KR20230165366A - 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용 - Google Patents

트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용 Download PDF

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KR20230165366A
KR20230165366A KR1020237040564A KR20237040564A KR20230165366A KR 20230165366 A KR20230165366 A KR 20230165366A KR 1020237040564 A KR1020237040564 A KR 1020237040564A KR 20237040564 A KR20237040564 A KR 20237040564A KR 20230165366 A KR20230165366 A KR 20230165366A
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compound
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Korean (ko)
Inventor
이쿠오 미타니
요스케 오고시
다쿠야 마츠이
마사히로 요코타
마사카즈 데라시타
다이 모토다
가즈히토 우에야마
히로유키 아베
다카히로 홋타
다카시 이토
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니뽄 다바코 산교 가부시키가이샤
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Priority claimed from KR1020217012148A external-priority patent/KR20210048589A/ko
Publication of KR20230165366A publication Critical patent/KR20230165366A/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06—Antianaemics

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
KR1020237040564A 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용 Ceased KR20230165366A (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
JPJP-P-2009-169565 2009-07-17
JP2009169565 2009-07-17
US27312709P 2009-07-30 2009-07-30
US61/273,127 2009-07-30
KR1020217012148A KR20210048589A (ko) 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용
PCT/JP2010/062037 WO2011007856A1 (ja) 2009-07-17 2010-07-16 トリアゾロピリジン化合物、ならびにそのプロリル水酸化酵素阻害剤およびエリスロポエチン産生誘導剤としての作用

Related Parent Applications (1)

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KR1020217012148A Division KR20210048589A (ko) 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용

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KR20230165366A true KR20230165366A (ko) 2023-12-05

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KR1020237040564A Ceased KR20230165366A (ko) 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용
KR1020187010331A Ceased KR20180042443A (ko) 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용
KR1020177003353A Active KR101850661B1 (ko) 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용
KR1020127004258A Active KR101706803B1 (ko) 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용

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KR1020187010331A Ceased KR20180042443A (ko) 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용
KR1020177003353A Active KR101850661B1 (ko) 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용
KR1020127004258A Active KR101706803B1 (ko) 2009-07-17 2010-07-16 트리아졸로피리딘 화합물, 그리고 그 프롤릴 수산화효소 저해제 및 에리트로포이에틴 생성 유도제로서의 작용

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JP6434575B2 (ja) 2018-12-05
EP2455381B1 (en) 2014-05-28
CO6430426A2 (es) 2012-04-30
JP5021797B2 (ja) 2012-09-12
SG178049A1 (en) 2012-03-29
JP2022126843A (ja) 2022-08-30
CN102471337A (zh) 2012-05-23
US8283465B2 (en) 2012-10-09
JP2019019144A (ja) 2019-02-07
AR077417A1 (es) 2011-08-24
NZ598242A (en) 2013-09-27
EP2455381A4 (en) 2012-12-12
PT2455381E (pt) 2014-06-24
HRP20140705T1 (hr) 2014-09-12
JP2012144571A (ja) 2012-08-02
JP2024091878A (ja) 2024-07-05
BR112012001157A2 (pt) 2016-02-23
TWI485150B (zh) 2015-05-21
JP2015003933A (ja) 2015-01-08
US20110077267A1 (en) 2011-03-31
HK1168346A1 (en) 2012-12-28
CA2768505A1 (en) 2011-01-20
JP2017214404A (ja) 2017-12-07
JP2020111612A (ja) 2020-07-27
ES2477968T3 (es) 2014-07-18
IL217541A0 (en) 2012-02-29
KR101850661B1 (ko) 2018-04-19
US20160145254A1 (en) 2016-05-26
TW201105671A (en) 2011-02-16
KR101706803B1 (ko) 2017-02-14
CN102471337B (zh) 2014-12-10
KR20180042443A (ko) 2018-04-25
PL2455381T3 (pl) 2014-10-31
WO2011007856A1 (ja) 2011-01-20
RS53499B1 (sr) 2015-02-27
RU2012105467A (ru) 2013-08-27
PE20120629A1 (es) 2012-05-30
ME01858B (me) 2014-12-20
ES2477968T9 (es) 2014-11-13
MX2012000766A (es) 2012-02-08
SMT201500122B (it) 2015-07-09
AU2010271732A1 (en) 2012-03-08
EP2746282A1 (en) 2014-06-25
JP2016040321A (ja) 2016-03-24
EP3594213A1 (en) 2020-01-15
DK2455381T3 (da) 2014-07-21
EP2455381B9 (en) 2014-10-22
US20130096155A1 (en) 2013-04-18
DK2455381T5 (en) 2015-02-09
SI2455381T1 (sl) 2014-08-29
IL217541A (en) 2014-07-31
EP2455381A1 (en) 2012-05-23
RU2538963C2 (ru) 2015-01-10
AU2010271732B2 (en) 2016-08-25
KR20170018105A (ko) 2017-02-15
CA2768505C (en) 2018-06-12
JP2011037841A (ja) 2011-02-24
MY160814A (en) 2017-03-31
KR20120051704A (ko) 2012-05-22

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