CN1140500C - 某些5-烷基-2-芳基氨基苯乙酸及其衍生物 - Google Patents

某些5-烷基-2-芳基氨基苯乙酸及其衍生物 Download PDF

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Publication number
CN1140500C
CN1140500C CNB988085208A CN98808520A CN1140500C CN 1140500 C CN1140500 C CN 1140500C CN B988085208 A CNB988085208 A CN B988085208A CN 98808520 A CN98808520 A CN 98808520A CN 1140500 C CN1140500 C CN 1140500C
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CN
China
Prior art keywords
ethyl
methyl
phenylacetic acid
compound
chloro
Prior art date
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Expired - Lifetime
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CNB988085208A
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English (en)
Chinese (zh)
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CN1268112A (zh
Inventor
R��A��Ī��
R·A·福吉莫托
L·W·麦克奎瑞
¸
B·B·穆格拉吉
J·H·范杜泽
许大强
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Swiss Iran Animal Health Care Co Ltd
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Novartis AG
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Publication of CN1268112A publication Critical patent/CN1268112A/zh
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/40—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/42—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton with carboxyl groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by saturated carbon chains
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CNB988085208A 1997-08-28 1998-08-26 某些5-烷基-2-芳基氨基苯乙酸及其衍生物 Expired - Lifetime CN1140500C (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US5780397P 1997-08-28 1997-08-28
US6983797P 1997-08-28 1997-08-28
US60/069,837 1997-08-28
US60/057,803 1997-08-28

Publications (2)

Publication Number Publication Date
CN1268112A CN1268112A (zh) 2000-09-27
CN1140500C true CN1140500C (zh) 2004-03-03

Family

ID=26736901

Family Applications (1)

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CNB988085208A Expired - Lifetime CN1140500C (zh) 1997-08-28 1998-08-26 某些5-烷基-2-芳基氨基苯乙酸及其衍生物

Country Status (34)

Country Link
US (5) US6291523B1 (enExample)
EP (1) EP1007505B1 (enExample)
JP (1) JP3704470B2 (enExample)
KR (1) KR100637296B1 (enExample)
CN (1) CN1140500C (enExample)
AR (1) AR015157A1 (enExample)
AT (1) ATE237580T1 (enExample)
AU (1) AU743371B2 (enExample)
BR (1) BR9812010B1 (enExample)
CA (1) CA2298033C (enExample)
CO (1) CO4960662A1 (enExample)
CY (1) CY2007020I1 (enExample)
CZ (1) CZ298522B6 (enExample)
DE (4) DE122009000013I1 (enExample)
DK (1) DK1007505T3 (enExample)
ES (1) ES2197508T3 (enExample)
FR (1) FR09C0011I2 (enExample)
HU (1) HU225774B1 (enExample)
ID (1) ID23953A (enExample)
IL (2) IL134498A0 (enExample)
LU (2) LU91346I2 (enExample)
MY (1) MY127881A (enExample)
NL (1) NL300379I2 (enExample)
NO (2) NO326196B1 (enExample)
NZ (1) NZ502669A (enExample)
PE (1) PE108099A1 (enExample)
PL (1) PL194480B1 (enExample)
PT (1) PT1007505E (enExample)
RU (1) RU2186762C2 (enExample)
SI (1) SI1007505T1 (enExample)
SK (1) SK283773B6 (enExample)
TR (1) TR200000447T2 (enExample)
TW (1) TWI250142B (enExample)
WO (1) WO1999011605A1 (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102812000A (zh) * 2010-01-06 2012-12-05 潘米拉制药公司 Dp2拮抗剂及其用途
CN109503399A (zh) * 2018-12-29 2019-03-22 江苏天和制药有限公司 一种罗本考昔的制备方法

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