JP2013540749A5 - - Google Patents

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Publication number
JP2013540749A5
JP2013540749A5 JP2013529373A JP2013529373A JP2013540749A5 JP 2013540749 A5 JP2013540749 A5 JP 2013540749A5 JP 2013529373 A JP2013529373 A JP 2013529373A JP 2013529373 A JP2013529373 A JP 2013529373A JP 2013540749 A5 JP2013540749 A5 JP 2013540749A5
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JP
Japan
Prior art keywords
skin
pain
diseases
disease
expansion
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JP2013529373A
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English (en)
Japanese (ja)
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JP6073229B2 (ja
JP2013540749A (ja
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Priority claimed from PCT/US2011/052004 external-priority patent/WO2012037499A1/en
Publication of JP2013540749A publication Critical patent/JP2013540749A/ja
Publication of JP2013540749A5 publication Critical patent/JP2013540749A5/ja
Application granted granted Critical
Publication of JP6073229B2 publication Critical patent/JP6073229B2/ja
Active legal-status Critical Current
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JP2013529373A 2010-09-16 2011-09-16 [3−(1−(1h−イミダゾール−4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ Active JP6073229B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38337010P 2010-09-16 2010-09-16
US61/383,370 2010-09-16
PCT/US2011/052004 WO2012037499A1 (en) 2010-09-16 2011-09-16 Ester pro-drugs of [3-(1-(1h-imidazol-4-yl)ethyl)-2-methylphenyl] methanol

Publications (3)

Publication Number Publication Date
JP2013540749A JP2013540749A (ja) 2013-11-07
JP2013540749A5 true JP2013540749A5 (https=) 2016-02-04
JP6073229B2 JP6073229B2 (ja) 2017-02-01

Family

ID=44675870

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2013529360A Withdrawn JP2013541527A (ja) 2010-09-16 2011-09-16 網膜疾患を治療するための[3−(1−(1h−イミダゾール4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ
JP2013529372A Active JP6045495B2 (ja) 2010-09-16 2011-09-16 眼圧を低下させるための[3−(1−(1h−イミダゾール−4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ
JP2013529373A Active JP6073229B2 (ja) 2010-09-16 2011-09-16 [3−(1−(1h−イミダゾール−4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ
JP2013529371A Withdrawn JP2013537236A (ja) 2010-09-16 2011-09-16 皮膚疾患及び状態を治療するための[3−(1−(1h−イミダゾール4−イル)エチル−2−メチルフェニル]メタノールのエステル・プロドラッグ

Family Applications Before (2)

Application Number Title Priority Date Filing Date
JP2013529360A Withdrawn JP2013541527A (ja) 2010-09-16 2011-09-16 網膜疾患を治療するための[3−(1−(1h−イミダゾール4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ
JP2013529372A Active JP6045495B2 (ja) 2010-09-16 2011-09-16 眼圧を低下させるための[3−(1−(1h−イミダゾール−4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2013529371A Withdrawn JP2013537236A (ja) 2010-09-16 2011-09-16 皮膚疾患及び状態を治療するための[3−(1−(1h−イミダゾール4−イル)エチル−2−メチルフェニル]メタノールのエステル・プロドラッグ

Country Status (28)

Country Link
US (9) US8492557B2 (https=)
EP (13) EP3050564B1 (https=)
JP (4) JP2013541527A (https=)
KR (7) KR101952457B1 (https=)
CN (5) CN103209694A (https=)
AR (4) AR083018A1 (https=)
AU (4) AU2011301932C1 (https=)
BR (4) BR112013006362A2 (https=)
CA (8) CA2812191C (https=)
CL (4) CL2013000735A1 (https=)
CY (3) CY1121024T1 (https=)
DK (9) DK2616068T3 (https=)
ES (10) ES2607084T3 (https=)
HU (5) HUE047476T2 (https=)
IL (4) IL225280A0 (https=)
MX (4) MX2013003004A (https=)
MY (4) MY161607A (https=)
NZ (1) NZ608751A (https=)
PL (7) PL3348264T3 (https=)
PT (7) PT2616069T (https=)
RU (4) RU2013116405A (https=)
SG (4) SG188571A1 (https=)
SI (5) SI3348264T1 (https=)
TR (1) TR201909249T4 (https=)
TW (4) TW201240661A (https=)
UA (1) UA112973C2 (https=)
WO (4) WO2012037453A1 (https=)
ZA (4) ZA201302193B (https=)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3241553B1 (en) * 2009-02-13 2019-04-10 Allergan, Inc. Pharmaceutical compositions comprising (3-(1-(1h-imidazol-4-yl)ethyl)-2-methylphenyl)methanol
MX344303B (es) 2010-01-11 2016-12-13 Orexigen Therapeutics Inc Metodos para proveer terapia de perdida de peso en pacientes con depresion mayor.
US8492557B2 (en) * 2010-09-16 2013-07-23 Allergan, Inc. Ester pro-drugs of [3-(1-(1H-imidazol-4-yl)ethyl)-2-methylphenyl] methanol
CA2842866A1 (en) * 2011-07-22 2013-01-31 Allergan, Inc. Alpha-2 adrenergic modulators for treating visual disorders mediated by central visual projections from the eye
EP2782569A1 (en) 2011-11-21 2014-10-01 Allergan, Inc. Pharmaceutical compositions comprising 4-[1-(2,3-dimethylphenyl)ethyl]-3h-imidazole derivatives for treating retinal diseases
USD794650S1 (en) 2014-11-28 2017-08-15 Samsung Electronics Co., Ltd. Display screen or portion thereof with a graphical user interface
CN108310442B (zh) * 2017-01-17 2021-08-27 台北科技大学 眼科用组合物
KR102050506B1 (ko) 2017-06-20 2019-11-29 한국식품연구원 망막 질환 예방, 개선, 완화 또는 치료용 조성물
CN108872431B (zh) * 2018-07-09 2021-03-23 成都倍特药业股份有限公司 一种检测4-(1-(2,5-二甲基苯基)乙基)-1h-咪唑或/和其盐酸盐的方法
JP7584802B2 (ja) * 2018-08-24 2024-11-18 アドライ・ノーティ・バイオファーマ・カンパニー・リミテッド 高活性stingタンパク質アゴニスト
WO2022221071A1 (en) * 2021-04-16 2022-10-20 Ads Therapeutics Llc Alpha2 adrenergic agonist codrugs conjugated with muscarinic agonist drugs
AU2024217271A1 (en) * 2023-02-08 2025-09-18 Bausch + Lomb Ireland Limited Alpha-2-adrenergic agonists for improving vision
WO2025179071A1 (en) * 2024-02-20 2025-08-28 Bausch + Lomb Ireland Limited Sustained-release drug delivery compositions for treating ocular diseases

