CA2454417A1 - Novel benzo-fused heterocycles as endothelin antagonists - Google Patents

Novel benzo-fused heterocycles as endothelin antagonists Download PDF

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Publication number
CA2454417A1
CA2454417A1 CA002454417A CA2454417A CA2454417A1 CA 2454417 A1 CA2454417 A1 CA 2454417A1 CA 002454417 A CA002454417 A CA 002454417A CA 2454417 A CA2454417 A CA 2454417A CA 2454417 A1 CA2454417 A1 CA 2454417A1
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CA
Canada
Prior art keywords
phenyl
benzo
lower alkyl
oxo
acetic acid
Prior art date
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Abandoned
Application number
CA002454417A
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English (en)
French (fr)
Inventor
Martin Bolli
Martine Clozel
Christoph Boss
Judith Marfurt
Thomas Weller
Walter Fischli
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Actelion Pharmaceuticals Ltd
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Individual
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8164539&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CA2454417(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Individual filed Critical Individual
Publication of CA2454417A1 publication Critical patent/CA2454417A1/en
Abandoned legal-status Critical Current

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    • C07D223/16—Benzazepines; Hydrogenated benzazepines
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CA002454417A 2001-08-09 2002-07-31 Novel benzo-fused heterocycles as endothelin antagonists Abandoned CA2454417A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EPPCT/EP01/09235 2001-08-09
EP0109235 2001-08-09
PCT/EP2002/008523 WO2003013545A1 (en) 2001-08-09 2002-07-31 Novel benzo-fused heterocycles as endothelin antagonisits

Publications (1)

Publication Number Publication Date
CA2454417A1 true CA2454417A1 (en) 2003-02-20

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Application Number Title Priority Date Filing Date
CA002454417A Abandoned CA2454417A1 (en) 2001-08-09 2002-07-31 Novel benzo-fused heterocycles as endothelin antagonists

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US (1) US7238685B2 (enExample)
JP (1) JP4364637B2 (enExample)
KR (1) KR100909122B1 (enExample)
CN (1) CN100418955C (enExample)
AR (1) AR036386A1 (enExample)
AU (1) AU2002328999B8 (enExample)
BR (1) BR0211729A (enExample)
CA (1) CA2454417A1 (enExample)
HU (1) HUP0401107A3 (enExample)
IL (1) IL159963A0 (enExample)
MX (1) MXPA04001252A (enExample)
NO (1) NO20040563L (enExample)
NZ (1) NZ530741A (enExample)
WO (1) WO2003013545A1 (enExample)
ZA (1) ZA200400803B (enExample)

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WO2008021038A2 (en) 2006-08-09 2008-02-21 Millennium Pharmaceuticals, Inc. Pyridobenzazepine compounds and methods for inhibiting mitotic progression
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