RU2186762C2 - Определенные 5-алкил-2-ариламинофенилуксусные кислоты и их производные - Google Patents

Определенные 5-алкил-2-ариламинофенилуксусные кислоты и их производные Download PDF

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RU2186762C2
RU2186762C2 RU2000107121/04A RU2000107121A RU2186762C2 RU 2186762 C2 RU2186762 C2 RU 2186762C2 RU 2000107121/04 A RU2000107121/04 A RU 2000107121/04A RU 2000107121 A RU2000107121 A RU 2000107121A RU 2186762 C2 RU2186762 C2 RU 2186762C2
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methyl
ethyl
phenylacetic acid
compound
chloro
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RU2000107121/04A
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Russian (ru)
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RU2000107121A (ru
Inventor
Роджер Аки Фуджимото
Лесли Уайтон МАККВАЙР
Бенджамин Биро МАГРЕЙДЖ
Джон Хенри ВАН-ДЮЗЕР
Дацян СЮЙ
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Новартис Аг
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/40—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/42—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton with carboxyl groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by saturated carbon chains
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RU2000107121/04A 1997-08-28 1998-08-26 Определенные 5-алкил-2-ариламинофенилуксусные кислоты и их производные RU2186762C2 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US6983797P 1997-08-28 1997-08-28
US5780397P 1997-08-28 1997-08-28
US60/069,837 1997-08-28
US60/057,803 1997-08-28

Publications (2)

Publication Number Publication Date
RU2000107121A RU2000107121A (ru) 2002-03-10
RU2186762C2 true RU2186762C2 (ru) 2002-08-10

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RU2000107121/04A RU2186762C2 (ru) 1997-08-28 1998-08-26 Определенные 5-алкил-2-ариламинофенилуксусные кислоты и их производные

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US (5) US6291523B1 (enExample)
EP (1) EP1007505B1 (enExample)
JP (1) JP3704470B2 (enExample)
KR (1) KR100637296B1 (enExample)
CN (1) CN1140500C (enExample)
AR (1) AR015157A1 (enExample)
AT (1) ATE237580T1 (enExample)
AU (1) AU743371B2 (enExample)
BR (1) BR9812010B1 (enExample)
CA (1) CA2298033C (enExample)
CO (1) CO4960662A1 (enExample)
CY (1) CY2007020I2 (enExample)
CZ (1) CZ298522B6 (enExample)
DE (4) DE69813570T2 (enExample)
DK (1) DK1007505T3 (enExample)
ES (1) ES2197508T3 (enExample)
FR (1) FR09C0011I2 (enExample)
HU (1) HU225774B1 (enExample)
ID (1) ID23953A (enExample)
IL (2) IL134498A0 (enExample)
LU (2) LU91346I2 (enExample)
MY (1) MY127881A (enExample)
NL (1) NL300379I2 (enExample)
NO (2) NO326196B1 (enExample)
NZ (1) NZ502669A (enExample)
PE (1) PE108099A1 (enExample)
PL (1) PL194480B1 (enExample)
PT (1) PT1007505E (enExample)
RU (1) RU2186762C2 (enExample)
SI (1) SI1007505T1 (enExample)
SK (1) SK283773B6 (enExample)
TR (1) TR200000447T2 (enExample)
TW (1) TWI250142B (enExample)
WO (1) WO1999011605A1 (enExample)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2318497C2 (ru) * 2002-03-07 2008-03-10 Новартис Аг Фармацевтические композиции
RU2439053C1 (ru) * 2010-08-03 2012-01-10 Государственное образовательное учреждение высшего профессионального образования "Пермский государственный университет" Диариламины и способ их получения
RU2454402C2 (ru) * 2006-06-26 2012-06-27 Новартис Аг Производные фенилуксусной кислоты, как ингибиторы цог-2 (циклооксигеназы-2)
RU2822483C1 (ru) * 2021-03-15 2024-07-08 Гуанчжоу Оцусунь Офталмик Биотекнолоджи Ко., Лтд. Пролекарство целекоксиба, способ его получения и применение

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