JPS58135883A - 新規化合物の３―アミノ―２―オキソアゼチジン―１―スルホン酸の誘導体及びそれらの製造法 - Google Patents

新規化合物の３―アミノ―２―オキソアゼチジン―１―スルホン酸の誘導体及びそれらの製造法

Info

Publication number
JPS58135883A
JPS58135883A JP57184814A JP18481482A JPS58135883A JP S58135883 A JPS58135883 A JP S58135883A JP 57184814 A JP57184814 A JP 57184814A JP 18481482 A JP18481482 A JP 18481482A JP S58135883 A JPS58135883 A JP S58135883A
Authority
JP
Japan
Prior art keywords
group
compound
formula
atom
water
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP57184814A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0471073B2 (fr
Inventor
ルネ・エ−ム
アラン・ボネ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Publication of JPS58135883A publication Critical patent/JPS58135883A/ja
Publication of JPH0471073B2 publication Critical patent/JPH0471073B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
JP57184814A 1981-10-23 1982-10-22 新規化合物の３―アミノ―２―オキソアゼチジン―１―スルホン酸の誘導体及びそれらの製造法 Granted JPS58135883A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8119946A FR2515182B1 (fr) 1981-10-23 1981-10-23 Nouveaux produits derives de l'acide 3-amino 2-oxo azetidine 1-sulfamique, leur procede de preparation, leur application comme medicaments et les produits intermediaires necessaires a leur preparation
FR81-19946 1981-10-23

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP3122828A Division JPH0730018B2 (ja) 1981-10-23 1991-04-26 新規化合物の３−アミノ−２−オキソアゼチジン誘導体及びそれらの製造法

Publications (2)

Publication Number Publication Date
JPS58135883A true JPS58135883A (ja) 1983-08-12
JPH0471073B2 JPH0471073B2 (fr) 1992-11-12

Family

ID=9263337

Family Applications (2)

Application Number Title Priority Date Filing Date
JP57184814A Granted JPS58135883A (ja) 1981-10-23 1982-10-22 新規化合物の３―アミノ―２―オキソアゼチジン―１―スルホン酸の誘導体及びそれらの製造法
JP3122828A Expired - Lifetime JPH0730018B2 (ja) 1981-10-23 1991-04-26 新規化合物の３−アミノ−２−オキソアゼチジン誘導体及びそれらの製造法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP3122828A Expired - Lifetime JPH0730018B2 (ja) 1981-10-23 1991-04-26 新規化合物の３−アミノ−２−オキソアゼチジン誘導体及びそれらの製造法

Country Status (12)

Country Link
JP (2) JPS58135883A (fr)
AT (1) AT382150B (fr)
BE (1) BE894785A (fr)
CA (1) CA1201439A (fr)
CH (1) CH655317A5 (fr)
DE (1) DE3239157C2 (fr)
FR (1) FR2515182B1 (fr)
GB (1) GB2111482B (fr)
IT (1) IT1157233B (fr)
LU (1) LU84434A1 (fr)
NL (1) NL8204089A (fr)
SE (2) SE461655B (fr)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58208288A (ja) * 1982-05-31 1983-12-03 Banyu Pharmaceut Co Ltd ２−オキソ−１−アゼチジンスルホン酸誘導体
JPS59175490A (ja) * 1983-03-24 1984-10-04 Banyu Pharmaceut Co Ltd ２−オキソ−１−アゼチジンスルホン酸誘導体
JPS59231086A (ja) * 1983-06-15 1984-12-25 Teikoku Hormone Mfg Co Ltd ４−メトキシエチル−２−アゼチジノン−１−スルホン酸誘導体
JPS6097978A (ja) * 1983-10-31 1985-05-31 Otsuka Chem Co Ltd ３−アシルアミノ−４−メチル−２−アゼチジノン−１−スルホン酸誘導体，その製造方法および該誘導体を含有する薬剤
JPS60202882A (ja) * 1984-03-27 1985-10-14 Teikoku Hormone Mfg Co Ltd 新規な２−アゼチジノン−１−スルホン酸誘導体
US6677028B1 (en) 1999-09-10 2004-01-13 3M Innovative Properties Company Retroreflective articles having multilayer films and methods of manufacturing same

