US6541498B2
(en)
|
1993-05-20 |
2003-04-01 |
Texas Biotechnology |
Benzenesulfonamides and the use thereof to modulate the activity of endothelin
|
ES2318899T3
(es)
*
|
1998-07-06 |
2009-05-01 |
Bristol-Myers Squibb Company |
Bifenil sulfonamidas como antagonistas duales de los receptores de angiotensina y endotelina.
|
MY125533A
(en)
|
1999-12-06 |
2006-08-30 |
Bristol Myers Squibb Co |
Heterocyclic dihydropyrimidine compounds
|
DE60030764T2
(de)
*
|
1999-12-15 |
2007-09-13 |
Bristol-Myers Squibb Co. |
Biphenyl - sulfonamide als duale angiotensin - endothelin - rezeptor - antagonisten
|
WO2001049289A1
(en)
*
|
1999-12-31 |
2001-07-12 |
Texas Biotechnology Corporation |
Pharmaceutical and veterinary uses of endothelin antagonists
|
US6271228B1
(en)
*
|
2000-04-28 |
2001-08-07 |
Pfizer Inc. |
Blood pressure stabilization during hemodialysis
|
US7622503B2
(en)
|
2000-08-24 |
2009-11-24 |
University Of Tennessee Research Foundation |
Selective androgen receptor modulators and methods of use thereof
|
WO2002043807A2
(en)
*
|
2000-12-01 |
2002-06-06 |
Novartis Ag |
Combinations of an angiotensin receptor antagonist and an anti-hypertensive drug or a statin, for the treatment of sexual dysfunction
|
CH1427415H1
(de)
|
2001-09-21 |
2023-12-21 |
Bristol Myers Squibb Holdings Ireland |
Lactamhaltige verbindungen und ihre derivate als faktor-xa-hemmer
|
PL377687A1
(pl)
|
2001-10-18 |
2006-02-06 |
Bristol-Myers Squibb Company |
Środki naśladujące ludzki peptyd glukagonopodobny typu 1 i ich zastosowanie w leczeniu cukrzycy i stanów związanych z cukrzycą
|
US7238671B2
(en)
|
2001-10-18 |
2007-07-03 |
Bristol-Myers Squibb Company |
Human glucagon-like-peptide-1 mimics and their use in the treatment of diabetes and related conditions
|
US8853266B2
(en)
|
2001-12-06 |
2014-10-07 |
University Of Tennessee Research Foundation |
Selective androgen receptor modulators for treating diabetes
|
US6831102B2
(en)
|
2001-12-07 |
2004-12-14 |
Bristol-Myers Squibb Company |
Phenyl naphthol ligands for thyroid hormone receptor
|
TWI328007B
(en)
|
2002-01-16 |
2010-08-01 |
Astrazeneca Ab |
Novel compounds
|
TW200307539A
(en)
|
2002-02-01 |
2003-12-16 |
Bristol Myers Squibb Co |
Cycloalkyl inhibitors of potassium channel function
|
US7435824B2
(en)
|
2002-04-19 |
2008-10-14 |
Bristol-Myers Squibb Company |
Prodrugs of potassium channel inhibitors
|
TW200403058A
(en)
|
2002-04-19 |
2004-03-01 |
Bristol Myers Squibb Co |
Heterocyclo inhibitors of potassium channel function
|
US7405234B2
(en)
|
2002-05-17 |
2008-07-29 |
Bristol-Myers Squibb Company |
Bicyclic modulators of androgen receptor function
|
US7057046B2
(en)
|
2002-05-20 |
2006-06-06 |
Bristol-Myers Squibb Company |
Lactam glycogen phosphorylase inhibitors and method of use
|
MY139563A
(en)
|
2002-09-04 |
2009-10-30 |
Bristol Myers Squibb Co |
Heterocyclic aromatic compounds useful as growth hormone secretagogues
|
WO2004037181A2
(en)
|
2002-10-23 |
2004-05-06 |
Bristol-Myers Squibb Company |
Glycinenitrile-based inhibitors of dipeptidyl peptidase iv and methods
|
US7098235B2
(en)
|
2002-11-14 |
2006-08-29 |
Bristol-Myers Squibb Co. |
Triglyceride and triglyceride-like prodrugs of glycogen phosphorylase inhibiting compounds
|
TW200504021A
(en)
|
2003-01-24 |
2005-02-01 |
Bristol Myers Squibb Co |
Substituted anilide ligands for the thyroid receptor
|
US7557143B2
(en)
|
2003-04-18 |
2009-07-07 |
Bristol-Myers Squibb Company |
Thyroid receptor ligands
|
US6846836B2
(en)
|
2003-04-18 |
2005-01-25 |
Bristol-Myers Squibb Company |
N-substituted phenylurea inhibitors of mitochondrial F1F0 ATP hydrolase
|
US6995183B2
(en)
|
2003-08-01 |
2006-02-07 |
Bristol Myers Squibb Company |
Adamantylglycine-based inhibitors of dipeptidyl peptidase IV and methods
|
US7820702B2
(en)
|
2004-02-04 |
2010-10-26 |
