NO20021111L - Anvendelse av 5-O-deoaminyl-6-O-metylerytronolid A-derivater for fremstilling av biologisk aktive produkter - Google Patents

Anvendelse av 5-O-deoaminyl-6-O-metylerytronolid A-derivater for fremstilling av biologisk aktive produkter

Info

Publication number
NO20021111L
NO20021111L NO20021111A NO20021111A NO20021111L NO 20021111 L NO20021111 L NO 20021111L NO 20021111 A NO20021111 A NO 20021111A NO 20021111 A NO20021111 A NO 20021111A NO 20021111 L NO20021111 L NO 20021111L
Authority
NO
Norway
Prior art keywords
deoaminyl
derivatives
preparation
biologically active
active products
Prior art date
Application number
NO20021111A
Other languages
English (en)
Other versions
NO20021111D0 (no
NO315048B1 (no
Inventor
Alain Bonnet
Michel Delthil
Alain Mazurie
Original Assignee
Hoechst Marion Roussel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9482423&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20021111(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Publication of NO20021111L publication Critical patent/NO20021111L/no
Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc
Publication of NO20021111D0 publication Critical patent/NO20021111D0/no
Publication of NO315048B1 publication Critical patent/NO315048B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO20021111A 1995-09-11 2002-03-06 Fremgangsmåte for fremstilling av 5-O-desosaminyl-6-O- metylerytronolid A-derivater NO315048B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9510601A FR2738571B1 (fr) 1995-09-11 1995-09-11 Nouveaux derives de la 5-0-desosaminyl 6-0-methyl- erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
PCT/FR1996/001384 WO1997010251A1 (fr) 1995-09-11 1996-09-10 Nouveaux derives de la 5-0-desosaminyl 6-0-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (3)

Publication Number Publication Date
NO20021111L true NO20021111L (no) 1998-03-10
NO20021111D0 NO20021111D0 (no) 2002-03-06
NO315048B1 NO315048B1 (no) 2003-06-30

Family

ID=9482423

Family Applications (2)

Application Number Title Priority Date Filing Date
NO19981053A NO312678B1 (no) 1995-09-11 1998-03-10 Nye 5-O-deoaminyl-6-O-metylerytronolid A-derivater, fremgangsmåte for fremstilling av disse, og mellomprodukter veddenne
NO20021111A NO315048B1 (no) 1995-09-11 2002-03-06 Fremgangsmåte for fremstilling av 5-O-desosaminyl-6-O- metylerytronolid A-derivater

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO19981053A NO312678B1 (no) 1995-09-11 1998-03-10 Nye 5-O-deoaminyl-6-O-metylerytronolid A-derivater, fremgangsmåte for fremstilling av disse, og mellomprodukter veddenne

Country Status (34)

