HUP0401107A3 - Novel benzo-fused heterocycles, their use process for their preparation and pharmaceutical compositions containing them - Google Patents

Novel benzo-fused heterocycles, their use process for their preparation and pharmaceutical compositions containing them

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Publication number
HUP0401107A3
HUP0401107A3 HU0401107A HUP0401107A HUP0401107A3 HU P0401107 A3 HUP0401107 A3 HU P0401107A3 HU 0401107 A HU0401107 A HU 0401107A HU P0401107 A HUP0401107 A HU P0401107A HU P0401107 A3 HUP0401107 A3 HU P0401107A3
Authority
HU
Hungary
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
use process
fused heterocycles
Prior art date
Application number
HU0401107A
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English (en)
Hungarian (hu)
Original Assignee
Actelion Pharmaceuticals Ltd
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8164539&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUP0401107(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of HUP0401107A2 publication Critical patent/HUP0401107A2/hu
Publication of HUP0401107A3 publication Critical patent/HUP0401107A3/hu

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    • C07ORGANIC CHEMISTRY
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    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16Benzazepines; Hydrogenated benzazepines
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    • C07D217/14Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
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    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
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    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
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    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

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HU0401107A 2001-08-09 2002-07-31 Novel benzo-fused heterocycles, their use process for their preparation and pharmaceutical compositions containing them HUP0401107A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP0109235 2001-08-09
PCT/EP2002/008523 WO2003013545A1 (en) 2001-08-09 2002-07-31 Novel benzo-fused heterocycles as endothelin antagonisits

Publications (2)

Publication Number Publication Date
HUP0401107A2 HUP0401107A2 (hu) 2004-08-30
HUP0401107A3 true HUP0401107A3 (en) 2004-10-28

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HU0401107A HUP0401107A3 (en) 2001-08-09 2002-07-31 Novel benzo-fused heterocycles, their use process for their preparation and pharmaceutical compositions containing them

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US (1) US7238685B2 (enExample)
JP (1) JP4364637B2 (enExample)
KR (1) KR100909122B1 (enExample)
CN (1) CN100418955C (enExample)
AR (1) AR036386A1 (enExample)
AU (1) AU2002328999B8 (enExample)
BR (1) BR0211729A (enExample)
CA (1) CA2454417A1 (enExample)
HU (1) HUP0401107A3 (enExample)
IL (1) IL159963A0 (enExample)
MX (1) MXPA04001252A (enExample)
NO (1) NO20040563L (enExample)
NZ (1) NZ530741A (enExample)
WO (1) WO2003013545A1 (enExample)
ZA (1) ZA200400803B (enExample)

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DE602005003951T4 (de) 2004-05-14 2012-10-11 Millennium Pharmaceuticals, Inc. Verbindungen und verfahren zur inhibierung der mitotischen progression durch hemmung von aurorakinase
WO2008021038A2 (en) 2006-08-09 2008-02-21 Millennium Pharmaceuticals, Inc. Pyridobenzazepine compounds and methods for inhibiting mitotic progression
CL2007003244A1 (es) 2006-11-16 2008-04-04 Millennium Pharm Inc Compuestos derivados de pirimido[5,4-d][2]benzazepina; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento del cancer.
WO2008108445A1 (ja) 2007-03-07 2008-09-12 Takeda Pharmaceutical Company Limited ベンゾオキサゼピン誘導体およびその用途
MX2009011923A (es) * 2007-05-10 2009-11-18 Amr Technology Inc Tetrahidrobenzo-1,4-diazepinas aril- y heteroaril-sustituidas y uso de las mismas para bloquear reabsorcion de norepinefrina, dopamina y serotonina.
AU2008265655B2 (en) 2007-06-21 2014-02-06 Cara Therapeutics, Inc. Substituted imidazoheterocycles
US8119629B2 (en) 2007-10-03 2012-02-21 Bristol-Meyers Squibb Company Carboxamide GABAA α2 modulators
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RU2535032C2 (ru) 2008-12-22 2014-12-10 Милленниум Фармасьютикалз, Инк. Сочетание ингибиторов аврора киназы и анти-cd 20 антител
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