Bristol-Myers Squibb Company |
Sulfonylpyrrolidine modulators of androgen receptor function and method
|
US7378426B2
(en)
|
2004-03-01 |
2008-05-27 |
Bristol-Myers Squibb Company |
Fused heterotricyclic compounds as inhibitors of 17β-hydroxysteroid dehydrogenase 3
|
US7696241B2
(en)
|
2004-03-04 |
2010-04-13 |
Bristol-Myers Squibb Company |
Bicyclic compounds as modulators of androgen receptor function and method
|
US7625923B2
(en)
|
2004-03-04 |
2009-12-01 |
Bristol-Myers Squibb Company |
Bicyclic modulators of androgen receptor function
|
US7772232B2
(en)
|
2004-04-15 |
2010-08-10 |
Bristol-Myers Squibb Company |
Quinazolinyl compounds as inhibitors of potassium channel function
|
US7550499B2
(en)
|
2004-05-12 |
2009-06-23 |
Bristol-Myers Squibb Company |
Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
|
US9889110B2
(en)
|
2004-06-07 |
2018-02-13 |
University Of Tennessee Research Foundation |
Selective androgen receptor modulator for treating hormone-related conditions
|
US9884038B2
(en)
|
2004-06-07 |
2018-02-06 |
University Of Tennessee Research Foundation |
Selective androgen receptor modulator and methods of use thereof
|
US7534763B2
(en)
|
2004-07-02 |
2009-05-19 |
Bristol-Myers Squibb Company |
Sustained release GLP-1 receptor modulators
|
TW200611704A
(en)
|
2004-07-02 |
2006-04-16 |
Bristol Myers Squibb Co |
Human glucagon-like-peptide-1 modulators and their use in the treatment of diabetes and related conditions
|
US7145040B2
(en)
|
2004-07-02 |
2006-12-05 |
Bristol-Myers Squibb Co. |
Process for the preparation of amino acids useful in the preparation of peptide receptor modulators
|
US7572805B2
(en)
|
2004-07-14 |
2009-08-11 |
Bristol-Myers Squibb Company |
Pyrrolo(oxo)isoquinolines as 5HT ligands
|
US7429611B2
(en)
|
2004-09-23 |
2008-09-30 |
Bristol-Myers Squibb Company |
Indole inhibitors of 15-lipoxygenase
|
AR051446A1
(es)
|
2004-09-23 |
2007-01-17 |
Bristol Myers Squibb Co |
Glucosidos de c-arilo como inhibidores selectivos de transportadores de glucosa (sglt2)
|
US7754755B2
(en)
|
2004-09-23 |
2010-07-13 |
Bristol-Myers Squibb Company |
Inhibitors of 15-lipoxygenase
|
US7517991B2
(en)
|
2004-10-12 |
2009-04-14 |
Bristol-Myers Squibb Company |
N-sulfonylpiperidine cannabinoid receptor 1 antagonists
|
US8143425B2
(en)
|
2004-10-12 |
2012-03-27 |
Bristol-Myers Squibb Company |
Heterocyclic aromatic compounds useful as growth hormone secretagogues
|
CN101087609B
(zh)
|
2004-10-26 |
2012-11-14 |
詹森药业有限公司 |
因子Xa化合物
|
US7589088B2
(en)
|
2004-12-29 |
2009-09-15 |
Bristol-Myers Squibb Company |
Pyrimidine-based inhibitors of dipeptidyl peptidase IV and methods
|
US7635699B2
(en)
|
2004-12-29 |
2009-12-22 |
Bristol-Myers Squibb Company |
Azolopyrimidine-based inhibitors of dipeptidyl peptidase IV and methods
|
WO2006076597A1
(en)
|
2005-01-12 |
2006-07-20 |
Bristol-Myers Squibb Company |
Bicyclic heterocycles as cannabinoid receptor modulators
|
US7314882B2
(en)
|
2005-01-12 |
2008-01-01 |
Bristol-Myers Squibb Company |
Bicyclic heterocycles as cannabinoid receptor modulators
|
WO2006076568A2
(en)
|
2005-01-12 |
2006-07-20 |
Bristol-Myers Squibb Company |
Thiazolopyridines as cannabinoid receptor modulators
|
WO2006076575A2
(en)
|
2005-01-13 |
2006-07-20 |
Bristol-Myers Squibb Company |
Substituted biaryl compounds as factor xia inhibitors
|
US20060160850A1
(en)
|
2005-01-18 |
2006-07-20 |
Chongqing Sun |
Bicyclic heterocycles as cannabinoid receptor modulators
|
MX2007008434A
(es)
|
2005-01-19 |
2007-07-25 |
Squibb Bristol Myers Co |
Derivados de 2-fenoxi-n-(1,3,4-tiadizol-2il)piridin-3-amina y compuestos relacionados como inhibidores del receptor p2y1 para el tratamiento de trastornos tromboembolicos.
|
ES2319461T3
(es)
|
2005-02-10 |
2009-05-07 |
Bristol-Myers Squibb Company |
Dihidroquinazolinonas como moduladores de 5ht.
