JP2014501740A5 - - Google Patents
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- JP2014501740A5 JP2014501740A5 JP2013544980A JP2013544980A JP2014501740A5 JP 2014501740 A5 JP2014501740 A5 JP 2014501740A5 JP 2013544980 A JP2013544980 A JP 2013544980A JP 2013544980 A JP2013544980 A JP 2013544980A JP 2014501740 A5 JP2014501740 A5 JP 2014501740A5
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- Prior art keywords
- pharmaceutically acceptable
- acceptable salt
- effective amount
- medicament
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201061426773P | 2010-12-23 | 2010-12-23 | |
| US61/426,773 | 2010-12-23 | ||
| CNPCT/CN2011/074569 | 2011-05-24 | ||
| PCT/CN2011/074569 WO2012159262A1 (en) | 2011-05-24 | 2011-05-24 | Selective glycosidase inhibitors and uses thereof |
| US201161507684P | 2011-07-14 | 2011-07-14 | |
| US61/507,684 | 2011-07-14 | ||
| PCT/CA2011/001397 WO2012083435A1 (en) | 2010-12-23 | 2011-12-21 | Selective glycosidase inhibitors and uses thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015230912A Division JP6322177B2 (ja) | 2010-12-23 | 2015-11-26 | 選択的グルコシダーゼインヒビターおよびその使用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2014501740A JP2014501740A (ja) | 2014-01-23 |
| JP2014501740A5 true JP2014501740A5 (https=) | 2015-10-15 |
| JP5861194B2 JP5861194B2 (ja) | 2016-02-16 |
Family
ID=46312954
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013544980A Expired - Fee Related JP5861194B2 (ja) | 2010-12-23 | 2011-12-21 | 選択的グルコシダーゼインヒビターおよびその使用 |
| JP2015230912A Active JP6322177B2 (ja) | 2010-12-23 | 2015-11-26 | 選択的グルコシダーゼインヒビターおよびその使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015230912A Active JP6322177B2 (ja) | 2010-12-23 | 2015-11-26 | 選択的グルコシダーゼインヒビターおよびその使用 |
Country Status (26)
| Country | Link |
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| US (2) | US9243020B2 (https=) |
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| CA2599843C (en) * | 2005-03-01 | 2013-08-27 | Simon Fraser University | Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof |
| AU2007291870B2 (en) | 2006-08-31 | 2012-12-06 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| EP2321289A4 (en) * | 2008-08-01 | 2011-11-16 | Univ Fraser Simon | SELECTIVE GLYCOSIDASE HEMMER AND ITS USE |
| WO2011140640A1 (en) | 2010-05-11 | 2011-11-17 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| US8933040B2 (en) | 2010-11-08 | 2015-01-13 | Craig A. Coburn | Selective glycosidase inhibitors and uses thereof |
| RU2609210C2 (ru) | 2010-12-23 | 2017-01-31 | Алектос Терапьютикс Инк. | Селективные ингибиторы гликозидазы и их применение |
| EP2688899B1 (en) | 2011-03-24 | 2017-02-22 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2691407B1 (en) | 2011-03-31 | 2017-02-22 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| BR112013033098B8 (pt) | 2011-06-27 | 2021-03-23 | Alectos Therapeutics Inc | inibidores de glicosidade seletivos e usos dos mesmos |
| US9701693B2 (en) | 2011-06-27 | 2017-07-11 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2726468B1 (en) | 2011-06-27 | 2017-04-12 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| ES2568603T3 (es) | 2011-08-25 | 2016-05-03 | Merck Patent Gmbh | Pirano[3,2-d][1,3]tiazol como inhibidores de glicosidasas |
| EP2890676B1 (en) | 2012-08-31 | 2018-12-05 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| EP2890675A4 (en) | 2012-08-31 | 2016-01-13 | Alectos Therapeutics Inc | GLYCOSIDASE INHIBITORS AND USES THEREOF |
| KR20150079711A (ko) * | 2012-10-31 | 2015-07-08 | 알렉토스 테라퓨틱스 인크. | 글리코시다아제 저해제 및 이의 용도 |
| WO2014100934A1 (en) * | 2012-12-24 | 2014-07-03 | Merck Sharp & Dohme Corp. | Glycosidase inhibitors and uses thereof |
| KR102043337B1 (ko) | 2014-08-28 | 2019-11-11 | 아셰뉴론 에스아 | 글리코시다제 저해제 |
| KR101777164B1 (ko) | 2015-07-20 | 2017-09-11 | 순천향대학교 산학협력단 | O-GlcNAc 트랜스퍼레즈 억제제용 UDP-GlcNAc의 C1-포스포네이트 유도체 |
| AR106977A1 (es) * | 2015-12-14 | 2018-03-07 | Amicus Therapeutics Inc | Compuestos para el tratamiento de la enfermedad de alzheimer y/o la angiopatía amiloide cerebral |
| AU2017222964B2 (en) | 2016-02-25 | 2020-01-02 | Asceneuron S. A. | Glycosidase inhibitors |
| KR20180132629A (ko) | 2016-02-25 | 2018-12-12 | 아셰뉴론 에스아 | 글리코시다제 저해제 |
| CA3014572C (en) | 2016-02-25 | 2023-10-03 | Asceneuron S.A. | Acid addition salts of piperazine derivatives |
| US11261183B2 (en) | 2016-02-25 | 2022-03-01 | Asceneuron Sa | Sulfoximine glycosidase inhibitors |
| US11213525B2 (en) | 2017-08-24 | 2022-01-04 | Asceneuron Sa | Linear glycosidase inhibitors |
| CN107814773B (zh) * | 2017-11-13 | 2020-05-22 | 西安交通大学 | 含有喹唑啉酮的二芳基脲类化合物及其制备方法和应用 |
| CN112312908A (zh) * | 2018-06-20 | 2021-02-02 | 詹森药业有限公司 | Oga抑制剂化合物 |
| JP7407171B2 (ja) | 2018-08-22 | 2023-12-28 | エースニューロン・ソシエテ・アノニム | グリコシダーゼ阻害剤として有用なピペラジン誘導体のコハク酸付加塩及びフマル酸付加塩 |
| WO2020039027A1 (en) | 2018-08-22 | 2020-02-27 | Asceneuron S. A. | Pyrrolidine glycosidase inhibitors |
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| CN111956656B (zh) * | 2020-08-28 | 2021-10-15 | 河北大学 | Oga抑制剂在制备抗肿瘤药物中的应用 |
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