PT2194043E - Processos - Google Patents

Processos Download PDF

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Publication number
PT2194043E
PT2194043E PT101550580T PT10155058T PT2194043E PT 2194043 E PT2194043 E PT 2194043E PT 101550580 T PT101550580 T PT 101550580T PT 10155058 T PT10155058 T PT 10155058T PT 2194043 E PT2194043 E PT 2194043E
Authority
PT
Portugal
Prior art keywords
processes
Prior art date
Application number
PT101550580T
Other languages
English (en)
Inventor
Gerald J Tanoury
John E Cochran
Minzhang Chen
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of PT2194043E publication Critical patent/PT2194043E/pt

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/14Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/468-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0802Tripeptides with the first amino acid being neutral
    • C07K5/0812Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02Linear peptides containing at least one abnormal peptide link
PT101550580T 2005-08-19 2006-08-18 Processos PT2194043E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70996405P 2005-08-19 2005-08-19
US81004206P 2006-06-01 2006-06-01

Publications (1)

Publication Number Publication Date
PT2194043E true PT2194043E (pt) 2014-03-04

Family

ID=37708299

Family Applications (2)

Application Number Title Priority Date Filing Date
PT06813568T PT1934179E (pt) 2005-08-19 2006-08-18 PROCESSOS E INTERMEDIáRIOS
PT101550580T PT2194043E (pt) 2005-08-19 2006-08-18 Processos

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PT06813568T PT1934179E (pt) 2005-08-19 2006-08-18 PROCESSOS E INTERMEDIáRIOS

Country Status (25)

Country Link
US (3) US7776887B2 (pt)
EP (4) EP2364970A1 (pt)
JP (1) JP5203203B2 (pt)
KR (4) KR20140069370A (pt)
CN (2) CN102382170A (pt)
AR (1) AR058025A1 (pt)
AT (1) ATE463480T1 (pt)
AU (1) AU2006279357B2 (pt)
BR (1) BRPI0615029A2 (pt)
CA (1) CA2619659A1 (pt)
CY (2) CY1110214T1 (pt)
DE (1) DE602006013492D1 (pt)
DK (2) DK1934179T3 (pt)
ES (2) ES2449268T3 (pt)
HK (2) HK1122801A1 (pt)
IL (2) IL189585A (pt)
NZ (3) NZ566049A (pt)
PL (3) PL385229A1 (pt)
PT (2) PT1934179E (pt)
RU (2) RU2446171C2 (pt)
SG (1) SG2014013338A (pt)
SI (2) SI1934179T1 (pt)
TW (2) TWI391376B (pt)
WO (1) WO2007022459A2 (pt)
ZA (1) ZA200801791B (pt)

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CN103450066B (zh) * 2012-05-30 2017-03-15 博瑞生物医药(苏州)股份有限公司 特拉匹韦中间体的制备方法
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PL1934179T4 (pl) 2014-03-31
TWI391376B (zh) 2013-04-01
IL228770A0 (en) 2013-12-31
DK1934179T3 (da) 2010-08-09
HK1145022A1 (en) 2011-03-25
ES2344156T3 (es) 2010-08-19
IL189585A (en) 2013-10-31
EP1934179A2 (en) 2008-06-25
PT1934179E (pt) 2010-07-12
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EP2194043A3 (en) 2010-11-24
RU2446171C2 (ru) 2012-03-27
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AU2006279357B2 (en) 2012-05-31
PL385229A1 (pl) 2008-09-29
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ZA200801791B (en) 2008-12-31
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US20070087973A1 (en) 2007-04-19
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PL1934179T3 (pl) 2010-09-30
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EP2194043B1 (en) 2013-12-25
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