Country Link
US (1) US5969161A (no)
EP (1) EP0854880B1 (no)
JP (1) JP4332218B2 (no)
KR (1) KR100457755B1 (no)
CN (2) CN1237069C (no)
AP (1) AP887A (no)
AR (1) AR004195A1 (no)
AT (1) ATE266035T1 (no)
AU (1) AU708811B2 (no)
BG (1) BG63822B1 (no)
BR (1) BR9610503A (no)
CA (1) CA2228670C (no)
CZ (3) CZ294866B6 (no)
DE (1) DE69632405T2 (no)
DK (1) DK0854880T3 (no)
EA (1) EA000575B1 (no)
EE (1) EE03774B1 (no)
ES (1) ES2219698T3 (no)
FR (1) FR2738571B1 (no)
GE (1) GEP20022838B (no)
HK (2) HK1016187A1 (no)
HU (1) HU227565B1 (no)
IL (1) IL123550A (no)
MX (1) MX9801859A (no)
NO (2) NO312678B1 (no)
PL (1) PL183652B1 (no)
PT (1) PT854880E (no)
RO (1) RO120137B1 (no)
SI (1) SI0854880T1 (no)
SK (3) SK285995B6 (no)
TR (1) TR199800438T1 (no)
UA (1) UA53628C2 (no)
WO (1) WO1997010251A1 (no)
ZA (1) ZA966837B (no)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100441591C (zh) * 1996-09-04 2008-12-10 艾博特公司 酮基内酯类化合物,其用途和制备方法以及药用组合物
UA51730C2 (uk) * 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
US6034069A (en) * 1997-09-30 2000-03-07 Abbott Laboratories 3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity
US6046171A (en) * 1997-10-29 2000-04-04 Abbott Laboratories 6,11-bridged erythromycin derivatives
US6124269A (en) * 1997-10-29 2000-09-26 Abbott Laboratories 2-Halo-6-O-substituted ketolide derivatives
US6054435A (en) * 1999-03-19 2000-04-25 Abbott Laboratories 6-O-substituted macrolides having antibacterial activity
US6420535B1 (en) 1999-06-07 2002-07-16 Abbott Laboratories 6-O-carbamate ketolide derivatives
EP1483277A4 (en) * 2002-02-15 2007-10-03 Merckle Gmbh CONJUGATES OF BIOLOGICALLY ACTIVE COMPOUNDS, METHODS OF PREPARATION AND USE, AND FORMULATION AND PHARMACEUTICAL APPLICATIONS
US6753318B1 (en) 2002-07-25 2004-06-22 Enanta Pharmaceuticals, Inc. 6,11-4-carbon bridged erythromycin derivatives
US6841664B2 (en) 2002-07-25 2005-01-11 Enanra Pharmaceuticals, Inc. 6,11-4-carbon bridged ketolides
US7273853B2 (en) * 2002-05-13 2007-09-25 Enanta Pharmaceuticals, Inc. 6-11 bicyclic ketolide derivatives
US6878691B2 (en) * 2002-05-13 2005-04-12 Enanta Pharmaceuticals, Inc. 6-11 bicyclic ketolide derivatives
JP2005536465A (ja) * 2002-05-13 2005-12-02 エナンタ ファーマシューティカルズ インコーポレイテッド 6,11二環式エリスロマイシン誘導体
US7064110B2 (en) * 2002-05-13 2006-06-20 Enanta Pharmaceuticals, Inc. 6-11 bicycle ketolide derivatives
US7910558B2 (en) * 2002-05-13 2011-03-22 Enanta Pharmaceuticals, Inc. Bridged macrocyclic compounds and processes for the preparation thereof
WO2005070918A1 (en) * 2002-05-13 2005-08-04 Enanta Pharmaceuticals, Inc. Process for the preparation of t-11 bicyclic erythromycin derivatives
US7135573B2 (en) * 2002-05-13 2006-11-14 Enanta Pharmaceuticals, Inc. Processes for the preparation of O-(6-Pyrazol-1-yl-pyridin-3-ylmethyl)-hydroxylamine
US6764998B1 (en) 2003-06-18 2004-07-20 Enanta Pharmaceuticals, Inc. 6,11-4C-bicyclic 9a-azalide derivatives
ITMI20021726A1 (it) * 2002-08-01 2004-02-02 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
US6645941B1 (en) 2003-03-26 2003-11-11 Enanta Pharmaceuticals, Inc. 6,11-3C-bicyclic 9a-azalide derivatives
US7276487B2 (en) * 2003-09-23 2007-10-02 Enanta Pharmaceuticals, Inc. 9a, 11-3C-bicyclic 9a-azalide derivatives
WO2005067564A2 (en) * 2004-01-07 2005-07-28 Enanta Pharmaceuticals, Inc. 6-11 bicyclic erythromycin derivatives
WO2005070113A2 (en) * 2004-01-09 2005-08-04 Enanta Pharmaceuticals, Inc. 9n-substituted 6-11 bicyclic erythromycin derivatives
JP2008522978A (ja) 2004-12-07 2008-07-03 エナンタ ファーマシューティカルズ インコーポレイテッド 3,6−ビシクロライド
US7229972B2 (en) 2004-12-07 2007-06-12 Enanta Pharmaceuticals, Inc. 3,6-Bicyclolides
WO2006065721A2 (en) 2004-12-13 2006-06-22 Enanta Pharmaceuticals, Inc. 11, 12-lactone bicyclolides
US7312201B2 (en) 2004-12-13 2007-12-25 Enanta Pharmaceuticals, Inc. Tetracyclic bicyclolides
US7384922B2 (en) * 2005-05-04 2008-06-10 Enanta Pharmaceuticals, Inc. 6-11 bridged oxime erythromycin derivatives
EP1907392A1 (en) * 2005-07-26 2008-04-09 Merckle Gmbh Macrolide conjugates of pyrrolizine and indolizine compounds as inhibitors of 5-lipooxygenase and cyclooxygenase
JP5642548B2 (ja) * 2007-09-17 2014-12-17 エナンタ ファーマシューティカルズ インコーポレイテッド 6,11−架橋ビアリールマクロライド
US8354383B2 (en) * 2007-09-17 2013-01-15 Enanta Pharmaceuticals, Inc. 6,11-bridged biaryl macrolides
US8273720B2 (en) * 2007-09-17 2012-09-25 Enanta Pharmaceuticals, Inc. 6,11-bicyclolides: bridged biaryl macrolide derivatives
CN103232501A (zh) * 2013-04-11 2013-08-07 宜昌东阳光药业股份有限公司 阿奇霉素或阿奇霉素的中间体脱去克拉定糖化合物的制备工艺