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DE69307505T2 (de) 1992-05-13 1997-07-24 Sandoz-Patent-Gmbh, 79539 Loerrach Opthalmische zusammensetzungen enthaltend ein cyclosporin
US5459133A (en) * 1992-06-05 1995-10-17 Telor Ophthalmic Pharmaceuticals, Inc. Methods and products for treating presbyopia
ATE234290T1 (de) 1993-11-15 2003-03-15 Schering Corp Phenylalkyl-imidazole als h3-rezeptor- antagonisten
US5474979A (en) 1994-05-17 1995-12-12 Allergan, Inc. Nonirritating emulsions for sensitive tissue
EP0957073A1 (en) * 1998-05-12 1999-11-17 Schwarz Pharma Ag Novel derivatives of 3,3-diphenylpropylamines
US20040214829A1 (en) * 2000-07-14 2004-10-28 Allergan, Inc. Compositions containing alpha-2-adrenergic agonist components
US20020198209A1 (en) 2001-05-03 2002-12-26 Allergan Sales Inc. Compositions having enhanced pharmacokinetic characteristics
MXPA05012679A (es) * 2003-05-27 2006-02-08 Sod Conseils Rech Applic Nuevos derivados de imidazoles, su preparacion y su uso como medicamento.
US7439241B2 (en) * 2003-05-27 2008-10-21 Galderma Laboratories, Inc. Compounds, formulations, and methods for treating or preventing rosacea
US20060209374A1 (en) * 2003-07-14 2006-09-21 Koninklijke Philips Electronics N.V. Projection device
MXPA06002716A (es) * 2003-09-12 2006-06-06 Allergan Inc Metodos y composiciones para el tratamiento de dolor y otras condiciones mediadas por adrenergicos de alfa-2.
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JP4955543B2 (ja) 2004-05-25 2012-06-20 サンズローザ ファーマシューティカル ディヴェロップメント インコーポレイテッド 炎症性皮膚疾患を治療又は予防するための化合物、製剤及び方法
US20050277584A1 (en) 2004-06-09 2005-12-15 Allergan, Inc. Pharmaceutical compositions comprising cyclosporins
NZ553341A (en) 2004-09-24 2010-11-26 Allergan Inc 4-(phenylmethyl and substituted phenylmethyl)-imidazole-2-thiones acting as specific alpha2 adrenergic agonists
US7931909B2 (en) 2005-05-10 2011-04-26 Allergan, Inc. Ocular therapy using alpha-2 adrenergic receptor compounds having enhanced anterior clearance rates
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US7902247B2 (en) 2008-01-09 2011-03-08 Allergan, Inc. Substituted-aryl-2-phenylethyl-1H-imidazole compounds as subtype selective modulators of alpha 2B and/or alpha 2C adrenergic receptors
JP2012517433A (ja) 2009-02-06 2012-08-02 アラーガン インコーポレイテッド アルファ2bおよび/またはアルファ2cアドレナリンレセプターのサブタイプ選択的モジュレーターとしてのピリジン化合物
EP3241553B1 (en) * 2009-02-13 2019-04-10 Allergan, Inc. Pharmaceutical compositions comprising (3-(1-(1h-imidazol-4-yl)ethyl)-2-methylphenyl)methanol
US8394800B2 (en) * 2009-11-19 2013-03-12 Galderma Laboratories, L.P. Method for treating psoriasis
US8492557B2 (en) * 2010-09-16 2013-07-23 Allergan, Inc. Ester pro-drugs of [3-(1-(1H-imidazol-4-yl)ethyl)-2-methylphenyl] methanol

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