JP2013540749A5 - - Google Patents

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Publication number
JP2013540749A5
JP2013540749A5 JP2013529373A JP2013529373A JP2013540749A5 JP 2013540749 A5 JP2013540749 A5 JP 2013540749A5 JP 2013529373 A JP2013529373 A JP 2013529373A JP 2013529373 A JP2013529373 A JP 2013529373A JP 2013540749 A5 JP2013540749 A5 JP 2013540749A5
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JP
Japan
Prior art keywords
skin
pain
diseases
disease
expansion
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JP2013529373A
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English (en)
Japanese (ja)
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JP6073229B2 (ja
JP2013540749A (ja
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Priority claimed from PCT/US2011/052004 external-priority patent/WO2012037499A1/en
Publication of JP2013540749A publication Critical patent/JP2013540749A/ja
Publication of JP2013540749A5 publication Critical patent/JP2013540749A5/ja
Application granted granted Critical
Publication of JP6073229B2 publication Critical patent/JP6073229B2/ja
Active legal-status Critical Current
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JP2013529373A 2010-09-16 2011-09-16 [3−(1−(1h−イミダゾール−4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ Active JP6073229B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38337010P 2010-09-16 2010-09-16
US61/383,370 2010-09-16
PCT/US2011/052004 WO2012037499A1 (en) 2010-09-16 2011-09-16 Ester pro-drugs of [3-(1-(1h-imidazol-4-yl)ethyl)-2-methylphenyl] methanol

Publications (3)

Publication Number Publication Date
JP2013540749A JP2013540749A (ja) 2013-11-07
JP2013540749A5 true JP2013540749A5 (https=) 2016-02-04
JP6073229B2 JP6073229B2 (ja) 2017-02-01

Family

ID=44675870

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2013529373A Active JP6073229B2 (ja) 2010-09-16 2011-09-16 [3−(1−(1h−イミダゾール−4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ
JP2013529371A Withdrawn JP2013537236A (ja) 2010-09-16 2011-09-16 皮膚疾患及び状態を治療するための[3−(1−(1h−イミダゾール4−イル)エチル−2−メチルフェニル]メタノールのエステル・プロドラッグ
JP2013529372A Active JP6045495B2 (ja) 2010-09-16 2011-09-16 眼圧を低下させるための[3−(1−(1h−イミダゾール−4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ
JP2013529360A Withdrawn JP2013541527A (ja) 2010-09-16 2011-09-16 網膜疾患を治療するための[3−(1−(1h−イミダゾール4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ

Family Applications After (3)

Application Number Title Priority Date Filing Date
JP2013529371A Withdrawn JP2013537236A (ja) 2010-09-16 2011-09-16 皮膚疾患及び状態を治療するための[3−(1−(1h−イミダゾール4−イル)エチル−2−メチルフェニル]メタノールのエステル・プロドラッグ
JP2013529372A Active JP6045495B2 (ja) 2010-09-16 2011-09-16 眼圧を低下させるための[3−(1−(1h−イミダゾール−4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ
JP2013529360A Withdrawn JP2013541527A (ja) 2010-09-16 2011-09-16 網膜疾患を治療するための[3−(1−(1h−イミダゾール4−イル)エチル)−2−メチルフェニル]メタノールのエステル・プロドラッグ

Country Status (28)

Country Link
US (9) US8653123B2 (https=)
EP (13) EP2616069B1 (https=)
JP (4) JP6073229B2 (https=)
KR (7) KR101840500B1 (https=)
CN (5) CN103221045A (https=)
AR (4) AR083017A1 (https=)
AU (4) AU2011301932C1 (https=)
BR (4) BR112013006362A2 (https=)
CA (8) CA3122745A1 (https=)
CL (4) CL2013000735A1 (https=)
CY (3) CY1121024T1 (https=)
DK (9) DK3050564T3 (https=)
ES (10) ES2684055T3 (https=)
HU (5) HUE039090T2 (https=)
IL (4) IL225280A0 (https=)
MX (4) MX2013003004A (https=)
MY (4) MY173846A (https=)
NZ (1) NZ608751A (https=)
PL (7) PL3050563T3 (https=)
PT (7) PT3053576T (https=)
RU (4) RU2013116405A (https=)
SG (4) SG188573A1 (https=)
SI (5) SI3338777T1 (https=)
TR (1) TR201909249T4 (https=)
TW (4) TW201240662A (https=)
UA (1) UA112973C2 (https=)
WO (4) WO2012037490A1 (https=)
ZA (4) ZA201302194B (https=)

