NL8400817A - Thiazolidinederivaten, werkwijze voor de bereiding ervan en farmaceutische preparaten ervan. - Google Patents

Thiazolidinederivaten, werkwijze voor de bereiding ervan en farmaceutische preparaten ervan. Download PDF

Info

Publication number
NL8400817A
NL8400817A NL8400817A NL8400817A NL8400817A NL 8400817 A NL8400817 A NL 8400817A NL 8400817 A NL8400817 A NL 8400817A NL 8400817 A NL8400817 A NL 8400817A NL 8400817 A NL8400817 A NL 8400817A
Authority
NL
Netherlands
Prior art keywords
formula
group
compound
ppm
thiazolidine
Prior art date
Application number
NL8400817A
Other languages
English (en)
Dutch (nl)
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of NL8400817A publication Critical patent/NL8400817A/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D277/10—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/18—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NL8400817A 1983-03-16 1984-03-15 Thiazolidinederivaten, werkwijze voor de bereiding ervan en farmaceutische preparaten ervan. NL8400817A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU83888A HU188852B (en) 1983-03-16 1983-03-16 Process for producing thiazolidine derivatives active against gastric ulcer and intestinal ulcer
HU88883 1983-03-16

Publications (1)

Publication Number Publication Date
NL8400817A true NL8400817A (nl) 1984-10-16

Family

ID=10951891

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8400817A NL8400817A (nl) 1983-03-16 1984-03-15 Thiazolidinederivaten, werkwijze voor de bereiding ervan en farmaceutische preparaten ervan.

Country Status (32)