|
EP1879881A2
(en)
|
2005-04-14 |
2008-01-23 |
Bristol-Myers Squibb Company |
Inhibitors of 11-beta hydroxysteroid dehydrogenase type i
|
US7521557B2
(en)
|
2005-05-20 |
2009-04-21 |
Bristol-Myers Squibb Company |
Pyrrolopyridine-based inhibitors of dipeptidyl peptidase IV and methods
|
US7629342B2
(en)
|
2005-06-17 |
2009-12-08 |
Bristol-Myers Squibb Company |
Azabicyclic heterocycles as cannabinoid receptor modulators
|
US7317012B2
(en)
|
2005-06-17 |
2008-01-08 |
Bristol-Myers Squibb Company |
Bicyclic heterocycles as cannabinoind-1 receptor modulators
|
US7452892B2
(en)
|
2005-06-17 |
2008-11-18 |
Bristol-Myers Squibb Company |
Triazolopyrimidine cannabinoid receptor 1 antagonists
|
US7632837B2
(en)
|
2005-06-17 |
2009-12-15 |
Bristol-Myers Squibb Company |
Bicyclic heterocycles as cannabinoid-1 receptor modulators
|
US7572808B2
(en)
|
2005-06-17 |
2009-08-11 |
Bristol-Myers Squibb Company |
Triazolopyridine cannabinoid receptor 1 antagonists
|
WO2007002634A1
(en)
|
2005-06-27 |
2007-01-04 |
Bristol-Myers Squibb Company |
Carbocycle and heterocycle antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
|
EP1896417B1
(en)
|
2005-06-27 |
2011-03-23 |
Bristol-Myers Squibb Company |
Linear urea mimics antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
|
DE602006017694D1
(de)
|
2005-06-27 |
2010-12-02 |
Bristol Myers Squibb Co |
C-verknüpfte zyklische antagonisten des p2y1-rezeptors mit eignung bei der behandlung thrombotischer leiden
|
AU2006261828A1
(en)
|
2005-06-27 |
2007-01-04 |
Bristol-Myers Squibb Company |
N-linked heterocyclic antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
|
EP1812411A2
(en)
*
|
2005-07-05 |
2007-08-01 |
Teva Pharmaceutical Industries Ltd. |
Process for preparing valsartan
|
EP1757290A1
(en)
|
2005-08-16 |
2007-02-28 |
Zentaris GmbH |
Novel triazole derivatives as ghrelin analogue ligands of growth hormone secretagogue receptors
|
US7795436B2
(en)
|
2005-08-24 |
2010-09-14 |
Bristol-Myers Squibb Company |
Substituted tricyclic heterocycles as serotonin receptor agonists and antagonists
|
US7534804B2
(en)
|
2005-08-24 |
2009-05-19 |
Bristol-Myers Squibb Company |
Benzoxazole inhibitors of 15-lipoxygenase
|
EP1931199A4
(en)
|
2005-08-31 |
2009-07-29 |
Univ Tennessee Res Foundation |
TREATMENT OF RENAL DISEASE, BURNS, INJURIES OR SPINAL CORD INJURY USING ANDROGEN RECEPTOR SELECTIVE MODULATORS
|
US8618115B2
(en)
|
2005-10-26 |
2013-12-31 |
Bristol-Myers Squibb Company |
Substituted thieno[3,2-d]pyrimidinones as MCHR1 antagonists and methods for using them
|
US7488725B2
(en)
|
2005-10-31 |
2009-02-10 |
Bristol-Myers Squibb Co. |
Pyrrolidinyl beta-amino amide-based inhibitors of dipeptidyl peptidase IV and methods
|
US7553836B2
(en)
|
2006-02-06 |
2009-06-30 |
Bristol-Myers Squibb Company |
Melanin concentrating hormone receptor-1 antagonists
|
MX2008011227A
(es)
*
|
2006-03-03 |
2009-02-10 |
Torrent Pharmaceuticals Ltd |
Receptores antagonistas de accion nueva y doble en los receptores at1 y eta.
|
WO2007109456A2
(en)
*
|
2006-03-16 |
2007-09-27 |
Pharmacopeia, Inc. |
Substituted biphenyl isoxazole sulfonamides as dual angiotensin endothelin receptor antagonists
|
WO2007139589A1
(en)
|
2006-05-26 |
2007-12-06 |
Bristol-Myers Squibb Company |
Sustained release glp-1 receptor modulators
|
US7919598B2
(en)
|
2006-06-28 |
2011-04-05 |
Bristol-Myers Squibb Company |
Crystal structures of SGLT2 inhibitors and processes for preparing same
|
CA2658394C
(en)
|
2006-07-12 |
2016-08-16 |
University Of Tennessee Research Foundation |
Substituted acylanilides and methods of use thereof
|
US7727978B2
(en)
|
2006-08-24 |
2010-06-01 |
Bristol-Myers Squibb Company |
Cyclic 11-beta hydroxysteroid dehydrogenase type I inhibitors
|
JP2010505881A
(ja)
|
2006-10-05 |
2010-02-25 |
