JP2017535555A5 - - Google Patents

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Publication number
JP2017535555A5
JP2017535555A5 JP2017526523A JP2017526523A JP2017535555A5 JP 2017535555 A5 JP2017535555 A5 JP 2017535555A5 JP 2017526523 A JP2017526523 A JP 2017526523A JP 2017526523 A JP2017526523 A JP 2017526523A JP 2017535555 A5 JP2017535555 A5 JP 2017535555A5
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JP
Japan
Prior art keywords
treprostinil
dcm
dmf
dioxane
coupling reagent
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JP2017526523A
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English (en)
Japanese (ja)
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JP2017535555A (ja
JP6866043B2 (ja
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Priority claimed from PCT/US2015/061427 external-priority patent/WO2016081658A1/en
Publication of JP2017535555A publication Critical patent/JP2017535555A/ja
Publication of JP2017535555A5 publication Critical patent/JP2017535555A5/ja
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JP2017526523A 2014-11-18 2015-11-18 トレプロスチニルプロドラッグおよびトレプロスチニル誘導体プロドラッグの製造方法 Active JP6866043B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462081515P 2014-11-18 2014-11-18
US62/081,515 2014-11-18
PCT/US2015/061427 WO2016081658A1 (en) 2014-11-18 2015-11-18 Methods of manufacturing treprostinil and treprostinil derivative prodrugs

Publications (3)

Publication Number Publication Date
JP2017535555A JP2017535555A (ja) 2017-11-30
JP2017535555A5 true JP2017535555A5 (https=) 2018-12-27
JP6866043B2 JP6866043B2 (ja) 2021-04-28

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JP2017526523A Active JP6866043B2 (ja) 2014-11-18 2015-11-18 トレプロスチニルプロドラッグおよびトレプロスチニル誘導体プロドラッグの製造方法

Country Status (7)

Country Link
US (5) US10343979B2 (https=)
EP (2) EP3221291B1 (https=)
JP (1) JP6866043B2 (https=)
AU (1) AU2015349969B2 (https=)
CA (1) CA2967385C (https=)
ES (1) ES2873873T3 (https=)
WO (1) WO2016081658A1 (https=)

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JP6866043B2 (ja) 2014-11-18 2021-04-28 インスメッド インコーポレイテッド トレプロスチニルプロドラッグおよびトレプロスチニル誘導体プロドラッグの製造方法
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JP7455144B2 (ja) 2019-04-29 2024-03-25 インスメッド インコーポレイテッド トレプロスチニルプロドラッグの乾燥粉末組成物およびその使用方法
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JP7455144B2 (ja) 2019-04-29 2024-03-25 インスメッド インコーポレイテッド トレプロスチニルプロドラッグの乾燥粉末組成物およびその使用方法

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