JP2014524911A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2014524911A5 JP2014524911A5 JP2014517357A JP2014517357A JP2014524911A5 JP 2014524911 A5 JP2014524911 A5 JP 2014524911A5 JP 2014517357 A JP2014517357 A JP 2014517357A JP 2014517357 A JP2014517357 A JP 2014517357A JP 2014524911 A5 JP2014524911 A5 JP 2014524911A5
- Authority
- JP
- Japan
- Prior art keywords
- fluoro
- pyrano
- tetrahydro
- thiazol
- hydroxyethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161501377P | 2011-06-27 | 2011-06-27 | |
| US61/501,377 | 2011-06-27 | ||
| PCT/CA2012/050433 WO2013000084A1 (en) | 2011-06-27 | 2012-06-27 | Selective glycosidase inhibitors and uses thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2014524911A JP2014524911A (ja) | 2014-09-25 |
| JP2014524911A5 true JP2014524911A5 (https=) | 2015-08-13 |
| JP6147737B2 JP6147737B2 (ja) | 2017-06-14 |
Family
ID=47423333
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014517357A Expired - Fee Related JP6147737B2 (ja) | 2011-06-27 | 2012-06-27 | 選択的グリコシダーゼ阻害剤およびその使用 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US9409924B2 (https=) |
| EP (1) | EP2723753B1 (https=) |
| JP (1) | JP6147737B2 (https=) |
| KR (1) | KR102054744B1 (https=) |
| CN (1) | CN103889996B (https=) |
| AU (1) | AU2012276257B2 (https=) |
| BR (1) | BR112013033098B8 (https=) |
| CA (1) | CA2840013C (https=) |
| MX (1) | MX364602B (https=) |
| RU (1) | RU2625308C2 (https=) |
| WO (1) | WO2013000084A1 (https=) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2007291870B2 (en) | 2006-08-31 | 2012-12-06 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| EP2321289A4 (en) | 2008-08-01 | 2011-11-16 | Univ Fraser Simon | SELECTIVE GLYCOSIDASE HEMMER AND ITS USE |
| WO2011140640A1 (en) | 2010-05-11 | 2011-11-17 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| US8933040B2 (en) | 2010-11-08 | 2015-01-13 | Craig A. Coburn | Selective glycosidase inhibitors and uses thereof |
| RU2609210C2 (ru) | 2010-12-23 | 2017-01-31 | Алектос Терапьютикс Инк. | Селективные ингибиторы гликозидазы и их применение |
| EP2688899B1 (en) | 2011-03-24 | 2017-02-22 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2691407B1 (en) | 2011-03-31 | 2017-02-22 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9701693B2 (en) | 2011-06-27 | 2017-07-11 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2726468B1 (en) | 2011-06-27 | 2017-04-12 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| BR112013033098B8 (pt) | 2011-06-27 | 2021-03-23 | Alectos Therapeutics Inc | inibidores de glicosidade seletivos e usos dos mesmos |
| EP2890676B1 (en) | 2012-08-31 | 2018-12-05 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| EP2890675A4 (en) | 2012-08-31 | 2016-01-13 | Alectos Therapeutics Inc | GLYCOSIDASE INHIBITORS AND USES THEREOF |
| KR20150079711A (ko) | 2012-10-31 | 2015-07-08 | 알렉토스 테라퓨틱스 인크. | 글리코시다아제 저해제 및 이의 용도 |
| WO2014100934A1 (en) | 2012-12-24 | 2014-07-03 | Merck Sharp & Dohme Corp. | Glycosidase inhibitors and uses thereof |
| SG11201510177WA (en) | 2013-06-11 | 2016-01-28 | Harvard College | SC-β CELLS AND COMPOSITIONS AND METHODS FOR GENERATING THE SAME |
| AR106977A1 (es) * | 2015-12-14 | 2018-03-07 | Amicus Therapeutics Inc | Compuestos para el tratamiento de la enfermedad de alzheimer y/o la angiopatía amiloide cerebral |
| US10800784B2 (en) * | 2018-02-01 | 2020-10-13 | Japan Tobacco Inc. | Nitrogen-containing heterocyclic amide compound and pharmaceutical use thereof |
| GB201907716D0 (en) | 2019-05-31 | 2019-07-17 | Smith & Nephew | Systems and methods for extending operational time of negative pressure wound treatment apparatuses |
| GB202000274D0 (en) | 2020-01-09 | 2020-02-26 | Smith & Nephew | Systems and methods for monitoring operational lifetime of negative pressure wound treatment apparatuses |