ギリアード・パロ・アルト・インコーポレイテッド |
ステアロイルCoAデサチュラーゼインヒビターとして使用するための二環式窒素含有複素環式化合物
|
US7960569B2
(en)
|
2006-10-17 |
2011-06-14 |
Bristol-Myers Squibb Company |
Indole antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
|
CN101641013B
(zh)
|
2007-01-22 |
2014-07-30 |
Gtx公司 |
核受体结合剂
|
US9604931B2
(en)
|
2007-01-22 |
2017-03-28 |
Gtx, Inc. |
Nuclear receptor binding agents
|
US9623021B2
(en)
|
2007-01-22 |
2017-04-18 |
Gtx, Inc. |
Nuclear receptor binding agents
|
TW200838501A
(en)
|
2007-02-02 |
2008-10-01 |
Theravance Inc |
Dual-acting antihypertensive agents
|
TW200904405A
(en)
|
2007-03-22 |
2009-02-01 |
Bristol Myers Squibb Co |
Pharmaceutical formulations containing an SGLT2 inhibitor
|
US20080255161A1
(en)
*
|
2007-04-11 |
2008-10-16 |
Dmitry Koltun |
3-HYDROQUINAZOLIN-4-ONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS
|
CN101687873A
(zh)
|
2007-04-17 |
2010-03-31 |
百时美施贵宝公司 |
具有稠合杂环的11β-羟基类固醇Ⅰ型脱氢酶抑制剂
|
PE20090696A1
(es)
|
2007-04-20 |
2009-06-20 |
Bristol Myers Squibb Co |
Formas cristalinas de saxagliptina y procesos para preparar las mismas
|
KR20100015886A
(ko)
|
2007-04-23 |
2010-02-12 |
사노피-아벤티스 |
P2y12 길항제로서의 퀴놀린-카복스아미드 유도체
|
TWI448284B
(zh)
|
2007-04-24 |
2014-08-11 |
Theravance Inc |
雙效抗高血壓劑
|
PE20090213A1
(es)
|
2007-05-04 |
2009-02-28 |
Bristol Myers Squibb Co |
Agonistas del receptor acoplado a la proteina g gpr119 [6,5]-biciclicos
|
ES2388967T3
(es)
|
2007-05-04 |
2012-10-22 |
Bristol-Myers Squibb Company |
Agonistas [6,6]- y [6,7]-bicíclicos del receptor GPR119 acoplado a la proteína G
|
TWI406850B
(zh)
|
2007-06-05 |
2013-09-01 |
Theravance Inc |
雙效苯并咪唑抗高血壓劑
|
US20090011994A1
(en)
|
2007-07-06 |
2009-01-08 |
Bristol-Myers Squibb Company |
Non-basic melanin concentrating hormone receptor-1 antagonists and methods
|
CA2693439A1
(en)
|
2007-07-17 |
2009-01-22 |
Bristol-Myers Squibb Company |
Pyridone gpr119 g protein-coupled receptor agonists
|
JP2010534722A
(ja)
|
2007-07-27 |
2010-11-11 |
ブリストル−マイヤーズ スクイブ カンパニー |
新規グルコキナーゼ活性化薬およびその使用方法
|
EP2200975A1
(en)
|
2007-09-07 |
2010-06-30 |
Theravance, Inc. |
Dual-acting antihypertensive agents
|
US7968603B2
(en)
|
2007-09-11 |
2011-06-28 |
University Of Tennessee Research Foundation |
Solid forms of selective androgen receptor modulators
|
CN101801954B
(zh)
|
2007-09-20 |
2013-10-09 |
Irm责任有限公司 |
作为gpr119活性调节剂的化合物和组合物
|
CA2705921A1
(en)
|
2007-12-11 |
2009-06-18 |
Theravance, Inc. |
Dual-acting benzoimidazole derivatives and their use as antihypertensive agents
|
WO2009080226A2
(en)
|
2007-12-26 |
2009-07-02 |
Sanofis-Aventis |
Heterocyclic pyrazole-carboxamides as p2y12 antagonists
|
EP2103602A1
(en)
|
2008-03-17 |
2009-09-23 |
AEterna Zentaris GmbH |
Novel 1,2,4-triazole derivatives and process of manufacturing thereof
|
JP2011518884A
(ja)
*
|
2008-04-29 |
2011-06-30 |
セラヴァンス, インコーポレーテッド |
二重活性抗高血圧剤
|
WO2009143039A2
(en)
|
2008-05-19 |
2009-11-26 |
Schering Corporation |
Heterocyclic compounds as factor ixa inhibitors
|
PE20091928A1
(es)
|
2008-05-29 |
2009-12-31 |
Bristol Myers Squibb Co |
Tienopirimidinas hidroxisustituidas como antagonistas de receptor-1 de hormona concentradora de melanina no basicos
|
WO2009155448A1
(en)
*
|
2008-06-20 |
2009-12-23 |
Ligand Pharmaceuticals Inc. |
Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
|
TW201006821A
(en)
|
2008-07-16 |
2010-02-16 |
Bristol Myers Squibb Co |
Pyridone and pyridazone analogues as GPR119 modulators
|
JP2011529072A
(ja)
|
2008-07-24 |
2011-12-01 |
セラヴァンス, インコーポレーテッド |
二重作用血圧降下薬
|
US8557983B2
(en)
|
2008-12-04 |
2013-10-15 |
Abbvie Inc. |
Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
|
US20100160322A1
(en)
|
2008-12-04 |
2010-06-24 |
Abbott Laboratories |
Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
|
US8586754B2
(en)
|
2008-12-05 |
2013-11-19 |
Abbvie Inc. |
