JP2011529857A5 - - Google Patents

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Publication number
JP2011529857A5
JP2011529857A5 JP2011520296A JP2011520296A JP2011529857A5 JP 2011529857 A5 JP2011529857 A5 JP 2011529857A5 JP 2011520296 A JP2011520296 A JP 2011520296A JP 2011520296 A JP2011520296 A JP 2011520296A JP 2011529857 A5 JP2011529857 A5 JP 2011529857A5
Authority
JP
Japan
Prior art keywords
disease
compound
acceptable salt
pharmaceutically acceptable
glcnacase
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011520296A
Other languages
English (en)
Japanese (ja)
Other versions
JP2011529857A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CA2009/001087 external-priority patent/WO2010012106A1/en
Publication of JP2011529857A publication Critical patent/JP2011529857A/ja
Publication of JP2011529857A5 publication Critical patent/JP2011529857A5/ja
Pending legal-status Critical Current

Links

JP2011520296A 2008-08-01 2009-07-31 選択的グリコシダーゼインヒビターおよびその使用 Pending JP2011529857A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8552708P 2008-08-01 2008-08-01
US61/085,527 2008-08-01
PCT/CA2009/001087 WO2010012106A1 (en) 2008-08-01 2009-07-31 Selective glycosidase inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
JP2011529857A JP2011529857A (ja) 2011-12-15
JP2011529857A5 true JP2011529857A5 (https=) 2012-09-06

Family

ID=41609896

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011520296A Pending JP2011529857A (ja) 2008-08-01 2009-07-31 選択的グリコシダーゼインヒビターおよびその使用

Country Status (6)

Country Link
US (2) US8541441B2 (https=)
EP (1) EP2340250B1 (https=)
JP (1) JP2011529857A (https=)
AU (1) AU2009276222B2 (https=)
CA (1) CA2732335A1 (https=)
WO (1) WO2010012106A1 (https=)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2599843C (en) * 2005-03-01 2013-08-27 Simon Fraser University Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof
AU2007291870B2 (en) 2006-08-31 2012-12-06 Simon Fraser University Selective glycosidase inhibitors and uses thereof
EP2321289A4 (en) * 2008-08-01 2011-11-16 Univ Fraser Simon SELECTIVE GLYCOSIDASE HEMMER AND ITS USE
WO2011140640A1 (en) 2010-05-11 2011-11-17 Simon Fraser University Selective glycosidase inhibitors and uses thereof
US8901087B2 (en) 2010-11-08 2014-12-02 Merck Sharp & Dohme Corp. Selective glycosidase inhibitors and uses thereof
US8933040B2 (en) 2010-11-08 2015-01-13 Craig A. Coburn Selective glycosidase inhibitors and uses thereof
TW201249848A (en) 2010-11-08 2012-12-16 Merck Sharp & Dohme Selective glycosidase inhibitors and uses thereof
RU2609210C2 (ru) 2010-12-23 2017-01-31 Алектос Терапьютикс Инк. Селективные ингибиторы гликозидазы и их применение
EP2688899B1 (en) 2011-03-24 2017-02-22 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
EP2691407B1 (en) 2011-03-31 2017-02-22 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
EP2726468B1 (en) 2011-06-27 2017-04-12 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
BR112013033098B8 (pt) 2011-06-27 2021-03-23 Alectos Therapeutics Inc inibidores de glicosidade seletivos e usos dos mesmos
US9701693B2 (en) 2011-06-27 2017-07-11 Alectos Therapeutics Inc. Selective glycosidase inhibitors and uses thereof
EP2788017B1 (en) 2011-12-05 2017-05-31 Ben-Gurion University of The Negev Research and Development Authority INHIBITORS OF IgG-A2BG2 FOR USE IN TREATING AND DIAGNOSING AMYOTROPHIC LATERAL SCLEROSIS
EP2847199B1 (en) 2012-05-08 2017-10-25 Merck Sharp & Dohme Corp. Permeable glycosidase inhibitors and uses thereof
EP2890676B1 (en) 2012-08-31 2018-12-05 Alectos Therapeutics Inc. Glycosidase inhibitors and uses thereof
EP2890675A4 (en) 2012-08-31 2016-01-13 Alectos Therapeutics Inc GLYCOSIDASE INHIBITORS AND USES THEREOF
KR20150079711A (ko) 2012-10-31 2015-07-08 알렉토스 테라퓨틱스 인크. 글리코시다아제 저해제 및 이의 용도
WO2024083820A1 (en) 2022-10-18 2024-04-25 Institut National de la Santé et de la Recherche Médicale Method and composition for determining the level of o-glcnacylation in horses

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1991000018A1 (en) 1989-06-26 1991-01-10 Fluid Dynamics Pty Limited Controlled atmosphere generating equipment
US5079254A (en) * 1990-06-04 1992-01-07 Merrell Dow Pharmaceuticals Inc. Derivatives of 6-aminooctahydroindolizinetriol
WO2006016904A2 (en) 2004-04-14 2006-02-16 Uab Research Foundation Activators of hexosamine biosynthesis as inhibitors of injury induced by ischemia or hemorrhagic shock
CA2599843C (en) 2005-03-01 2013-08-27 Simon Fraser University Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof
AU2007291870B2 (en) 2006-08-31 2012-12-06 Simon Fraser University Selective glycosidase inhibitors and uses thereof

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