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1982001873A1 (fr) * 1980-12-05 1982-06-10 Takeda Chemical Industries Ltd Derives 1-sulfo-2-oxoazetidine et leur procede de preparation
US4673739A (en) * 1980-12-05 1987-06-16 Takeda Chemical Industries, Ltd. 4-carbamoyloxymethyl-1-sulfo-2-oxoazetidine derivatives and their production
US4675397A (en) * 1980-12-05 1987-06-23 Takeda Chemical Industries, Ltd. 1-sulfo-2-oxoazetidine derivatives and their production
MX7096E (es) * 1980-12-05 1987-06-19 Takeda Chemical Industries Ltd Metodo para preparacion de derivados de 2-oxoazetidina
US4572801A (en) * 1981-04-30 1986-02-25 Takeda Chemical Industries, Ltd. 4-Carbamoyloxymethyl-1-sulfo-2-oxoazetidine derivatives and their production
FR2558467B2 (fr) * 1981-10-23 1987-03-20 Roussel Uclaf Nouveau produit derive de l'acide 3-amino 2-oxo azetidine 1-sulfamique, son procede de preparation, son application comme medicament et un produit intermediaire necessaire a sa preparation
US4443374A (en) * 1982-02-01 1984-04-17 E. R. Squibb & Sons, Inc. Process for preparing (3S)-3-[[(2-amino-4-thiazolyl)[(1-carboxy-1-methylethoxy)imino]-acetyl]amino]-2-oxo-1-azetidinesulfonic acid, and 4-substituted derivatives
DE3377061D1 (en) * 1982-06-03 1988-07-21 Hoffmann La Roche Process for the preparation of 1-sulfo-2-oxoazetidine derivatives
DE3372768D1 (de) * 1982-06-03 1987-09-03 Hoffmann La Roche 1-sulfo-2-oxoazetidine derivatives
JPS5982359A (ja) * 1982-11-02 1984-05-12 Kanegafuchi Chem Ind Co Ltd ４（Ｒ）配位光学活性β−ラクタム化合物の製法
EP0117053A1 (fr) * 1983-02-10 1984-08-29 Ajinomoto Co., Inc. Dérivés de l'azétidinone
US4501697A (en) * 1983-06-17 1985-02-26 E. R. Squibb & Sons, Inc. 4-[[(Amidomethyl)oxy]methyl]-2-oxo-1-azetidinesulfonic acid salts
WO1986006722A1 (fr) * 1985-05-09 1986-11-20 The Upjohn Company Monobactames substitues par du carbonate servant d'antibiotiques
US4837318A (en) * 1985-05-09 1989-06-06 The Upjohn Company Carbonate substituted monobactams as antibiotics
DE19642530A1 (de) * 1996-10-15 1998-04-16 Bayer Ag Halogenalkoximinoessigsäureamide

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57131758A (en) * 1980-12-05 1982-08-14 Takeda Chem Ind Ltd 1-sulfo-2-oxoazetidine derivative, its preparation and use