BCL-2-selective apoptosis-inducing agents for the treatment of cancer and immune diseases
|
US8563735B2
(en)
|
2008-12-05 |
2013-10-22 |
Abbvie Inc. |
Bcl-2-selective apoptosis-inducing agents for the treatment of cancer and immune diseases
|
RU2011141794A
(ru)
*
|
2009-03-17 |
2013-04-27 |
Дайити Санкио Компани, Лимитед |
Амидное производное
|
CA2756786A1
(en)
|
2009-03-27 |
2010-09-30 |
Bristol-Myers Squibb Company |
Methods for preventing major adverse cardiovascular events with dpp-iv inhibitors
|
EP3708163A1
(en)
*
|
2009-03-31 |
2020-09-16 |
Ligand Pharmaceuticals, Inc. |
Use of sparsentan for the treatment of chronic inflammatory diseases
|
US9034875B2
(en)
|
2009-05-26 |
2015-05-19 |
Abbvie Inc. |
Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
|
US20220315555A1
(en)
|
2009-05-26 |
2022-10-06 |
Abbvie Inc. |
Apoptosis inducing agents for the treatment of cancer and immune and autoimmune diseases
|
US8546399B2
(en)
|
2009-05-26 |
2013-10-01 |
Abbvie Inc. |
Apoptosis inducing agents for the treatment of cancer and immune and autoimmune diseases
|
DK2435432T6
(da)
*
|
2009-05-26 |
2023-12-18 |
Abbvie Ireland Unlimited Co |
Apoptose-inducerende midler til behandling af cancer og immune og autoimmune sygdomme
|
WO2010147978A1
(en)
|
2009-06-16 |
2010-12-23 |
Pfizer Inc. |
Dosage forms of apixaban
|
EP2451782B1
(en)
|
2009-07-07 |
2016-11-09 |
Theravance Biopharma R&D IP, LLC |
Dual-acting pyrazole antihypertensive agents
|
WO2011011232A1
(en)
|
2009-07-22 |
2011-01-27 |
Theravance, Inc. |
Dual-acting oxazole antihypertensive agents
|
WO2011014520A2
(en)
|
2009-07-29 |
2011-02-03 |
Irm Llc |
Compounds and compositions as modulators of gpr119 activity
|
EP2462123B1
(en)
|
2009-08-04 |
2013-10-02 |
Merck Sharp & Dohme Corp. |
4,5,6-trisubstituted pyrimidine derivatives as factor ixa inhibitors
|
CA2774573A1
(en)
|
2009-10-09 |
2011-04-14 |
Irm Llc |
Compounds and compositions as modulators of gpr119 activity
|
RS57926B1
(sr)
|
2009-11-13 |
2019-01-31 |
Astrazeneca Ab |
Formulacije tablete sa trenutnim oslobađanjem
|
CA2780939C
(en)
|
2009-11-13 |
2018-06-12 |
Bristol-Myers Squibb Company |
Bilayer tablet formulations
|
RU2564901C2
(ru)
|
2009-11-13 |
2015-10-10 |
Бристол-Майерс Сквибб Кампани |
Композиции метформина с уменьшенной массой
|
CN101891735B
(zh)
*
|
2009-11-25 |
2012-07-18 |
北京理工大学 |
联苯磺胺异噁唑类化合物、合成方法及用途
|
CN101921265B
(zh)
*
|
2009-11-25 |
2012-07-04 |
北京理工大学 |
联苯酰胺四唑类化合物、合成方法及用途
|
US8394858B2
(en)
|
2009-12-03 |
2013-03-12 |
Novartis Ag |
Cyclohexane derivatives and uses thereof
|
EP2526095A1
(en)
|
2010-01-19 |
2012-11-28 |
Theravance, Inc. |
Dual-acting thiophene, pyrrole, thiazole and furan antihypertensive agents
|
TWI562775B
(en)
|
2010-03-02 |
2016-12-21 |
Lexicon Pharmaceuticals Inc |
Methods of using inhibitors of sodium-glucose cotransporters 1 and 2
|
WO2011127106A1
(en)
|
2010-04-08 |
2011-10-13 |
Bristol-Myers Squibb Company |
Pyrimidinylpiperidinyloxypyridinone analogues as gpr119 modulators
|
WO2011130459A1
(en)
|
2010-04-14 |
2011-10-20 |
Bristol-Myers Squibb Company |
Novel glucokinase activators and methods of using same
|
JP2013525489A
(ja)
|
2010-05-06 |
2013-06-20 |
ブリストル−マイヤーズ スクイブ カンパニー |
Gpr119修飾因子としての二環式ヘテロアリール類似体
|
EP2566862B1
(en)
|
2010-05-06 |
2015-09-16 |
Bristol-Myers Squibb Company |
Benzofuranyl analogues as gpr119 modulators
|
US8697739B2
(en)
|
2010-07-29 |
2014-04-15 |
Novartis Ag |
Bicyclic acetyl-CoA carboxylase inhibitors and uses thereof
|
EP2431035A1
(en)
|
2010-09-16 |
2012-03-21 |
Æterna Zentaris GmbH |
Novel Triazole Derivatives with Improved Receptor Activity and Bioavailability Properties as Ghrelin Antagonists of Growth Hormone Secretagogue Receptors
|
CA2811805A1
(en)
|
2010-10-29 |
2012-05-03 |
Abbvie Inc. |
Solid dispersions containing an apoptosis-inducing agent
