ZA200400803B - Novel benzo-fused heterocycles as endothelin antagonists. - Google Patents

Novel benzo-fused heterocycles as endothelin antagonists.

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Publication number
ZA200400803B
ZA200400803B ZA200400803A ZA200400803A ZA200400803B ZA 200400803 B ZA200400803 B ZA 200400803B ZA 200400803 A ZA200400803 A ZA 200400803A ZA 200400803 A ZA200400803 A ZA 200400803A ZA 200400803 B ZA200400803 B ZA 200400803B
Authority
ZA
South Africa
Prior art keywords
endothelin antagonists
fused heterocycles
novel benzo
benzo
novel
Prior art date
Application number
ZA200400803A
Other languages
English (en)
Inventor
Martin Bolli
Martine Clozel
Thomas Weller
Christoph Boss
Walter Fischli
Judith Marfurt
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8164539&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200400803(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of ZA200400803B publication Critical patent/ZA200400803B/xx

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    • C07D223/16Benzazepines; Hydrogenated benzazepines
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ZA200400803A 2001-08-09 2004-01-30 Novel benzo-fused heterocycles as endothelin antagonists. ZA200400803B (en)

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Application Number Priority Date Filing Date Title
EP0109235 2001-08-09

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US (1) US7238685B2 (enExample)
JP (1) JP4364637B2 (enExample)
KR (1) KR100909122B1 (enExample)
CN (1) CN100418955C (enExample)
AR (1) AR036386A1 (enExample)
AU (1) AU2002328999B8 (enExample)
BR (1) BR0211729A (enExample)
CA (1) CA2454417A1 (enExample)
HU (1) HUP0401107A3 (enExample)
IL (1) IL159963A0 (enExample)
MX (1) MXPA04001252A (enExample)
NO (1) NO20040563L (enExample)
NZ (1) NZ530741A (enExample)
WO (1) WO2003013545A1 (enExample)
ZA (1) ZA200400803B (enExample)

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WO2008108445A1 (ja) 2007-03-07 2008-09-12 Takeda Pharmaceutical Company Limited ベンゾオキサゼピン誘導体およびその用途
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US8119629B2 (en) 2007-10-03 2012-02-21 Bristol-Meyers Squibb Company Carboxamide GABAA α2 modulators
WO2010068520A2 (en) * 2008-12-11 2010-06-17 Cara Therapeutics, Inc. Substituted imidazoheterocycle derivatives
RU2535032C2 (ru) 2008-12-22 2014-12-10 Милленниум Фармасьютикалз, Инк. Сочетание ингибиторов аврора киназы и анти-cd 20 антител
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CN104031049A (zh) 2010-02-19 2014-09-10 米伦纽姆医药公司 极光激酶抑制剂的结晶形式
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JP4364637B2 (ja) 2009-11-18
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