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK194776A (da) * 1975-05-05 1976-11-06 Smithkline Corp Antibakterielle midler og mellemprodukter dertil
US4166816A (en) * 1975-05-05 1979-09-04 Smithkline Corporation Methods and intermediates for preparing cis-4-oxoazetidine intermediates
FR2361885A1 (fr) * 1975-09-03 1978-03-17 Smithkline Corp Analogues de la penicilline, leurs intermediaires et procedes pour leur obtention
US4085100A (en) * 1976-11-01 1978-04-18 Smithkline Corporation Intermediate for dephthaloylation of azetidinone compounds
US4144333A (en) * 1976-11-15 1979-03-13 Smithkline Corporation Monocyclic beta-lactams with antibacterial activity
EP0005507A1 (fr) * 1978-05-18 1979-11-28 Ciba-Geigy Ag Procédé pour la scission de dérivés de 3-(2-hydroxyimino-acétylamino)-2-oxo-azétidine et les composés obtenus
EP0021678B1 (fr) * 1979-06-08 1984-11-07 Takeda Chemical Industries, Ltd. Dérivés de 1-sulfo-2-azétidinone, leur préparation et leurs compositions pharmaceutiques
NZ205240A (en) * 1980-02-07 1984-07-31 Squibb & Sons Inc Sulphonamide derivatives,being starting materials for producing beta-lactams
WO1982001873A1 (fr) * 1980-12-05 1982-06-10 Takeda Chemical Industries Ltd Derives 1-sulfo-2-oxoazetidine et leur procede de preparation
JPS58189176A (ja) 1982-04-30 1983-11-04 Takeda Chem Ind Ltd １−スルホ−２−アゼチジノン誘導体およびその製造法
JPS58210061A (ja) 1982-05-31 1983-12-07 Takeda Chem Ind Ltd １−スルホ−２−オキソアゼチジン誘導体、その製造法および用途
EP0076758B1 (fr) * 1981-10-05 1987-01-07 E.R. Squibb & Sons, Inc. Dérivés 4-éther d'acides 2-azétidinone-1-sulfoniques
AU564150B2 (en) * 1982-04-30 1987-08-06 Takeda Chemical Industries Ltd. 1-sulfo-2-azetidinone derivatives
HU189290B (en) * 1982-05-31 1986-06-30 Banyu Pharmaceutical Co Ltd,Jp Process for preparing new 2-oxo-1-azetidine-sulphonic acid derivatives and pharmaceutically acceptable salts thereof, further pharmaceutical compositions containing such derivatives as active substances
JPS59175490A (ja) * 1983-03-24 1984-10-04 Banyu Pharmaceut Co Ltd ２−オキソ−１−アゼチジンスルホン酸誘導体
JPS58208288A (ja) * 1982-05-31 1983-12-03 Banyu Pharmaceut Co Ltd ２−オキソ−１−アゼチジンスルホン酸誘導体

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57131758A (en) * 1980-12-05 1982-08-14 Takeda Chem Ind Ltd 1-sulfo-2-oxoazetidine derivative, its preparation and use

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58208288A (ja) * 1982-05-31 1983-12-03 Banyu Pharmaceut Co Ltd ２−オキソ−１−アゼチジンスルホン酸誘導体
JPH0343272B2 (fr) * 1982-05-31 1991-07-01 Banyu Pharma Co Ltd
JPS59175490A (ja) * 1983-03-24 1984-10-04 Banyu Pharmaceut Co Ltd ２−オキソ−１−アゼチジンスルホン酸誘導体
JPH0340028B2 (fr) * 1983-03-24 1991-06-17
JPS59231086A (ja) * 1983-06-15 1984-12-25 Teikoku Hormone Mfg Co Ltd ４−メトキシエチル−２−アゼチジノン−１−スルホン酸誘導体
JPS6097978A (ja) * 1983-10-31 1985-05-31 Otsuka Chem Co Ltd ３−アシルアミノ−４−メチル−２−アゼチジノン−１−スルホン酸誘導体，その製造方法および該誘導体を含有する薬剤
JPH0541634B2 (fr) * 1983-10-31 1993-06-24 Otsuka Kagaku Kk
JPS60202882A (ja) * 1984-03-27 1985-10-14 Teikoku Hormone Mfg Co Ltd 新規な２−アゼチジノン−１−スルホン酸誘導体
US6677028B1 (en) 1999-09-10 2004-01-13 3M Innovative Properties Company Retroreflective articles having multilayer films and methods of manufacturing same

Also Published As

Publication number Publication date
FR2515182B1 (fr) 1986-05-09
IT8249341A0 (it) 1982-10-22
SE8205870D0 (sv) 1982-10-15
DE3239157C2 (de) 1994-04-28
SE8205870L (sv) 1983-04-24
IT1157233B (it) 1987-02-11
LU84434A1 (fr) 1983-06-13
SE8702330D0 (sv) 1987-06-04
NL8204089A (nl) 1983-05-16
JPH0471073B2 (fr) 1992-11-12
GB2111482A (en) 1983-07-06
SE461655B (sv) 1990-03-12
CH655317A5 (fr) 1986-04-15
AT382150B (de) 1987-01-12
FR2515182A1 (fr) 1983-04-29
SE500849C2 (sv) 1994-09-19
JPH04234844A (ja) 1992-08-24
BE894785A (fr) 1983-04-22
CA1201439A (fr) 1986-03-04
ATA391182A (de) 1986-06-15
DE3239157A1 (de) 1983-05-05
GB2111482B (en) 1985-11-06
JPH0730018B2 (ja) 1995-04-05
SE8702330L (sv) 1987-06-04

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