|
UA113500C2
(xx)
|
2010-10-29 |
2017-02-10 |
|
Одержані екструзією розплаву тверді дисперсії, що містять індукуючий апоптоз засіб
|
KR101923364B1
(ko)
|
2010-11-23 |
2018-11-30 |
애브비 인코포레이티드 |
아폽토시스유도제의 염 및 결정형
|
DK2642999T3
(en)
|
2010-11-23 |
2017-01-09 |
Abbvie Ireland Unlimited Co |
METHODS OF TREATMENT FOR USING selectivity-VE BCL-2 INHIBITORS
|
CA2822769C
(en)
|
2010-12-23 |
2016-10-04 |
Purdue Pharma L.P. |
Tamper resistant solid oral dosage forms
|
TWI631963B
(zh)
|
2011-01-05 |
2018-08-11 |
雷西肯製藥股份有限公司 |
包含鈉-葡萄糖共同輸送體1與2之抑制劑的組合物與應用方法
|
WO2013068875A1
(en)
|
2011-11-11 |
2013-05-16 |
Pfizer Inc. |
2-thiopyrimidinones
|
US9296745B2
(en)
|
2012-04-06 |
2016-03-29 |
Pfizer Inc. |
Diacylglycerol acyltransferase 2 inhibitors
|
US9174965B2
(en)
|
2012-05-16 |
2015-11-03 |
Bristol-Myers Squibb Company |
Pyrimidinylpiperidinyloxypyridone analogues as GPR119 modulators
|
NZ703632A
(en)
|
2012-06-11 |
2016-01-29 |
Bristol Myers Squibb Co |
Phosphoramidic acid prodrugs of 5-[5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl]pyridine-3-sulfonamide
|
US10258596B2
(en)
|
2012-07-13 |
2019-04-16 |
Gtx, Inc. |
Method of treating HER2-positive breast cancers with selective androgen receptor modulators (SARMS)
|
KR102238970B1
(ko)
|
2012-07-13 |
2021-04-09 |
지티엑스, 인코포레이티드 |
선택적 안드로겐 수용체 조절자(sarms)를 이용한 안드로겐 수용체(ar) 양성 유방암의 치료 방법
|
US9622992B2
(en)
|
2012-07-13 |
2017-04-18 |
Gtx, Inc. |
Method of treating androgen receptor (AR)-positive breast cancers with selective androgen receptor modulator (SARMs)
|
US9744149B2
(en)
|
2012-07-13 |
2017-08-29 |
Gtx, Inc. |
Method of treating androgen receptor (AR)-positive breast cancers with selective androgen receptor modulator (SARMs)
|
US10987334B2
(en)
|
2012-07-13 |
2021-04-27 |
University Of Tennessee Research Foundation |
Method of treating ER mutant expressing breast cancers with selective androgen receptor modulators (SARMs)
|
US10314807B2
(en)
|
2012-07-13 |
2019-06-11 |
Gtx, Inc. |
Method of treating HER2-positive breast cancers with selective androgen receptor modulators (SARMS)
|
US9969683B2
(en)
|
2012-07-13 |
2018-05-15 |
Gtx, Inc. |
Method of treating estrogen receptor (ER)-positive breast cancers with selective androgen receptor modulator (SARMS)
|
LT6043B
(lt)
|
2012-08-27 |
2014-06-25 |
Uab "Mibarsas" |
Organinės trąšos sapropelio pagrindu ir jų gamybos būdas
|
EP2892897A1
(en)
|
2012-09-05 |
2015-07-15 |
Bristol-Myers Squibb Company |
Pyrrolone or pyrrolidinone melanin concentrating hormone receptor-1 antagonists
|
WO2014039411A1
(en)
|
2012-09-05 |
2014-03-13 |
Bristol-Myers Squibb Company |
Pyrrolone or pyrrolidinone melanin concentrating hormore receptor-1 antagonists
|
WO2014052619A1
(en)
|
2012-09-27 |
2014-04-03 |
Irm Llc |
Piperidine derivatives and compositions as modulators of gpr119 activity
|
KR102165224B1
(ko)
|
2012-11-20 |
2020-10-13 |
렉시컨 파마슈티컬스 인코퍼레이티드 |
나트륨 글루코스 공동수송체 1의 억제제
|
WO2014143609A1
(en)
|
2013-03-11 |
2014-09-18 |
Bristol-Myers Squibb Company |
Isoquinolines as potassium ion channel inhibitors
|
US9242966B2
(en)
|
2013-03-11 |
2016-01-26 |
Bristol-Myers Squibb Company |
Phthalazines as potassium ion channel inhibitors
|
US9050345B2
(en)
|
2013-03-11 |
2015-06-09 |
Bristol-Myers Squibb Company |
Pyrrolotriazines as potassium ion channel inhibitors
|
ES2616026T3
(es)
|
2013-03-11 |
2017-06-09 |
Bristol-Myers Squibb Company |
Pirrolopiridazinas como inhibidores de canales de iones potasio
|
JP6395798B2
(ja)
|
2013-03-11 |
2018-09-26 |
ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company |
カリウムイオンチャネル阻害剤としてのピロロトリアジン
|
US20140275082A1
(en)
|
2013-03-14 |
2014-09-18 |
Abbvie Inc. |
Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
|
CA2911376C
(en)
*
|
2013-03-15 |
2021-03-30 |
