JP2018530595A5 - - Google Patents

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Publication number
JP2018530595A5
JP2018530595A5 JP2018519749A JP2018519749A JP2018530595A5 JP 2018530595 A5 JP2018530595 A5 JP 2018530595A5 JP 2018519749 A JP2018519749 A JP 2018519749A JP 2018519749 A JP2018519749 A JP 2018519749A JP 2018530595 A5 JP2018530595 A5 JP 2018530595A5
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JP
Japan
Prior art keywords
trifluoromethyl
ethyl
imidazo
pyrazole
dihydro
Prior art date
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Application number
JP2018519749A
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English (en)
Japanese (ja)
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JP2018530595A (ja
JP6860559B2 (ja
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Priority claimed from PCT/US2016/057135 external-priority patent/WO2017066633A1/en
Publication of JP2018530595A publication Critical patent/JP2018530595A/ja
Publication of JP2018530595A5 publication Critical patent/JP2018530595A5/ja
Priority to JP2021053182A priority Critical patent/JP7090770B2/ja
Application granted granted Critical
Publication of JP6860559B2 publication Critical patent/JP6860559B2/ja
Active legal-status Critical Current
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JP2018519749A 2015-10-16 2016-10-14 Ep4アンタゴニスト Active JP6860559B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021053182A JP7090770B2 (ja) 2015-10-16 2021-03-26 Ep4アンタゴニスト

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201562242734P 2015-10-16 2015-10-16
US201562242748P 2015-10-16 2015-10-16
US62/242,734 2015-10-16
US62/242,748 2015-10-16
BD252/2016 2016-10-13
BD2522016 2016-10-13
PCT/US2016/057135 WO2017066633A1 (en) 2015-10-16 2016-10-14 Ep4 antagonists

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2021053182A Division JP7090770B2 (ja) 2015-10-16 2021-03-26 Ep4アンタゴニスト

Publications (3)

Publication Number Publication Date
JP2018530595A JP2018530595A (ja) 2018-10-18
JP2018530595A5 true JP2018530595A5 (enExample) 2019-11-28
JP6860559B2 JP6860559B2 (ja) 2021-04-14

Family

ID=58518017

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2018519749A Active JP6860559B2 (ja) 2015-10-16 2016-10-14 Ep4アンタゴニスト
JP2021053182A Active JP7090770B2 (ja) 2015-10-16 2021-03-26 Ep4アンタゴニスト

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2021053182A Active JP7090770B2 (ja) 2015-10-16 2021-03-26 Ep4アンタゴニスト

Country Status (11)

Country Link
US (3) US10316040B2 (enExample)
EP (1) EP3362454B1 (enExample)
JP (2) JP6860559B2 (enExample)
KR (1) KR102684436B1 (enExample)
CN (1) CN108473497B (enExample)
AU (1) AU2016338679B2 (enExample)
BR (1) BR112018007664B1 (enExample)
CA (1) CA3002144C (enExample)
IL (1) IL258737A (enExample)
MX (1) MX390051B (enExample)
WO (1) WO2017066633A1 (enExample)

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AU2018268311B2 (en) 2017-05-18 2022-02-10 Idorsia Pharmaceuticals Ltd Pyrimidine derivatives as PGE2 receptor modulators
EP3625224B1 (en) 2017-05-18 2021-08-04 Idorsia Pharmaceuticals Ltd N-substituted indole derivatives
US11325899B2 (en) 2017-05-18 2022-05-10 Idorsia Pharmaceuticals Ltd Benzofurane and benzothiophene derivatives as PGE2 receptor modulators
WO2018210994A1 (en) 2017-05-18 2018-11-22 Idorsia Pharmaceuticals Ltd Phenyl derivatives as pge2 receptor modulators
WO2019149286A1 (en) * 2018-02-05 2019-08-08 Shenzhen Ionova Life Science Co., Ltd. Heterobicyclic carboxylic acids for treating cancer or inflammatory diseases
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JP7488269B2 (ja) 2019-01-22 2024-05-21 キーセラ・(スーチョウ)・ファーマシューティカルズ・カンパニー・リミテッド Pge2/ep4シグナル伝達を阻害する化合物、その製造方法及びその医薬における応用
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