KR101679642B1 - Ｐｉ3­키나아제 억제제로서 옥사졸 치환된 인다졸 - Google Patents

Ｐｉ3­키나아제 억제제로서 옥사졸 치환된 인다졸 Download PDF

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KR101679642B1
KR101679642B1 KR1020117028746A KR20117028746A KR101679642B1 KR 101679642 B1 KR101679642 B1 KR 101679642B1 KR 1020117028746 A KR1020117028746 A KR 1020117028746A KR 20117028746 A KR20117028746 A KR 20117028746A KR 101679642 B1 KR101679642 B1 KR 101679642B1
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methyl
oxazol
compound
pharmaceutically acceptable
indazole
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KR20120079852A (ko
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줄리 니콜 햄블린
폴 스펜서 존스
수잔 일레인 킬링
조엘 리
샬롯 제인 미첼
나이젤 제임스 파
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글락소 그룹 리미티드
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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KR1020117028746A 2009-04-30 2010-04-28 Ｐｉ3­키나아제 억제제로서 옥사졸 치환된 인다졸 Expired - Fee Related KR101679642B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17403309P 2009-04-30 2009-04-30
US61/174,033 2009-04-30
PCT/EP2010/055666 WO2010125082A1 (en) 2009-04-30 2010-04-28 Oxazole substituted indazoles as pi3-kinase inhibitors

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KR1020167032300A Division KR101771193B1 (ko) 2009-04-30 2010-04-28 Ｐｉ3­키나아제 억제제로서 옥사졸 치환된 인다졸

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Publication Number Publication Date
KR20120079852A KR20120079852A (ko) 2012-07-13
KR101679642B1 true KR101679642B1 (ko) 2016-11-25

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KR1020167032300A Expired - Fee Related KR101771193B1 (ko) 2009-04-30 2010-04-28 Ｐｉ3­키나아제 억제제로서 옥사졸 치환된 인다졸
KR1020117028746A Expired - Fee Related KR101679642B1 (ko) 2009-04-30 2010-04-28 Ｐｉ3­키나아제 억제제로서 옥사졸 치환된 인다졸

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Families Citing this family (75)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2445199T3 (es) * 2008-06-05 2014-02-28 Glaxo Group Limited Derivados de benzpirazol como inhibidores de PI3-quinasas
ES2526966T3 (es) 2008-06-05 2015-01-19 Glaxo Group Limited Compuestos novedosos
ES2383246T3 (es) 2008-06-05 2012-06-19 Glaxo Group Limited 4-amino-indazoles
ES2542551T3 (es) 2009-03-09 2015-08-06 Glaxo Group Limited 4-Oxadiazol-2-il-indazoles como inhibidores de PI3 cinasas
AU2010243613B2 (en) 2009-04-30 2015-05-07 Glaxo Group Limited Oxazole substituted indazoles as PI3-kinase inhibitors
CN102372675B (zh) * 2010-08-14 2013-12-18 王娜 6-氯-4-碘吲唑及其制备方法与应用
US9102668B2 (en) 2010-09-08 2015-08-11 Glaxo Group Limited Polymorphs and salts
EP2613781B1 (en) 2010-09-08 2016-08-24 GlaxoSmithKline Intellectual Property Development Limited Indazole derivatives for use in the treatment of influenza virus infection
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