HRP20140705T1 - Spoj triazolopiridina i njegovo djelovanje kao inhibitora prolil hidroksilaze i induktora proizvodnje eritropoetina - Google Patents

Spoj triazolopiridina i njegovo djelovanje kao inhibitora prolil hidroksilaze i induktora proizvodnje eritropoetina Download PDF

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Publication number
HRP20140705T1
HRP20140705T1 HRP20140705AT HRP20140705T HRP20140705T1 HR P20140705 T1 HRP20140705 T1 HR P20140705T1 HR P20140705A T HRP20140705A T HR P20140705AT HR P20140705 T HRP20140705 T HR P20140705T HR P20140705 T1 HRP20140705 T1 HR P20140705T1
Authority
HR
Croatia
Prior art keywords
group
solvate
pharmaceutically acceptable
acceptable salt
compound according
Prior art date
Application number
HRP20140705AT
Other languages
English (en)
Croatian (hr)
Inventor
Ikuo Mitani
Yosuke Ogoshi
Takuya Matsui
Masahiro Yokota
Masakazu Terashita
Dai Motoda
Kazuhito Ueyama
Hiroyuki Abe
Takahiro Hotta
Takashi Ito
Original Assignee
Japan Tobacco, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Japan Tobacco, Inc. filed Critical Japan Tobacco, Inc.
Publication of HRP20140705T1 publication Critical patent/HRP20140705T1/hr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06—Antianaemics

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
HRP20140705AT 2009-07-17 2010-07-16 Spoj triazolopiridina i njegovo djelovanje kao inhibitora prolil hidroksilaze i induktora proizvodnje eritropoetina HRP20140705T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2009169565 2009-07-17
US27312709P 2009-07-30 2009-07-30
PCT/JP2010/062037 WO2011007856A1 (ja) 2009-07-17 2010-07-16 トリアゾロピリジン化合物、ならびにそのプロリル水酸化酵素阻害剤およびエリスロポエチン産生誘導剤としての作用

Publications (1)

Publication Number Publication Date
HRP20140705T1 true HRP20140705T1 (hr) 2014-09-12

Family

ID=43449466

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20140705AT HRP20140705T1 (hr) 2009-07-17 2010-07-16 Spoj triazolopiridina i njegovo djelovanje kao inhibitora prolil hidroksilaze i induktora proizvodnje eritropoetina

Country Status (28)

Country Link
US (3) US8283465B2 (enExample)
EP (3) EP3594213A1 (enExample)
JP (9) JP5021797B2 (enExample)
KR (4) KR20180042443A (enExample)
CN (1) CN102471337B (enExample)
AR (1) AR077417A1 (enExample)
AU (1) AU2010271732B2 (enExample)
BR (1) BR112012001157A2 (enExample)
CA (1) CA2768505C (enExample)
CO (1) CO6430426A2 (enExample)
DK (1) DK2455381T5 (enExample)
ES (1) ES2477968T3 (enExample)
HR (1) HRP20140705T1 (enExample)
IL (1) IL217541A (enExample)
ME (1) ME01858B (enExample)
MX (1) MX2012000766A (enExample)
MY (1) MY160814A (enExample)
NZ (1) NZ598242A (enExample)
PE (1) PE20120629A1 (enExample)
PL (1) PL2455381T3 (enExample)
PT (1) PT2455381E (enExample)
RS (1) RS53499B1 (enExample)
RU (1) RU2538963C2 (enExample)
SG (1) SG178049A1 (enExample)
SI (1) SI2455381T1 (enExample)
SM (1) SMT201500122B (enExample)
TW (1) TWI485150B (enExample)
WO (1) WO2011007856A1 (enExample)

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Also Published As

Publication number Publication date
TWI485150B (zh) 2015-05-21
JP2020111612A (ja) 2020-07-27
JP2024091878A (ja) 2024-07-05
KR20120051704A (ko) 2012-05-22
JP2019019144A (ja) 2019-02-07
NZ598242A (en) 2013-09-27
AU2010271732A1 (en) 2012-03-08
US20160145254A1 (en) 2016-05-26
MY160814A (en) 2017-03-31
ES2477968T3 (es) 2014-07-18
IL217541A0 (en) 2012-02-29
RS53499B1 (sr) 2015-02-27
KR101706803B1 (ko) 2017-02-14
SMT201500122B (it) 2015-07-09
EP3594213A1 (en) 2020-01-15
KR20170018105A (ko) 2017-02-15
EP2455381A4 (en) 2012-12-12
ME01858B (me) 2014-12-20
CA2768505C (en) 2018-06-12
TW201105671A (en) 2011-02-16
JP2012144571A (ja) 2012-08-02
ES2477968T9 (es) 2014-11-13
WO2011007856A1 (ja) 2011-01-20
MX2012000766A (es) 2012-02-08
CN102471337A (zh) 2012-05-23
DK2455381T5 (en) 2015-02-09
PE20120629A1 (es) 2012-05-30
US20110077267A1 (en) 2011-03-31
BR112012001157A2 (pt) 2016-02-23
EP2455381A1 (en) 2012-05-23
JP5021797B2 (ja) 2012-09-12
EP2455381B9 (en) 2014-10-22
PL2455381T3 (pl) 2014-10-31
JP2017214404A (ja) 2017-12-07
KR20180042443A (ko) 2018-04-25
JP2015003933A (ja) 2015-01-08
PT2455381E (pt) 2014-06-24
RU2012105467A (ru) 2013-08-27
US8283465B2 (en) 2012-10-09
CA2768505A1 (en) 2011-01-20
EP2746282A1 (en) 2014-06-25
DK2455381T3 (da) 2014-07-21
AU2010271732B2 (en) 2016-08-25
JP2016040321A (ja) 2016-03-24
KR20230165366A (ko) 2023-12-05
RU2538963C2 (ru) 2015-01-10
JP2022126843A (ja) 2022-08-30
CO6430426A2 (es) 2012-04-30
US20130096155A1 (en) 2013-04-18
EP2455381B1 (en) 2014-05-28
HK1168346A1 (en) 2012-12-28
JP2011037841A (ja) 2011-02-24
CN102471337B (zh) 2014-12-10
IL217541A (en) 2014-07-31
JP6434575B2 (ja) 2018-12-05
SI2455381T1 (sl) 2014-08-29
AR077417A1 (es) 2011-08-24
KR101850661B1 (ko) 2018-04-19
SG178049A1 (en) 2012-03-29

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