RU2199541C2 - Тиенопиримидины, способ их получения (варианты), фармацевтическая композиция и способ ее получения - Google Patents

Тиенопиримидины, способ их получения (варианты), фармацевтическая композиция и способ ее получения Download PDF

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Publication number
RU2199541C2
RU2199541C2 RU99104796/04A RU99104796A RU2199541C2 RU 2199541 C2 RU2199541 C2 RU 2199541C2 RU 99104796/04 A RU99104796/04 A RU 99104796/04A RU 99104796 A RU99104796 A RU 99104796A RU 2199541 C2 RU2199541 C2 RU 2199541C2
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RU
Russia
Prior art keywords
pyrimidine
chloro
pyridin
thieno
methylthieno
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Application number
RU99104796/04A
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English (en)
Russian (ru)
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RU99104796A (ru
Inventor
Йонас Рохус
Пьер ШЕЛЛИНГ
Франц-Вернер КЛУКСЕН
Мария Кристадлер
Original Assignee
Мерк Патент Гмбх
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Publication of RU99104796A publication Critical patent/RU99104796A/ru
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Gynecology & Obstetrics (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RU99104796/04A 1996-08-12 1997-07-30 Тиенопиримидины, способ их получения (варианты), фармацевтическая композиция и способ ее получения RU2199541C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19632423.8 1996-08-12
DE19632423A DE19632423A1 (de) 1996-08-12 1996-08-12 Thienopyrimidine

Publications (2)

Publication Number Publication Date
RU99104796A RU99104796A (ru) 2001-01-20
RU2199541C2 true RU2199541C2 (ru) 2003-02-27

Family

ID=7802392

Family Applications (1)

Application Number Title Priority Date Filing Date
RU99104796/04A RU2199541C2 (ru) 1996-08-12 1997-07-30 Тиенопиримидины, способ их получения (варианты), фармацевтическая композиция и способ ее получения

Country Status (28)

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US (1) US6110920A (cg-RX-API-DMAC7.html)
EP (1) EP0920431B1 (cg-RX-API-DMAC7.html)
JP (1) JP4405593B2 (cg-RX-API-DMAC7.html)
KR (1) KR100502271B1 (cg-RX-API-DMAC7.html)
CN (1) CN1081638C (cg-RX-API-DMAC7.html)
AR (1) AR009052A1 (cg-RX-API-DMAC7.html)
AT (1) ATE233265T1 (cg-RX-API-DMAC7.html)
AU (1) AU725227B2 (cg-RX-API-DMAC7.html)
BR (1) BR9711062A (cg-RX-API-DMAC7.html)
CA (1) CA2263561C (cg-RX-API-DMAC7.html)
CZ (1) CZ287772B6 (cg-RX-API-DMAC7.html)
DE (2) DE19632423A1 (cg-RX-API-DMAC7.html)
DK (1) DK0920431T3 (cg-RX-API-DMAC7.html)
ES (1) ES2191192T3 (cg-RX-API-DMAC7.html)
HU (1) HUP0001607A3 (cg-RX-API-DMAC7.html)
IL (1) IL128504A (cg-RX-API-DMAC7.html)
NO (1) NO990643L (cg-RX-API-DMAC7.html)
NZ (1) NZ334600A (cg-RX-API-DMAC7.html)
PL (1) PL190174B1 (cg-RX-API-DMAC7.html)
PT (1) PT920431E (cg-RX-API-DMAC7.html)
RU (1) RU2199541C2 (cg-RX-API-DMAC7.html)
SI (1) SI0920431T1 (cg-RX-API-DMAC7.html)
SK (1) SK282823B6 (cg-RX-API-DMAC7.html)
TR (1) TR199900308T2 (cg-RX-API-DMAC7.html)
TW (1) TW359672B (cg-RX-API-DMAC7.html)
UA (1) UA55421C2 (cg-RX-API-DMAC7.html)
WO (1) WO1998006722A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA977156B (cg-RX-API-DMAC7.html)

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WO1995019774A1 (en) * 1994-01-25 1995-07-27 Warner-Lambert Company Bicyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family

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US4196207A (en) * 1977-05-23 1980-04-01 Ici Australia Limited Process for controlling eradicating or preventing infestations of animals by Ixodid ticks
WO1995019774A1 (en) * 1994-01-25 1995-07-27 Warner-Lambert Company Bicyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family

Also Published As

Publication number Publication date
KR100502271B1 (ko) 2005-07-22
SK282823B6 (sk) 2002-12-03
NZ334600A (en) 2000-07-28
PL331538A1 (en) 1999-07-19
NO990643D0 (no) 1999-02-11
AR009052A1 (es) 2000-03-08
TW359672B (en) 1999-06-01
IL128504A0 (en) 2000-01-31
CA2263561C (en) 2007-02-20
ZA977156B (en) 1998-02-19
US6110920A (en) 2000-08-29
JP4405593B2 (ja) 2010-01-27
JP2000516223A (ja) 2000-12-05
EP0920431B1 (de) 2003-02-26
HUP0001607A2 (hu) 2000-10-28
BR9711062A (pt) 1999-08-17
ES2191192T3 (es) 2003-09-01
HK1021731A1 (en) 2000-06-30
AU725227B2 (en) 2000-10-12
DK0920431T3 (da) 2003-06-02
AU4203597A (en) 1998-03-06
KR20000029932A (ko) 2000-05-25
PL190174B1 (pl) 2005-11-30
IL128504A (en) 2003-01-12
EP0920431A1 (de) 1999-06-09
CN1081638C (zh) 2002-03-27
CA2263561A1 (en) 1998-02-19
CN1227560A (zh) 1999-09-01
NO990643L (no) 1999-02-11
DE19632423A1 (de) 1998-02-19
SK16499A3 (en) 1999-06-11
TR199900308T2 (xx) 1999-04-21
CZ287772B6 (en) 2001-01-17
WO1998006722A1 (de) 1998-02-19
UA55421C2 (uk) 2003-04-15
ATE233265T1 (de) 2003-03-15
DE59709404D1 (en) 2003-04-03
PT920431E (pt) 2003-07-31
SI0920431T1 (en) 2003-08-31
CZ44899A3 (cs) 1999-05-12
HUP0001607A3 (en) 2002-09-30

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Effective date: 20060731