20210402T1 (hr) 2021-04-16
JP6838045B2 (ja) 2021-03-03
RU2018107657A3 (lt) 2019-11-21
KR102652898B1 (ko) 2024-04-01
ZA201800733B (en) 2019-07-31
DK3331885T3 (da) 2021-01-18
SI3331885T1 (sl) 2021-03-31
TW201718590A (zh) 2017-06-01
BR112018002597B1 (pt) 2020-09-24
AU2016307230B2 (en) 2019-02-21
PL3331885T3 (pl) 2021-06-14
HUE052932T2 (hu) 2021-05-28
RS61434B1 (sr) 2021-03-31
CN108137599A (zh) 2018-06-08
EP3331885B1 (en) 2020-12-23
KR20180043289A (ko) 2018-04-27
US10479792B2 (en) 2019-11-19
AR105606A1 (es) 2017-10-18
CY1124151T1 (el) 2022-05-27

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