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR960000434B1 (ko) * 1986-12-17 1996-01-06 다이쇼 세이야꾸 가부시끼가이샤 에리스로마이신 a유도체 및 그의 제조 방법
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives

Also Published As

Publication number Publication date
JP4332218B2 (ja) 2009-09-16
IL123550A0 (en) 1998-10-30
PT854880E (pt) 2004-09-30
ES2219698T3 (es) 2004-12-01
HUP9802930A3 (en) 1999-12-28
CA2228670A1 (fr) 1997-03-20
EP0854880A1 (fr) 1998-07-29
BG63822B1 (bg) 2003-02-28
SK283690B6 (sk) 2003-12-02
DE69632405T2 (de) 2005-05-19
CN1237069C (zh) 2006-01-18
AP9801210A0 (en) 1998-03-31
RO120137B1 (ro) 2005-09-30
UA53628C2 (uk) 2003-02-17
KR19990044543A (ko) 1999-06-25
AP887A (en) 2000-11-10
CZ294865B6 (cs) 2005-04-13
NO981053D0 (no) 1998-03-10
CZ289945B6 (cs) 2002-04-17
WO1997010251A1 (fr) 1997-03-20
NO981053L (no) 1998-03-10
EP0854880B1 (fr) 2004-05-06
HUP9802930A1 (hu) 1999-04-28
US5969161A (en) 1999-10-19
GEP20022838B (en) 2002-11-25
EE9800065A (et) 1998-08-17
NO20021111D0 (no) 2002-03-06
SK29498A3 (en) 1998-12-02
FR2738571A1 (fr) 1997-03-14
HK1016187A1 (en) 1999-10-29
ZA966837B (en) 1997-08-13
HU227565B1 (en) 2011-08-29
TR199800438T1 (xx) 1998-05-21
HK1041489B (zh) 2006-09-08
CZ294866B6 (cs) 2005-04-13
DK0854880T3 (da) 2004-08-16
NO315048B1 (no) 2003-06-30
BR9610503A (pt) 1999-07-06
CN1070498C (zh) 2001-09-05
DE69632405D1 (de) 2004-06-09
ATE266035T1 (de) 2004-05-15
AU708811B2 (en) 1999-08-12
CZ71798A3 (cs) 1998-07-15
NO312678B1 (no) 2002-06-17
MX9801859A (es) 1998-11-30
EE03774B1 (et) 2002-06-17
SK285853B6 (sk) 2007-09-06
EA199800288A1 (ru) 1998-08-27
PL326274A1 (en) 1998-08-31
SK285995B6 (sk) 2008-01-07
AR004195A1 (es) 1998-11-04
CA2228670C (fr) 2005-04-12
HK1041489A1 (en) 2002-07-12
FR2738571B1 (fr) 1997-10-17
EA000575B1 (ru) 1999-12-29
IL123550A (en) 2002-09-12
CN1201462A (zh) 1998-12-09
SI0854880T1 (en) 2004-12-31
KR100457755B1 (ko) 2005-02-28
CN1319602A (zh) 2001-10-31
PL183652B1 (pl) 2002-06-28
JPH11512416A (ja) 1999-10-26
AU6991096A (en) 1997-04-01
BG102312A (en) 1998-09-30

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Legal Events

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