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ES2733905T3 (es) * 2009-02-13 2019-12-03 Allergan Inc Composiciones farmacéuticas que comprenden (3-(1-(1H-imidazol-4-il)etil)-2-metilfenil)metanol
ES2762113T3 (es) 2010-01-11 2020-05-22 Nalpropion Pharmaceuticals Inc Métodos de proporcionar terapia de pérdida de peso en pacientes con depresión mayor
US8653123B2 (en) * 2010-09-16 2014-02-18 Allergan, Inc. Ester pro-drugs of [3-(1-(1H-imidazol-4-yl)ethyl)-2-methylphenyl] methanol for treating retinal diseases
JP2014521643A (ja) * 2011-07-22 2014-08-28 アラーガン インコーポレイテッド 眼の中枢視覚投影によって媒介される視覚障害を治療するためのα−2アドレナリン調節剤
AU2012340806B2 (en) 2011-11-21 2017-10-19 Allergan, Inc. Pharmaceutical compositions comprising 4-[1-(2,3-dimethylphenyl)ethyl]-3H-imidazole derivatives for treating retinal diseases
USD794650S1 (en) 2014-11-28 2017-08-15 Samsung Electronics Co., Ltd. Display screen or portion thereof with a graphical user interface
CN108310442B (zh) * 2017-01-17 2021-08-27 台北科技大学 眼科用组合物
KR102050506B1 (ko) 2017-06-20 2019-11-29 한국식품연구원 망막 질환 예방, 개선, 완화 또는 치료용 조성물
CN108872431B (zh) * 2018-07-09 2021-03-23 成都倍特药业股份有限公司 一种检测4-(1-(2,5-二甲基苯基)乙基)-1h-咪唑或/和其盐酸盐的方法
AU2019326633B2 (en) * 2018-08-24 2022-09-08 Adlai Nortye Biopharma Co., Ltd. High activity sting protein agonist
JP2024514870A (ja) * 2021-04-16 2024-04-03 エーディーエス・セラピューティクス・エルエルシー ムスカリン作動薬が結合したα2アドレナリン作動薬コドラッグ
AU2024217271A1 (en) * 2023-02-08 2025-09-18 Bausch + Lomb Ireland Limited Alpha-2-adrenergic agonists for improving vision
WO2025179071A1 (en) * 2024-02-20 2025-08-28 Bausch + Lomb Ireland Limited Sustained-release drug delivery compositions for treating ocular diseases

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HK1004520A1 (en) 1992-05-13 1998-11-27 Novartis Ag Ophthalmic compositions containing a cyclosporin
US5459133A (en) * 1992-06-05 1995-10-17 Telor Ophthalmic Pharmaceuticals, Inc. Methods and products for treating presbyopia
JPH09505298A (ja) 1993-11-15 1997-05-27 シェーリング コーポレイション H▲下3▼‐レセプターアンタゴニストとしてのフェニル‐アルキルイミダゾール
US5474979A (en) 1994-05-17 1995-12-12 Allergan, Inc. Nonirritating emulsions for sensitive tissue
EP0957073A1 (en) * 1998-05-12 1999-11-17 Schwarz Pharma Ag Novel derivatives of 3,3-diphenylpropylamines
US20040214829A1 (en) * 2000-07-14 2004-10-28 Allergan, Inc. Compositions containing alpha-2-adrenergic agonist components
US20020198209A1 (en) 2001-05-03 2002-12-26 Allergan Sales Inc. Compositions having enhanced pharmacokinetic characteristics
MXPA05012679A (es) * 2003-05-27 2006-02-08 Sod Conseils Rech Applic Nuevos derivados de imidazoles, su preparacion y su uso como medicamento.
US7439241B2 (en) * 2003-05-27 2008-10-21 Galderma Laboratories, Inc. Compounds, formulations, and methods for treating or preventing rosacea
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WO2005034998A2 (en) 2003-09-12 2005-04-21 Allergan, Inc. Methods and compositions for the treatment of pain and other alpha 2 adrenergic-mediated conditions
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US20050244463A1 (en) * 2004-04-30 2005-11-03 Allergan, Inc. Sustained release intraocular implants and methods for treating ocular vasculopathies
PT1761266E (pt) 2004-05-25 2013-06-04 Galderma Pharma Sa Compostos, formulações, e métodos para tratamento ou prevenção de distúrbios inflamatórios da pele
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WO2006036480A1 (en) * 2004-09-24 2006-04-06 Allergan, Inc. 4-(phenylmethyl and substituted phenylmethyl)-imidazole-2-thiones acting as specific alpha2 adrenergic agonists
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JP2012517433A (ja) 2009-02-06 2012-08-02 アラーガン インコーポレイテッド アルファ2bおよび/またはアルファ2cアドレナリンレセプターのサブタイプ選択的モジュレーターとしてのピリジン化合物
ES2733905T3 (es) * 2009-02-13 2019-12-03 Allergan Inc Composiciones farmacéuticas que comprenden (3-(1-(1H-imidazol-4-il)etil)-2-metilfenil)metanol
US8394800B2 (en) * 2009-11-19 2013-03-12 Galderma Laboratories, L.P. Method for treating psoriasis
US8653123B2 (en) * 2010-09-16 2014-02-18 Allergan, Inc. Ester pro-drugs of [3-(1-(1H-imidazol-4-yl)ethyl)-2-methylphenyl] methanol for treating retinal diseases

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