University Of Southern California |
Phenyl(sulfonylcarbamate) derivatives and pharmaceutical compositions thereof for the treatment of angiotensin-related diseases
|
ES2665153T3
(es)
|
2013-10-09 |
2018-04-24 |
Pfizer Inc. |
Antagonistas del receptor EP3 de prostaglandina
|
US9580422B2
(en)
|
2013-10-22 |
2017-02-28 |
Bristol-Myers Squibb Company |
Isotopically labeled triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors
|
CN106103425A
(zh)
|
2014-03-17 |
2016-11-09 |
辉瑞公司 |
用于治疗代谢及相关病症的二酰甘油酰基转移酶2抑制剂
|
ES2718552T3
(es)
|
2014-04-04 |
2019-07-02 |
Pfizer |
Compuestos de heteroarilo o arilo bicíclicos fusionados y su uso como inhibidores de IRAK4
|
US9969724B2
(en)
|
2014-04-16 |
2018-05-15 |
Merck Sharp & Dohme Corp. |
Factor IXa inhibitors
|
WO2015181676A1
(en)
|
2014-05-30 |
2015-12-03 |
Pfizer Inc. |
Carbonitrile derivatives as selective androgen receptor modulators
|
JP2017538769A
(ja)
|
2014-12-22 |
2017-12-28 |
ファイザー・インク |
プロスタグランジンep3受容体の拮抗薬
|
CN104761548B
(zh)
*
|
2015-04-27 |
2017-09-12 |
梯尔希(南京)药物研发有限公司 |
一种稳定同位素标记的二苯基磺酰胺类药物的制备方法
|
WO2016178113A1
(en)
|
2015-05-05 |
2016-11-10 |
Pfizer Inc. |
2-thiopyrimidinones
|
CA2987179C
(en)
|
2015-05-29 |
2020-08-25 |
Pfizer Inc. |
Heterocyclic compounds as inhibitors of vanin-1 enzyme
|
WO2016203347A1
(en)
|
2015-06-17 |
2016-12-22 |
Pfizer Inc. |
Tricyclic compounds and their use as phosphodiesterase inhibitors
|
WO2016203335A1
(en)
|
2015-06-18 |
2016-12-22 |
Pfizer Inc. |
Novel pyrido[2,3-b]pyrazinones as bet-family bromodomain inhibitors
|
US20180230127A1
(en)
|
2015-08-13 |
2018-08-16 |
Pfizer Inc. |
Bicyclic-Fused Heteroaryl Or Aryl Compounds
|
MX2018002402A
(es)
|
2015-08-27 |
2018-04-11 |
Pfizer |
Compuestos de heteroarilo o arilo biciclicos fusionados como moduladores de la quinasa 4 asociada al receptor de la interleucina 1 (irak4).
|
WO2017037567A1
(en)
|
2015-09-03 |
2017-03-09 |
Pfizer Inc. |
Regulators of frataxin
|
CN105481844A
(zh)
*
|
2015-12-08 |
2016-04-13 |
梁彦云 |
一种治疗高血压的药物组合物
|
SG11201804363UA
(en)
|
2015-12-29 |
2018-07-30 |
Pfizer |
Substituted 3-azabicyclo[3.1.0]hexanes as ketohexokinase inhibitors
|
CN106188115A
(zh)
*
|
2016-07-13 |
2016-12-07 |
北京理工大学 |
廉价高效合成2‑二羟硼基‑n‑二甲异噁唑基‑n‑甲氧乙氧甲基苯磺酰胺的新方法
|
WO2018011681A1
(en)
|
2016-07-14 |
2018-01-18 |
Pfizer Inc. |
Novel pyrimidine carboxamides as inhibitors of vanin-1 enzyme
|
US10604541B2
(en)
|
2016-07-22 |
2020-03-31 |
Bristol-Myers Squibb Company |
Glucokinase activators and methods of using same
|
AR109179A1
(es)
|
2016-08-19 |
2018-11-07 |
Pfizer |
Inhibidores de diacilglicerol aciltransferasa 2
|
EP3525784A1
(en)
|
2016-10-13 |
2019-08-21 |
Retrophin, Inc. |
Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders
|
WO2018162625A1
(en)
|
2017-03-09 |
2018-09-13 |
Truly Translational Sweden Ab |
Prodrugs of sulfasalazine, pharmaceutical compositions thereof and their use in the treatment of autoimmune disease
|
DK3630188T3
(da)
|
2017-05-31 |
2021-11-15 |
Amplio Pharma Ab |
Farmaceutisk sammensætning omfattende en kombination af methotrexat og novobiocin og anvendelse af sammensætningen til behandling
|
EP3488868B1
(en)
|
2017-11-23 |
2023-09-13 |
medac Gesellschaft für klinische Spezialpräparate mbH |
Pharmaceutical composition for oral administration containing sulfasalazine and / or a sulfasalazine organic salt, production process and use
|
EP3489222A1
(en)
|
2017-11-23 |
2019-05-29 |
medac Gesellschaft für klinische Spezialpräparate mbH |
Sulfasalazine salts, production processes and uses
|
CN111518770B
(zh)
|
2017-12-19 |
2023-01-06 |
北京吉源生物科技有限公司 |
一种表达glp1和fgf21的干细胞及其用途
|
WO2019133445A1
(en)
|
2017-12-28 |
2019-07-04 |
Inception Ibd, Inc. |
Aminothiazoles as inhibitors of vanin-1
|
CA3105626A1
(en)
|
2018-07-19 |
2020-01-23 |
Astrazeneca Ab |
