JP2020506903A5 - - Google Patents
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- JP2020506903A5 JP2020506903A5 JP2019538585A JP2019538585A JP2020506903A5 JP 2020506903 A5 JP2020506903 A5 JP 2020506903A5 JP 2019538585 A JP2019538585 A JP 2019538585A JP 2019538585 A JP2019538585 A JP 2019538585A JP 2020506903 A5 JP2020506903 A5 JP 2020506903A5
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762449242P | 2017-01-23 | 2017-01-23 | |
| US62/449,242 | 2017-01-23 | ||
| PCT/IB2018/050128 WO2018134698A1 (en) | 2017-01-23 | 2018-01-09 | Heterocyclic spiro compounds as magl inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2020506903A JP2020506903A (ja) | 2020-03-05 |
| JP2020506903A5 true JP2020506903A5 (enExample) | 2021-02-12 |
Family
ID=61028112
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019538585A Withdrawn JP2020506903A (ja) | 2017-01-23 | 2018-01-09 | Ｍａｇｌ阻害薬としての複素環式スピロ化合物 |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US20180208608A1 (enExample) |
| EP (1) | EP3571202B1 (enExample) |
| JP (1) | JP2020506903A (enExample) |
| KR (1) | KR20190097242A (enExample) |
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| US10927105B1 (en) | 2017-05-23 | 2021-02-23 | Lundbeck La Jolla Research Center, Inc. | Pyrazole MAGL inhibitors |
| JP7189143B2 (ja) * | 2017-09-29 | 2022-12-13 | 武田薬品工業株式会社 | 複素環化合物 |
| US10662159B2 (en) * | 2017-11-22 | 2020-05-26 | Makscientific, Llc | ABHD6 and dual ABHD6/MGL inhibitors and their uses |
| WO2019134985A1 (en) | 2018-01-08 | 2019-07-11 | F. Hoffmann-La Roche Ag | Octahydropyrido[1,2-alpha]pyrazines as magl inhibitors |
| MX2021000549A (es) * | 2018-07-19 | 2021-03-25 | Pfizer | Compuestos espiro heterociclicos como inhibidores de magl. |
| RS67557B1 (sr) * | 2018-08-24 | 2026-01-30 | Pharmacosmos Holding As | Unapređena sinteza 1,4-diazaspiro[5.5]undekan-3-ona |
| TW202035409A (zh) | 2018-09-28 | 2020-10-01 | 比利時商健生藥品公司 | 單醯基甘油脂肪酶調節劑 |
| MY205440A (en) | 2018-09-28 | 2024-10-21 | Janssen Pharmaceutica Nv | Monoacylglycerol lipase modulators |
| KR20210097734A (ko) * | 2018-11-28 | 2021-08-09 | 하. 룬드벡 아크티에셀스카브 | Magl 저해제에 의해 질병을 치료하는 방법 |
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| IL301492A (en) | 2020-09-22 | 2023-05-01 | Janssen Pharmaceutica Nv | Cyclobutyl amide monoacylglycerol lipase modulators |
| US12029718B2 (en) | 2021-11-09 | 2024-07-09 | Cct Sciences, Llc | Process for production of essentially pure delta-9-tetrahydrocannabinol |
| TWI904281B (zh) * | 2020-11-13 | 2025-11-11 | 丹麥商Ｈ 朗德貝克公司 | Magl抑制劑 |
| WO2022135462A1 (zh) * | 2020-12-22 | 2022-06-30 | 鲁南制药集团股份有限公司 | Magl抑制剂的医药用途 |
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-
2018
- 2018-01-09 EP EP18701578.9A patent/EP3571202B1/en active Active
- 2018-01-09 KR KR1020197021451A patent/KR20190097242A/ko not_active Withdrawn
- 2018-01-09 SG SG11201906427QA patent/SG11201906427QA/en unknown
- 2018-01-09 RU RU2019123020A patent/RU2726631C1/ru active
- 2018-01-09 BR BR112019014099-9A patent/BR112019014099A2/pt not_active Application Discontinuation
- 2018-01-09 AU AU2018208848A patent/AU2018208848A1/en not_active Abandoned
- 2018-01-09 JP JP2019538585A patent/JP2020506903A/ja not_active Withdrawn
- 2018-01-09 WO PCT/IB2018/050128 patent/WO2018134698A1/en not_active Ceased
- 2018-01-09 MX MX2019008690A patent/MX2019008690A/es unknown
- 2018-01-09 CA CA3050853A patent/CA3050853A1/en not_active Abandoned
- 2018-01-09 CN CN201880007992.7A patent/CN110198944A/zh active Pending
- 2018-01-18 TW TW107101775A patent/TWI665199B/zh not_active IP Right Cessation
- 2018-01-22 US US15/876,698 patent/US20180208608A1/en not_active Abandoned
-
2019
- 2019-06-03 US US16/429,678 patent/US10858373B2/en active Active
- 2019-07-01 IL IL267781A patent/IL267781A/en unknown
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