| WO2022073762A1 (en) | 2020-10-05 | 2022-04-14 | T.J.Smith And Nephew,Limited | Temperature monitoring and control for negative pressure wound therapy systems |
| GB202104922D0 (en) | 2021-04-07 | 2021-05-19 | Smith & Nephew | Temperature monitoring and control for negative pressure wound therapy systems |
| KR102533471B1 (ko) | 2020-11-23 | 2023-05-19 | (주) 메디프론디비티 | O-GlcNAcase 저해 활성을 갖는 화합물 및 이의 용도 |
| GB202109154D0 (en) | 2021-06-25 | 2021-08-11 | Smith & Nephew | Liquid ingress protection for negative pressure wound therapy systems |
| US20240285847A1 (en) | 2021-06-25 | 2024-08-29 | T.J.Smith And Nephew,Limited | Liquid ingress protection and design of electronic circuitry for negative pressure wound therapy systems |
| GB202110240D0 (en) | 2021-07-16 | 2021-09-01 | Smith & Nephew | Reduced pressure apparatuses and methods |
| US20250050008A1 (en) | 2022-01-10 | 2025-02-13 | T.J.Smith And Nephew,Limited | Temperature detection and protection for negative pressure wound therapy systems |
| WO2023135177A1 (en) | 2022-01-14 | 2023-07-20 | T.J.Smith And Nephew, Limited | Self-calibration with dynamic therapy performance for negative pressure wound therapy devices |
| GB202304922D0 (en) | 2023-04-03 | 2023-05-17 | Smith & Nephew | Printed circuit board configurations for negative pressure wound therapy devices |
Family Cites Families (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU1441749A1 (ru) * | 1987-03-16 | 1996-01-10 | Институт Тонкой Органической Химии Им.А.Л.Мнджояна | 2-АМИНО-5,5-ДИМЕТИЛ-4,5-ДИГИДРО-7Н-ПИРАНО [4,3-d] ТИАЗОЛ, ОБЛАДАЮЩИЙ ТРАНКВИЛИЗИРУЮЩЕЙ АКТИВНОСТЬЮ |
| JPH01180894A (ja) | 1988-01-07 | 1989-07-18 | Wako Pure Chem Ind Ltd | アミノ糖誘導体の新規な製造法 |
| JPH07316178A (ja) | 1994-05-25 | 1995-12-05 | Sankyo Co Ltd | 糖アミノオキサゾリン類 |
| JPH09132585A (ja) | 1995-11-10 | 1997-05-20 | Shin Etsu Chem Co Ltd | 新規アミノ糖及びキトオリゴ糖又はその類似オリゴ糖の製造方法 |
| JP4233262B2 (ja) | 2001-03-14 | 2009-03-04 | 生化学工業株式会社 | カルバ糖アミン誘導体及びそれを用いるグリコシダーゼ阻害剤 |
| JP4866515B2 (ja) | 2001-07-02 | 2012-02-01 | 生化学工業株式会社 | 糖オキサゾリン誘導体の製造方法 |
| WO2006016904A2 (en) | 2004-04-14 | 2006-02-16 | Uab Research Foundation | Activators of hexosamine biosynthesis as inhibitors of injury induced by ischemia or hemorrhagic shock |
| CA2599843C (en) | 2005-03-01 | 2013-08-27 | Simon Fraser University | Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof |
| CN107253970A (zh) | 2006-08-31 | 2017-10-17 | 西蒙·弗雷瑟大学 | 选择性糖苷酶抑制剂及其用途 |
| AU2007291870B2 (en) | 2006-08-31 | 2012-12-06 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| CA2732335A1 (en) | 2008-08-01 | 2010-02-04 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| EP2321289A4 (en) | 2008-08-01 | 2011-11-16 | Univ Fraser Simon | SELECTIVE GLYCOSIDASE HEMMER AND ITS USE |
| CA2737267A1 (en) | 2008-09-16 | 2010-04-08 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| WO2011140640A1 (en) | 2010-05-11 | 2011-11-17 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| WO2012061971A1 (en) | 2010-11-08 | 2012-05-18 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| TW201249848A (en) | 2010-11-08 | 2012-12-16 | Merck Sharp & Dohme | Selective glycosidase inhibitors and uses thereof |
| US8933040B2 (en) | 2010-11-08 | 2015-01-13 | Craig A. Coburn | Selective glycosidase inhibitors and uses thereof |
| WO2012061972A1 (en) | 2010-11-08 | 2012-05-18 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| RU2609210C2 (ru) * | 2010-12-23 | 2017-01-31 | Алектос Терапьютикс Инк. | Селективные ингибиторы гликозидазы и их применение |
| GB201103526D0 (en) | 2011-03-02 | 2011-04-13 | Summit Corp Plc | Selective glycosidase inhibitors and uses thereof |
| EP2688899B1 (en) | 2011-03-24 | 2017-02-22 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2691407B1 (en) | 2011-03-31 | 2017-02-22 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| WO2012129802A1 (en) | 2011-03-31 | 2012-10-04 | Alectos Therapeutics Inc. | Pyrano[3,2-d]thiazol derivatives and uses as selective glycosidase inhibitors thereof |