Methods of treating hfpef employing dapagliflozin and compositions comprising the same
|
KR102614808B1
(ko)
|
2018-08-31 |
2023-12-19 |
화이자 인코포레이티드 |
Nash/nafld 및 관련 질환의 치료를 위한 조합물
|
AU2019346497A1
(en)
|
2018-09-26 |
2021-04-08 |
Lexicon Pharmaceuticals, Inc. |
Crystalline forms of n-(1 -((2-(dimethylamino)ethyl)amino)-2-m ethyl-1 -oopropan-2-yl)-4-(4-(2-methyl-5- (2s,3r,4r,5s,6r)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2h-pyran-2-yl)benzyl) phenl)butanamide and methods of their synthesis
|
WO2020072814A1
(en)
|
2018-10-04 |
2020-04-09 |
Retrophin, Inc. |
Biphenyl sulfonamide compounds for the treatment of type iv collagen diseases
|
WO2020102575A1
(en)
|
2018-11-16 |
2020-05-22 |
Inception Ibd, Inc. |
Heterocyclic aminothiazoles and uses thereof
|
EP3972596A1
(en)
|
2019-05-20 |
2022-03-30 |
Pfizer Inc. |
Combinations comprising benzodioxol as glp-1r agonists for use in the treatment of nash/nafld and related diseases
|
TW202115086A
(zh)
|
2019-06-28 |
2021-04-16 |
美商輝瑞大藥廠 |
Bckdk抑制劑
|
WO2020261144A1
(en)
|
2019-06-28 |
2020-12-30 |
Pfizer Inc. |
5-(thiophen-2-yl)-1h-tetrazole derivatives as bckdk inhibitors useful for treating various diseases
|
TWI771766B
(zh)
|
2019-10-04 |
2022-07-21 |
美商輝瑞股份有限公司 |
二醯基甘油醯基轉移酶2 抑制劑
|
JP2022058085A
(ja)
|
2020-02-24 |
2022-04-11 |
ファイザー・インク |
ジアシルグリセロールアシルトランスフェラーゼ2阻害剤とアセチル-CoAカルボキシラーゼ阻害剤との組合せ
|
CA3186348A1
(en)
|
2020-06-09 |
2021-12-16 |
Pfizer Inc. |
Spiro compounds as melanocortin 4 receptor antagonists and uses thereof
|
WO2022022865A1
(en)
|
2020-07-27 |
2022-02-03 |
Astrazeneca Ab |
Methods of treating chronic kidney disease with dapagliflozin
|
WO2022266370A1
(en)
|
2021-06-17 |
2022-12-22 |
Aria Pharmaceuticals, Inc. |
Sparsentan for treating idiopathic pulmonary fibrosis
|
WO2023275715A1
(en)
|
2021-06-30 |
2023-01-05 |
Pfizer Inc. |
Metabolites of selective androgen receptor modulators
|
CN117836294A
(zh)
*
|
2021-08-26 |
2024-04-05 |
上海翰森生物医药科技有限公司 |
含芳环类生物拮抗剂、其制备方法和应用
|
WO2023026180A1
(en)
|
2021-08-26 |
2023-03-02 |
Pfizer Inc. |
Amorphous form of (s)-2-(5-((3-ethoxypyridin-2-yl)oxy)pyridin-3-yl)-n-(tetrahydrofuran-3- yl)pyrimidine-5-carboxamide
|
CN118119617A
(zh)
|
2021-10-21 |
2024-05-31 |
年衍药业(上海)有限公司 |
一种双重拮抗剂及其用途
|
IL312296A
(en)
|
2021-12-01 |
2024-06-01 |
Pfizer |
3-PHENYL-1-BENZOTHIOPEN-2-CARBOXYLIC ACID DERIVATIVES AS INHIBITORS OF BRANCHED ALPHA KETO ACID DEHYDROGENSIS KINASE FOR THE TREATMENT OF DIABETES, KIDNEY DISEASES, NASH AND HEART
|
WO2023105387A1
(en)
|
2021-12-06 |
2023-06-15 |
Pfizer Inc. |
Melanocortin 4 receptor antagonists and uses thereof
|
WO2023144722A1
(en)
|
2022-01-26 |
2023-08-03 |
Astrazeneca Ab |
Dapagliflozin for use in the treatment of prediabetes or reducing the risk of developing type 2 diabetes
|
WO2023169456A1
(en)
|
2022-03-09 |
2023-09-14 |
Gasherbrum Bio , Inc. |
Heterocyclic glp-1 agonists
|
WO2023198140A1
(en)
|
2022-04-14 |
2023-10-19 |
Gasherbrum Bio, Inc. |
Heterocyclic glp-1 agonists
|
WO2023224963A1
(en)
*
|
2022-05-16 |
2023-11-23 |
Aria Pharmaceuticals, Inc. |
Dual-acting angiotensin and endothelin receptor antagonists
|
WO2024075051A1
(en)
|
2022-10-07 |
2024-04-11 |
Pfizer Inc. |
Hsd17b13 inhibitors and/or degraders
|
WO2024084360A1
(en)
|
2022-10-18 |
2024-04-25 |
Pfizer Inc. |
Patatin-like phospholipase domain-containing protein 3 (pnpla3) modifiers
|
US20240182468A1
(en)
|
2022-10-18 |
2024-06-06 |
Pfizer Inc. |
Compounds for the activation of ampk
|
CN115745983A
(zh)
*
|
2022-11-23 |
2023-03-07 |
深圳信立泰药业股份有限公司 |
一种血管紧张肽和内皮肽受体拮抗剂及其应用
|
WO2024125602A1
(en)
|
2022-12-15 |
2024-06-20 |
Gasherbrum Bio, Inc. |
Salts and solid forms of a compound having glp-1 agonist activity
|
WO2024127297A1
(en)
|
2022-12-16 |
2024-06-20 |
Pfizer Inc. |
3-fluoro-4-hydroxybenzmide-containing inhibitors and/or degraders and uses thereof
|