JP2016505071A5 - - Google Patents

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Publication number
JP2016505071A5
JP2016505071A5 JP2015555276A JP2015555276A JP2016505071A5 JP 2016505071 A5 JP2016505071 A5 JP 2016505071A5 JP 2015555276 A JP2015555276 A JP 2015555276A JP 2015555276 A JP2015555276 A JP 2015555276A JP 2016505071 A5 JP2016505071 A5 JP 2016505071A5
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JP
Japan
Prior art keywords
compound
pharmaceutical composition
chlorophenoxy
isoquinoline
cyano
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2015555276A
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English (en)
Japanese (ja)
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JP2016505071A (ja
JP6437456B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2014/012780 external-priority patent/WO2014116849A1/en
Publication of JP2016505071A publication Critical patent/JP2016505071A/ja
Publication of JP2016505071A5 publication Critical patent/JP2016505071A5/ja
Application granted granted Critical
Publication of JP6437456B2 publication Critical patent/JP6437456B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2015555276A 2013-01-24 2014-01-23 {[1−シアノ−5−(4−クロロフェノキシ)−4−ヒドロキシ−イソキノリン−3−カルボニル]−アミノ}−酢酸の結晶形態 Expired - Fee Related JP6437456B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361756361P 2013-01-24 2013-01-24
US61/756,361 2013-01-24
PCT/US2014/012780 WO2014116849A1 (en) 2013-01-24 2014-01-23 Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid

Publications (3)

Publication Number Publication Date
JP2016505071A JP2016505071A (ja) 2016-02-18
JP2016505071A5 true JP2016505071A5 (enExample) 2017-02-23
JP6437456B2 JP6437456B2 (ja) 2018-12-12

Family

ID=50073508

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015555276A Expired - Fee Related JP6437456B2 (ja) 2013-01-24 2014-01-23 {[1−シアノ−5−(4−クロロフェノキシ)−4−ヒドロキシ−イソキノリン−3−カルボニル]−アミノ}−酢酸の結晶形態

Country Status (15)

Country Link
US (1) US9643928B2 (enExample)
EP (1) EP2951159B1 (enExample)
JP (1) JP6437456B2 (enExample)
KR (1) KR102233081B1 (enExample)
CN (1) CN105452227B (enExample)
AU (1) AU2014209319B2 (enExample)
CA (1) CA2899024C (enExample)
DK (1) DK2951159T3 (enExample)
ES (1) ES2694297T3 (enExample)
IL (1) IL240066B (enExample)
MX (1) MX360048B (enExample)
RU (1) RU2666144C2 (enExample)
SG (2) SG11201505748UA (enExample)
TW (1) TWI685487B (enExample)
WO (1) WO2014116849A1 (enExample)

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SG10201700873UA (en) 2012-07-16 2017-04-27 Fibrogen Inc Crystalline forms of the prolyl hydroxylase inhibitor [(4-hydroxy-1-methyl-7-phenoxy-isoquinoline-3-carbonyl)-amino]-acetic acid
CA2879238C (en) 2012-07-16 2021-08-10 Fibrogen, Inc. Process for making isoquinoline compounds
JP6437456B2 (ja) 2013-01-24 2018-12-12 フィブロジェン インコーポレイテッド {[1−シアノ−5−(4−クロロフェノキシ)−4−ヒドロキシ−イソキノリン−3−カルボニル]−アミノ}−酢酸の結晶形態
CN110448537A (zh) 2013-06-06 2019-11-15 菲布罗根有限公司 Hif羟化酶抑制剂的药物制剂
WO2016034108A1 (zh) 2014-09-02 2016-03-10 广东东阳光药业有限公司 喹啉酮类化合物及其应用
EP4121009A4 (en) * 2020-03-17 2024-04-17 Zydus Lifesciences Limited Formulation comprising hif prolyl hydroxylase inhibitors

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