JP6914834B2 - (S)−N−(5−((R)−2−(2,5−ジフルオロフェニル)−ピロリジン−1−イル)−ピラゾロ[1,5−a]ピリミジン−3−イル)−3−ヒドロキシピロリジン−1−カルボキサミド硫酸水素塩の結晶形 - Google Patents

(S)−N−(5−((R)−2−(2,5−ジフルオロフェニル)−ピロリジン−1−イル)−ピラゾロ[1,5−a]ピリミジン−3−イル)−3−ヒドロキシピロリジン−1−カルボキサミド硫酸水素塩の結晶形 Download PDF

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JP6914834B2
JP6914834B2 JP2017526116A JP2017526116A JP6914834B2 JP 6914834 B2 JP6914834 B2 JP 6914834B2 JP 2017526116 A JP2017526116 A JP 2017526116A JP 2017526116 A JP2017526116 A JP 2017526116A JP 6914834 B2 JP6914834 B2 JP 6914834B2
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trka
crystalline form
trk
cancer
composition
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アリシャ ビー. アリゴ,
アリシャ ビー. アリゴ,
デリック ユルンスト,
デリック ユルンスト,
カリード シャー,
カリード シャー,
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アレイ バイオファーマ インコーポレイテッド
アレイ バイオファーマ インコーポレイテッド
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JP2017526116A 2014-11-16 2015-11-16 (S)−N−(5−((R)−2−(2,5−ジフルオロフェニル)−ピロリジン−1−イル)−ピラゾロ[1,5−a]ピリミジン−3−イル)−3−ヒドロキシピロリジン−1−カルボキサミド硫酸水素塩の結晶形 Active JP6914834B2 (ja)

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JP2021116073A JP2021169496A (ja) 2014-11-16 2021-07-14 (S)−N−(5−((R)−2−(2,5−ジフルオロフェニル)−ピロリジン−1−イル)−ピラゾロ[1,5−a]ピリミジン−3−イル)−3−ヒドロキシピロリジン−1−カルボキサミド硫酸水素塩の結晶形

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US201462080374P 2014-11-16 2014-11-16
US62/080,374 2014-11-16
US201562169545P 2015-06-01 2015-06-01
US62/169,545 2015-06-01
PCT/US2015/060953 WO2016077841A1 (en) 2014-11-16 2015-11-16 Crystalline form of (s)-n-(5-((r)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide hydrogen sulfate

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JP2017535550A5 JP2017535550A5 (ko) 2018-12-27
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JP2021116073A Pending JP2021169496A (ja) 2014-11-16 2021-07-14 (S)−N−(5−((R)−2−(2,5−ジフルオロフェニル)−ピロリジン−1−イル)−ピラゾロ[1,5−a]ピリミジン−3−イル)−3−ヒドロキシピロリジン−1−カルボキサミド硫酸水素塩の結晶形

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KR (1) KR102649887B1 (ko)
CN (2) CN107428760B (ko)
AU (1) AU2015346046B2 (ko)
BR (1) BR112017010141A2 (ko)
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UA (1) UA123044C2 (ko)
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