Country Link
US (1) US4616025A (es)
JP (1) JPS59196877A (es)
KR (1) KR840008001A (es)
AT (1) AT383596B (es)
AU (1) AU559753B2 (es)
BE (1) BE899132A (es)
CA (1) CA1273933A (es)
CH (1) CH660592A5 (es)
CS (1) CS241074B2 (es)
DD (1) DD216929A5 (es)
DE (1) DE3409801A1 (es)
DK (1) DK143284A (es)
ES (2) ES530738A0 (es)
FI (1) FI79843C (es)
FR (1) FR2542740B1 (es)
GB (1) GB2140412B (es)
GR (1) GR81883B (es)
HU (1) HU188852B (es)
IE (1) IE57101B1 (es)
IL (1) IL71249A (es)
IN (1) IN157738B (es)
IT (1) IT1196048B (es)
LU (1) LU85248A1 (es)
NL (1) NL8400817A (es)
NO (1) NO162858C (es)
NZ (1) NZ207516A (es)
PL (2) PL142909B1 (es)
PT (1) PT78260B (es)
SE (1) SE455945B (es)
SU (2) SU1240355A3 (es)
YU (1) YU47384A (es)
ZA (1) ZA841938B (es)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6051184A (ja) * 1983-08-30 1985-03-22 Fujimoto Seiyaku Kk Ν−シアノイミノチアゾリジン誘導体およびその製造法
ATE67493T1 (de) * 1985-02-04 1991-10-15 Bayer Agrochem Kk Heterocyclische verbindungen.
JPH0730070B2 (ja) * 1985-10-03 1995-04-05 日本バイエルアグロケム株式会社 新規複素環式化合物
US5001138B1 (en) * 1985-02-04 1998-01-20 Bayer Agrochem Kk Heterocyclic compounds
JPH066585B2 (ja) * 1985-02-04 1994-01-26 日本バイエルアグロケム株式会社 ニトロメチレン誘導体、その製法及び殺虫剤
US5204360A (en) * 1985-02-04 1993-04-20 Nihon Bayer Agrochem K.K. Heterocyclic compounds
JPH0649699B2 (ja) * 1985-02-04 1994-06-29 日本バイエルアグロケム株式会社 ニトロメチレン誘導体、その製法及び殺虫剤
JPH0717621B2 (ja) * 1986-03-07 1995-03-01 日本バイエルアグロケム株式会社 新規ヘテロ環式化合物
USRE39130E1 (en) 1986-03-07 2006-06-13 Bayer Cropscience K.K. Heterocyclic compounds
JP2607369B2 (ja) * 1987-02-20 1997-05-07 興和株式会社 新規な複素環化合物
US5122522A (en) * 1989-06-21 1992-06-16 The Trustees Of The University Of Pennsylvania Treatment and control of ocular development
CA2058768C (en) * 1989-06-21 2004-08-03 Alan M. Laties Treatment and control of ocular development
HU207047B (en) * 1989-11-07 1993-03-01 Richter Gedeon Vegyeszet Process for producing new pyridine derivatives and pharmaceutical copositions comprising same
CA2063865A1 (en) * 1992-03-24 1993-09-25 Karoly Lempert 2-(substituted imino)-thiazolidines and process for the preparation thereof
JP2721805B2 (ja) * 1994-07-22 1998-03-04 日本バイエルアグロケム株式会社 新規ヘテロ環式化合物
DE4427539A1 (de) * 1994-08-04 1996-02-08 Sueddeutsche Kalkstickstoff Verfahren zur Herstellung von 2-Cyaniminothiazolidin
DE4427569A1 (de) * 1994-08-04 1996-02-08 Bayer Ag Verfahren zur Herstellung von Cyanimino-1,3-thiazolidin
DE19904310A1 (de) 1999-01-28 2000-08-03 Bayer Ag Verfahren zur Herstellung heterocyclischer Verbindungen
CN1198803C (zh) * 1999-03-05 2005-04-27 第一三得利制药株式会社 具有激活烟碱性乙酰胆碱α4β2受体作用的杂环化合物
KR20040018380A (ko) * 2001-05-25 2004-03-03 밸리 포지 파마슈티컬즈, 인크. 피렌제핀 안약 겔제
EA008865B1 (ru) * 2002-11-22 2007-08-31 Смитклайн Бичам Корпорейшн Производные 2-имино-4-оксотиазолидина
CA2521606A1 (en) * 2003-04-07 2004-10-21 Cortical Pty Ltd. Novel methods for the treatment of inflammatory diseases
US8309733B2 (en) 2008-07-01 2012-11-13 Meji Seika Pharma Co., Ltd. Imino derivatives, methods for producing the same and insecticides containing the same
CN103797008B (zh) * 2011-09-02 2016-08-17 拜耳知识产权有限责任公司 用于制备[3-[(6-氯-3-吡啶基)甲基]-2-噻唑烷亚基]氰胺的方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3264316A (en) * 1963-09-18 1966-08-02 Res Lab Dr C Janssen N V Certain 2-acylimino-3-substitutedthiazoline-4 compounds
DE2205745A1 (de) * 1972-02-08 1973-08-23 Thomae Gmbh Dr K Neue durch den n-cyaniminorest substituierten heterocyclen und verfahren zu ihrer herstellung
US4006156A (en) * 1975-06-27 1977-02-01 Shell Oil Company 3-Alkyl-2-(nitromethylene) thiazolidine
DK173777A (da) * 1976-05-03 1977-11-04 Merck & Co Inc Fremgangsmade til fremstilling af derivater af 2-iminothiazolidiner og thiazoliner
JPS57171986A (en) * 1981-04-14 1982-10-22 Taiho Yakuhin Kogyo Kk Heterocylic ring compound containing sulfur
JPS5823682A (ja) * 1981-08-03 1983-02-12 Santen Pharmaceut Co Ltd 複素五員環化合物
DE3133918A1 (de) * 1981-08-27 1983-03-17 Bayer Ag, 5090 Leverkusen 2-arylhydrazino-2-thiazoline, acylderivate derselben, 2-arylazo-2-thiazoline, herstellungsverfahren und ihre verwendung zur bekaempfung von ekto- und endoparasiten
JPS58222886A (ja) * 1982-06-19 1983-12-24 Ricoh Co Ltd 感熱記録シ−ト
JPS5933267A (ja) * 1982-08-19 1984-02-23 Fujimoto Seiyaku Kk グアニジン誘導体およびその製造法