| EP2726468B1 (en) | 2011-06-27 | 2017-04-12 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9701693B2 (en) | 2011-06-27 | 2017-07-11 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| BR112013033098B8 (pt) | 2011-06-27 | 2021-03-23 | Alectos Therapeutics Inc | inibidores de glicosidade seletivos e usos dos mesmos |
| US9126957B2 (en) | 2011-08-18 | 2015-09-08 | Merck Sharp & Dohme Corp. | Selective glycosidase inhibitors and uses thereof |
| ES2568603T3 (es) | 2011-08-25 | 2016-05-03 | Merck Patent Gmbh | Pirano[3,2-d][1,3]tiazol como inhibidores de glicosidasas |
| EP2847199B1 (en) | 2012-05-08 | 2017-10-25 | Merck Sharp & Dohme Corp. | Permeable glycosidase inhibitors and uses thereof |
| EP2890679A4 (en) | 2012-08-31 | 2016-05-04 | Alectos Therapeutics Inc | GLYCOSIDASE INHIBITORS AND USES THEREOF |
| EP2890676B1 (en) | 2012-08-31 | 2018-12-05 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| US9522883B2 (en) | 2012-08-31 | 2016-12-20 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| EP2890675A4 (en) | 2012-08-31 | 2016-01-13 | Alectos Therapeutics Inc | GLYCOSIDASE INHIBITORS AND USES THEREOF |
| KR20150079711A (ko) | 2012-10-31 | 2015-07-08 | 알렉토스 테라퓨틱스 인크. | 글리코시다아제 저해제 및 이의 용도 |
| WO2014100934A1 (en) | 2012-12-24 | 2014-07-03 | Merck Sharp & Dohme Corp. | Glycosidase inhibitors and uses thereof |
-
2012
- 2012-06-27 BR BR112013033098A patent/BR112013033098B8/pt not_active IP Right Cessation
- 2012-06-27 US US14/129,177 patent/US9409924B2/en active Active
- 2012-06-27 RU RU2014102232A patent/RU2625308C2/ru active
- 2012-06-27 KR KR1020147001472A patent/KR102054744B1/ko not_active Expired - Fee Related
- 2012-06-27 WO PCT/CA2012/050433 patent/WO2013000084A1/en not_active Ceased
- 2012-06-27 CN CN201280040350.XA patent/CN103889996B/zh not_active Expired - Fee Related
- 2012-06-27 EP EP12804294.2A patent/EP2723753B1/en active Active
- 2012-06-27 CA CA2840013A patent/CA2840013C/en active Active
- 2012-06-27 MX MX2014000258A patent/MX364602B/es active IP Right Grant
- 2012-06-27 AU AU2012276257A patent/AU2012276257B2/en not_active Ceased
- 2012-06-27 JP JP2014517357A patent/JP6147737B2/ja not_active Expired - Fee Related
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2014524911A5 (https=) | ||
| JP2014501740A5 (https=) | ||
| JP2015534991A5 (https=) | ||
| RU2014102232A (ru) | Селективные ингибиторы гликозидазы и их применение | |
| JP2010501598A5 (https=) | ||
| RU2013134345A (ru) | Селективные ингибиторы гликозидазы и их применение | |
| JP2012502884A5 (https=) | ||
| JP2013541596A5 (https=) | ||
| WO2008025170B1 (en) | Selective glycosidase inhibitors and uses thereof | |
| RU2015120556A (ru) | Ингибиторы гликозидаз и их применения | |
| CN110291080B (zh) | 布鲁顿酪氨酸激酶的咪唑并吡嗪抑制剂 | |
| US6653313B2 (en) | 1,4-dihydropyridine compounds as bradykinin antagonists | |
| KR101749778B1 (ko) | 칸나비노이드 수용체 조절제 | |
| JP6218260B2 (ja) | Ｊａｋ阻害剤としてのアミノピリミジニル化合物 | |
| JP2011529858A5 (https=) | ||
| JP6214643B2 (ja) | ピリミジニルチロシンキナーゼ阻害剤 | |
| RU2757218C2 (ru) | Аминопиразолы в качестве селективных ингибиторов янус-киназы | |
| JP2011529857A5 (https=) | ||
| Zhi et al. | Hybrid antibacterials. DNA polymerase− topoisomerase inhibitors | |
| JP2014531449A (ja) | キナーゼ阻害剤としてのピラゾロ［４，３―ｃ］ピリジン誘導体 | |
| RU2013126531A (ru) | Селективные ингибиторы гликозидазы и их применение | |
| TW200948364A (en) | Thiophenyl-substituted 2-imino-3-methyl pyrrolo pyrimidinone compounds as BACE-1 inhibitors, compositions, and their use | |
| JP2014503527A5 (https=) | ||
| EA200970852A1 (ru) | Производные пиразоло[3,4-в]пиридина в качестве ингибиторов фосфодиэстеразы | |
| CA2545092A1 (en) | Quinolonecarboxylic acid compounds having 5-ht4 receptor agonistic activity |