JP4364637B2 - 新規なベンゾ縮合へテロ環化合物 - Google Patents

新規なベンゾ縮合へテロ環化合物 Download PDF

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Publication number
JP4364637B2
JP4364637B2 JP2003518554A JP2003518554A JP4364637B2 JP 4364637 B2 JP4364637 B2 JP 4364637B2 JP 2003518554 A JP2003518554 A JP 2003518554A JP 2003518554 A JP2003518554 A JP 2003518554A JP 4364637 B2 JP4364637 B2 JP 4364637B2
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phenyl
benzo
lower alkyl
oxo
yloxy
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JP2005502644A (ja
JP2005502644A5 (enExample
Inventor
ボリィ マーチン
ボス クリストフ
クローゼル マーチン
フィシュリ ウオルター
ウィラー トーマス
マルフート ジュデット
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Actelion Pharmaceuticals Ltd
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Actelion Pharmaceuticals Ltd
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    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16Benzazepines; Hydrogenated benzazepines
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JP2003518554A 2001-08-09 2002-07-31 新規なベンゾ縮合へテロ環化合物 Expired - Fee Related JP4364637B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP0109235 2001-08-09
PCT/EP2002/008523 WO2003013545A1 (en) 2001-08-09 2002-07-31 Novel benzo-fused heterocycles as endothelin antagonisits

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JP2005502644A JP2005502644A (ja) 2005-01-27
JP2005502644A5 JP2005502644A5 (enExample) 2006-01-12
JP4364637B2 true JP4364637B2 (ja) 2009-11-18

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US (1) US7238685B2 (enExample)
JP (1) JP4364637B2 (enExample)
KR (1) KR100909122B1 (enExample)
CN (1) CN100418955C (enExample)
AR (1) AR036386A1 (enExample)
AU (1) AU2002328999B8 (enExample)
BR (1) BR0211729A (enExample)
CA (1) CA2454417A1 (enExample)
HU (1) HUP0401107A3 (enExample)
IL (1) IL159963A0 (enExample)
MX (1) MXPA04001252A (enExample)
NO (1) NO20040563L (enExample)
NZ (1) NZ530741A (enExample)
WO (1) WO2003013545A1 (enExample)
ZA (1) ZA200400803B (enExample)

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DE602005003951T4 (de) 2004-05-14 2012-10-11 Millennium Pharmaceuticals, Inc. Verbindungen und verfahren zur inhibierung der mitotischen progression durch hemmung von aurorakinase
WO2008021038A2 (en) 2006-08-09 2008-02-21 Millennium Pharmaceuticals, Inc. Pyridobenzazepine compounds and methods for inhibiting mitotic progression
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WO2003013545A1 (en) 2003-02-20
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AU2002328999B2 (en) 2008-05-15
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