Also Published As

Publication number Publication date
SE8401463L (sv) 1984-09-17
PT78260B (en) 1986-04-30
IT1196048B (it) 1988-11-10
GR81883B (es) 1984-12-12
NO162858C (no) 1990-02-28
YU47384A (es) 1986-10-31
HU188852B (en) 1986-05-28
GB2140412A (en) 1984-11-28
IE840655L (en) 1984-09-16
CS188584A2 (en) 1985-06-13
PL142909B1 (en) 1987-12-31
ES8601170A1 (es) 1985-11-01
FI841066A (fi) 1984-09-17
IL71249A (en) 1987-02-27
US4616025A (en) 1986-10-07
AU559753B2 (en) 1987-03-19
ZA841938B (en) 1985-05-29
BE899132A (fr) 1984-09-12
SU1240355A3 (ru) 1986-06-23
SE455945B (sv) 1988-08-22
PL252129A1 (en) 1985-11-19
DK143284D0 (da) 1984-02-29
ES8604179A1 (es) 1986-01-16
NO841002L (no) 1984-09-17
ES530738A0 (es) 1985-11-01
FR2542740A1 (fr) 1984-09-21
IT8420057A0 (it) 1984-03-15
FR2542740B1 (fr) 1987-02-20
JPS59196877A (ja) 1984-11-08
AU2583384A (en) 1984-09-20
IN157738B (es) 1986-05-31
PL142749B1 (en) 1987-11-30
ATA88284A (de) 1986-12-15
CA1273933A (en) 1990-09-11
DE3409801A1 (de) 1984-09-20
FI79843B (fi) 1989-11-30
CH660592A5 (de) 1987-05-15
PT78260A (en) 1984-04-01
IL71249A0 (en) 1984-06-29
NO162858B (no) 1989-11-20
PL246683A1 (en) 1985-07-16
SE8401463D0 (sv) 1984-03-15
CS241074B2 (en) 1986-03-13
FI79843C (fi) 1990-03-12
FI841066A0 (fi) 1984-03-16
ES544286A0 (es) 1986-01-16
KR840008001A (ko) 1984-12-12
LU85248A1 (fr) 1985-10-14
DK143284A (da) 1984-09-17
AT383596B (de) 1987-07-27
GB2140412B (en) 1987-02-11
DD216929A5 (de) 1985-01-02
SU1240356A3 (ru) 1986-06-23
NZ207516A (en) 1986-06-11
IE57101B1 (en) 1992-04-22
GB8406790D0 (en) 1984-04-18

Similar Documents

Publication Publication Date Title
NL8400817A (nl) Thiazolidinederivaten, werkwijze voor de bereiding ervan en farmaceutische preparaten ervan.
US5252580A (en) Indole derivatives and anti-ulcer compositions thereof
EP0116769B1 (en) Dihydropyridines
JPS597703B2 (ja) ピリジン誘導体の製造方法
EP0254588A1 (en) Imidazo[4,5-b] pyridine compounds, process for preparing same and pharmaceutical compositions containing same
GB2243832A (en) 2-substituted 4-acetamido-5-chloro-n-[2-(diethylamino)ethyl]-benzamide derivative
KR900000552B1 (ko) 항알레르기 및 소염 제제와 그의 제조방법
JPH0390062A (ja) 置換ｎ―（キノリン―２―イル―メトキシ）ベンジルスルホニルウレア
JPH07278148A (ja) イミダゾピラゾール誘導体
JPS6019767A (ja) カルボスチリル誘導体を有効成分とする抗潰瘍剤
US4187303A (en) Thiazine derivatives
PL179032B1 (pl) kwasu hydroksamowego oraz kompozycje farmaceutyczne zawierajace nowe pochodnekwasu hydroksamowego PL PL
US4152440A (en) Novel derivatives of imidazole, and pharmaceutical compositions containing them
US4713388A (en) Certain 3- or 4-benzoyl-2-[(2-aminoethyl)thio-pyridines] and their anti-ulcer properties
JPH0625151B2 (ja) ２−置換シクロヘプトイミダゾ−ル誘導体、抗潰瘍剤及びその製造方法
EP0074229B1 (en) Triazole gastric anti-secretory agents
US4213986A (en) Novel derivatives of imidazole and pharmaceutical compositions containing them and method of use
JPH0753730B2 (ja) イミダゾピラゾール誘導体
JP2794640B2 (ja) イミダゾール誘導体およびその製造法ならびにこれを含有する抗潰瘍剤
US4276297A (en) Pyridylaminotriazole therapeutic agents
NL8201264A (nl) 1-oxo-2h-isochinolinen en zuuradditie-zouten daarvan, en preparaten die ze bevatten.
IE51110B1 (en) 4-hydroxy-1,2-benzisothiazol-3(2h)-one-1.1-dioxide
JPS5951542B2 (ja) ５−フエニル−チアゾリジン−４−オン誘導体の製造方法
IL95091A (en) History of 3,4-dihydro-6,8-similar acid H-6H2-pyrimido, B-1 [] 1,3 [] 2H HTZHI-7 carboxylic acid, preparation and pharmaceutical preparations
JPS6125035B2 (es)

Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BI The patent application has been withdrawn