JP2019503385A5 - - Google Patents

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JP2019503385A5
JP2019503385A5 JP2018539070A JP2018539070A JP2019503385A5 JP 2019503385 A5 JP2019503385 A5 JP 2019503385A5 JP 2018539070 A JP2018539070 A JP 2018539070A JP 2018539070 A JP2018539070 A JP 2018539070A JP 2019503385 A5 JP2019503385 A5 JP 2019503385A5
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methyl
benzo
imidazole
carboxamide
dioxol
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JP2018539070A
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JP6948333B2 (ja
JP2019503385A (ja
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Priority claimed from PCT/US2017/015220 external-priority patent/WO2017132432A1/en
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Priority to JP2021150729A priority Critical patent/JP2021193131A/ja
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Publication of JP6948333B2 publication Critical patent/JP6948333B2/ja
Expired - Fee Related legal-status Critical Current
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JP2018539070A 2016-01-29 2017-01-27 Ror−ガンマのモジュレータとしてのベンズイミダゾール誘導体 Expired - Fee Related JP6948333B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021150729A JP2021193131A (ja) 2016-01-29 2021-09-16 Ror−ガンマのモジュレータとしてのベンズイミダゾール誘導体

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662288487P 2016-01-29 2016-01-29
US62/288,487 2016-01-29
US201662320893P 2016-04-11 2016-04-11
US62/320,893 2016-04-11
PCT/US2017/015220 WO2017132432A1 (en) 2016-01-29 2017-01-27 Benzimidazole derivatives as modulators of ror-gamma

Related Child Applications (1)

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JP2021150729A Division JP2021193131A (ja) 2016-01-29 2021-09-16 Ror−ガンマのモジュレータとしてのベンズイミダゾール誘導体

Publications (3)

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JP2019503385A JP2019503385A (ja) 2019-02-07
JP2019503385A5 true JP2019503385A5 (OSRAM) 2020-03-05
JP6948333B2 JP6948333B2 (ja) 2021-10-13

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JP2018539070A Expired - Fee Related JP6948333B2 (ja) 2016-01-29 2017-01-27 Ror−ガンマのモジュレータとしてのベンズイミダゾール誘導体
JP2021150729A Pending JP2021193131A (ja) 2016-01-29 2021-09-16 Ror−ガンマのモジュレータとしてのベンズイミダゾール誘導体

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JP2021150729A Pending JP2021193131A (ja) 2016-01-29 2021-09-16 Ror−ガンマのモジュレータとしてのベンズイミダゾール誘導体

Country Status (15)

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US (2) US10829481B2 (OSRAM)
EP (2) EP3408268B8 (OSRAM)
JP (2) JP6948333B2 (OSRAM)
KR (1) KR20180100697A (OSRAM)
CN (2) CN109071509B (OSRAM)
AU (1) AU2017212577B2 (OSRAM)
BR (1) BR112018015273A2 (OSRAM)
CA (1) CA3011838A1 (OSRAM)
MA (2) MA45646A (OSRAM)
MX (1) MX381313B (OSRAM)
RU (2) RU2021133444A (OSRAM)
SA (1) SA518392101B1 (OSRAM)
TW (2) TW202220968A (OSRAM)
UY (1) UY37098A (OSRAM)
WO (1) WO2017132432A1 (OSRAM)

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CN114502535B (zh) * 2019-10-31 2024-04-12 江苏恒瑞医药股份有限公司 一种RORγ调节剂的酸加成盐
CN112745268B (zh) * 2019-10-31 2022-09-16 江苏恒瑞医药股份有限公司 苯并咪唑衍生物的晶型及制备方法
TW202136237A (zh) 2020-01-06 2021-10-01 大陸商廣東東陽光藥業有限公司 RORγt抑制劑及其製備方法和用途
CN111333552B (zh) * 2020-04-09 2021-07-20 广州安岩仁医药科技有限公司 β-苯并氨基酸类化合物的合成方法
CN111606868B (zh) * 2020-06-23 2023-02-17 温州大学新材料与产业技术研究院 一种双齿噁唑啉手性配体的制备方法
CN113912563B (zh) * 2020-07-10 2025-05-27 中国科学院广州生物医药与健康研究院 一种苯并五元氮杂环化合物及其应用
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