JP5138938B2 - Ret調節剤の開発のための化合物および方法 - Google Patents

Ret調節剤の開発のための化合物および方法 Download PDF

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JP5138938B2
JP5138938B2 JP2006545481A JP2006545481A JP5138938B2 JP 5138938 B2 JP5138938 B2 JP 5138938B2 JP 2006545481 A JP2006545481 A JP 2006545481A JP 2006545481 A JP2006545481 A JP 2006545481A JP 5138938 B2 JP5138938 B2 JP 5138938B2
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optionally substituted
compound
ret
binding
aryl
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JP2007521334A (ja
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イブラヒム,プラバ
ウェスト,ブライアン
クマール,アブヒナブ
クルプカ,ハイケ
ズッカーマン,レベッカ
ジュー,ヨン
ジャン,ジャジョン
ジャン,チャオ
ネスピ,マリカ
マモ,シュメイエ
ハート,クラレンス,アール
ハベッツ,ガストン
ブリマー,ライアン
アーティス,リチャード,ディーン
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Plexxikon Inc
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
JP2006545481A 2003-12-19 2004-12-17 Ret調節剤の開発のための化合物および方法 Active JP5138938B2 (ja)

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US53128103P 2003-12-19 2003-12-19
US60/531,281 2003-12-19
US55858104P 2004-03-31 2004-03-31
US60/558,581 2004-03-31
PCT/US2004/042470 WO2005062795A2 (en) 2003-12-19 2004-12-17 Compounds and methods for development of ret modulators

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JP2007521334A JP2007521334A (ja) 2007-08-02
JP5138938B2 true JP5138938B2 (ja) 2013-02-06

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PT (1) PT1696920E (US07504509-20090317-C00001.png)
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US8067434B2 (en) 2011-11-29
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EP1696920A4 (en) 2009-09-02
CN1925855A (zh) 2007-03-07
US20070049615A1 (en) 2007-03-01
CA2550361C (en) 2014-04-29
SI1696920T1 (sl) 2015-02-27
PT1696920E (pt) 2015-01-14
DK1696920T3 (en) 2015-01-19
US7504509B2 (en) 2009-03-17
CN1925855B (zh) 2010-06-16
AU2004308299B2 (en) 2011-11-24
EP1696920B1 (en) 2014-10-29
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HK1094878A1 (en) 2007-04-13
JP2007521334A (ja) 2007-08-02
CA2550361A1 (en) 2005-07-14
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AU2004308299A1 (en) 2005-07-14
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WO2005062795A3 (en) 2006-02-09
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