KR100637296B1 - 특정 5-알킬-2-아릴아미노페닐아세트산 및 유도체 - Google Patents

특정 5-알킬-2-아릴아미노페닐아세트산 및 유도체 Download PDF

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Publication number
KR100637296B1
KR100637296B1 KR1020007001982A KR20007001982A KR100637296B1 KR 100637296 B1 KR100637296 B1 KR 100637296B1 KR 1020007001982 A KR1020007001982 A KR 1020007001982A KR 20007001982 A KR20007001982 A KR 20007001982A KR 100637296 B1 KR100637296 B1 KR 100637296B1
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KR
South Korea
Prior art keywords
ethyl
methyl
formula
phenylacetic acid
fluoro
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Expired - Lifetime
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KR1020007001982A
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English (en)
Korean (ko)
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KR20010023344A (ko
Inventor
로저 아끼 후지모또
레슬리 윙톤 맥퀴르
벤자민 비로 무그라쥐
죤 헨리 반두저
다퀴앙 츄
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노파르티스 아게
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Application filed by 노파르티스 아게 filed Critical 노파르티스 아게
Publication of KR20010023344A publication Critical patent/KR20010023344A/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/40—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/42—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton with carboxyl groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by saturated carbon chains
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020007001982A 1997-08-28 1998-08-26 특정 5-알킬-2-아릴아미노페닐아세트산 및 유도체 Expired - Lifetime KR100637296B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US6983797P 1997-08-28 1997-08-28
US5780397P 1997-08-28 1997-08-28
US60/069,837 1997-08-28
US60/057,803 1997-08-28
PCT/EP1998/005414 WO1999011605A1 (en) 1997-08-28 1998-08-26 Certain 5-alkyl-2-arylaminophenylacetic acids and derivatives

Publications (2)

Publication Number Publication Date
KR20010023344A KR20010023344A (ko) 2001-03-26
KR100637296B1 true KR100637296B1 (ko) 2006-10-23

Family

ID=26736901

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020007001982A Expired - Lifetime KR100637296B1 (ko) 1997-08-28 1998-08-26 특정 5-알킬-2-아릴아미노페닐아세트산 및 유도체

Country Status (34)

Country Link
US (5) US6291523B1 (enExample)
EP (1) EP1007505B1 (enExample)
JP (1) JP3704470B2 (enExample)
KR (1) KR100637296B1 (enExample)
CN (1) CN1140500C (enExample)
AR (1) AR015157A1 (enExample)
AT (1) ATE237580T1 (enExample)
AU (1) AU743371B2 (enExample)
BR (1) BR9812010B1 (enExample)
CA (1) CA2298033C (enExample)
CO (1) CO4960662A1 (enExample)
CY (1) CY2007020I2 (enExample)
CZ (1) CZ298522B6 (enExample)
DE (4) DE122007000035I1 (enExample)
DK (1) DK1007505T3 (enExample)
ES (1) ES2197508T3 (enExample)
FR (1) FR09C0011I2 (enExample)
HU (1) HU225774B1 (enExample)
ID (1) ID23953A (enExample)
IL (2) IL134498A0 (enExample)
LU (2) LU91346I2 (enExample)
MY (1) MY127881A (enExample)
NL (1) NL300379I2 (enExample)
NO (2) NO326196B1 (enExample)
NZ (1) NZ502669A (enExample)
PE (1) PE108099A1 (enExample)
PL (1) PL194480B1 (enExample)
PT (1) PT1007505E (enExample)
RU (1) RU2186762C2 (enExample)
SI (1) SI1007505T1 (enExample)
SK (1) SK283773B6 (enExample)
TR (1) TR200000447T2 (enExample)
TW (1) TWI250142B (enExample)
WO (1) WO1999011605A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2019031774A1 (ko) * 2017-08-09 2019-02-14 연성정밀화학(주) 라타노프로스틴 부노드의 제조 방법 및 그를 위한 중간체

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